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N-ethyl-1-[(3-methoxyphenyl)methyl]-5-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-(1,2-dihydroacenaphthylene-5-carbonyl)-1-(1H-pyrazole-4-carbonyl)piperidine
4-(2,6-dimethylpyridin-3-yl)-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}pyrimidin-2-amine
N-(1-cyclohexyl-1H-pyrazol-5-yl)-2-[4-methyl-3-(4-methylphenyl)-1H-pyrazol-1-yl]acetamide
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(pyridin-2-yl)piperidin-3-yl]propanoic acid
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-methoxyethyl)-N-(propan-2-yl)acetamide
N-{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}cyclobutanamine
2-{1-methyl-4-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperazin-2-yl}ethan-1-ol
3-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-2,6,6-trimethyl-1-propyl-4,5,6,7-tetrahydro-1H-indol-4-one
1-(4-cyclopentyl-1,4-diazepan-1-yl)-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butan-1-one
N-(2-hydroxyethyl)-1-[(1s,4s)-4-{[(4-methoxy-2,3-dimethylphenyl)methyl]amino}cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
4-(3-{[1-(3-methylthiophene-2-carbonyl)piperidin-4-yl]oxy}benzoyl)morpholine
2-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-4-{3-[4-(2,3-dimethylphenyl)piperazine-1-carbonyl]piperidin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
2-(4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carbonyl}piperazin-1-yl)-4-methoxypyrimidine
5-fluoro-2-[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]-1H-indole
N4-[(2-ethoxy-3-methoxyphenyl)methyl]-N4-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
3-[4-methyl-2-(oxolan-2-ylmethyl)phenyl]-1,3-oxazolidin-2-one
2-(4-methylphenyl)-1-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
methyl (1R,3S,3aR,6aS)-3-[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
2,3-dimethyl-7-[(3-methylthiophen-2-yl)sulfonyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
N-(4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-4-oxobutyl)acetamide
2-[4-(3-methoxy-5-methylthiophene-2-carbonyl)morpholin-3-yl]-N-(pyridin-3-ylmethyl)acetamide
9-(propane-1-sulfonyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
(1S,5R)-3-methyl-6-{[2-(trifluoromethyl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonane
[(1,3-dimethyl-1H-pyrazol-5-yl)methyl](ethyl){[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}amine
1-[(4-fluorophenyl)methyl]-5-(2-methoxyacetamido)-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
methyl 1-[6,7-dimethoxy-2-(thiomorpholin-4-ylmethyl)quinazolin-4-yl]piperidine-4-carboxylate
N-({2-[2-(2,5-dimethylfuran-3-amido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-1,3-thiazole-4-carboxamide
N-[(2S)-1-(2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-1-oxopropan-2-yl]acetamide
(3S,4R)-1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-4-(3-methylthiophen-2-yl)piperidin-3-ol
(4aS,7aR)-1-(2-methylfuran-3-carbonyl)-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N,N-dimethyl-2-[methyl(2-{[4-(trifluoromethyl)pyridin-2-yl]oxy}hex-5-en-1-yl)amino]acetamide
3-[(2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]-4H-chromen-4-one
1-[3-(2-methoxyphenoxy)azetidin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
5-(6-methoxypyridin-3-yl)-4-(4-methylphenyl)-2-(4-methylpiperazin-1-yl)pyrimidine
{1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-3-[(2-methylphenyl)methyl]piperidin-3-yl}methanol
2-({methyl[(5-phenyl-1,2-oxazol-3-yl)methyl]amino}methyl)pyridine-3-carboxylic acid
N'-(3-chloro-2-methylphenyl)-N-(1,2-oxazol-3-ylmethyl)butanediamide
2-[4-(3-chloropyridin-2-yl)-1-[(4-ethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
2-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-4-carboxylic acid
(1S,6R)-9-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
N-[(2R,3R)-2-(prop-2-en-1-yloxy)-1'-[4-(trifluoromethyl)benzoyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]cyclopropanecarboxamide
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N,5-dimethyl-1H-indazole-3-carboxamide
3-hexyl-8-[2-(pyridin-3-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}-4-(methoxymethyl)piperidine
(3aS,7aR)-5-methyl-2-[3-(1H-pyrazol-4-yl)propanoyl]-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
[(5-tert-butyl-1H-pyrazol-3-yl)methyl][2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]methylamine
2-amino-4-(2-ethoxyphenyl)-6-(pyridin-2-ylmethyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
8-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one