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(4aS,7aR)-1-(3-chloro-4-methylbenzoyl)-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-[4-(propan-2-yl)morpholin-2-yl]ethan-1-one
2-(morpholin-2-yl)-1-{4-[3-(trifluoromethyl)phenoxy]piperidin-1-yl}ethan-1-one
ethyl 3-[(3-chlorophenyl)methyl]-1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)piperidine-3-carboxylate
N-{2-chloro-4-[2-(pyridin-2-yl)acetamido]phenyl}propanamide
7-methyl-11-(trimethylpyrimidin-4-yl)-3,7,11-triazaspiro[5.6]dodecane
(1R,5R)-6-[(6-methylpyridin-2-yl)methyl]-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-[(1-methyl-1H-pyrazol-4-yl)methyl]-5-(2-phenylethyl)-5-(piperidin-4-yl)imidazolidine-2,4-dione
1-cyclobutanecarbonyl-4-(3-phenoxyazetidine-1-carbonyl)piperidine
1-(cyclopropylmethyl)-N-[3-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
2-(1H-1,3-benzodiazol-1-yl)-1-[1-(6-methylpyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]ethan-1-one
N-(6-chloro-2-methylpyridin-3-yl)-2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine-1-carboxamide
N-{1-[1-(3-methylbutyl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide
N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}-2-(1H-1,2,4-triazol-1-yl)propanamide
(5S,9aS,9bS)-5-[4-(dimethylamino)phenyl]-2-(2-phenylethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-(benzenesulfonyl)-4-{imidazo[1,2-a]pyridine-6-carbonyl}piperazine
1-(2H-1,3-benzodioxol-5-ylmethyl)-3-(methoxymethyl)pyrrolidine
3-[(3S,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[3-(trifluoromethyl)phenyl]urea
2-[5-({methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}methyl)furan-2-yl]benzonitrile
N-[(3S,5S)-5-(diethylcarbamoyl)-1-(1H-imidazol-4-ylmethyl)pyrrolidin-3-yl]pyrazine-2-carboxamide
N-ethyl-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-2,6-dimethylpyrimidine-4-carboxamide
2,3-dimethoxy-N-[(3S)-2-oxoazepan-3-yl]-N-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}benzamide
(3R,9aR)-3-benzyl-8-(2,3-difluorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(2R,6S)-4-{1-[(5-chlorothiophen-2-yl)methyl]piperidin-4-yl}-2,6-dimethylmorpholine
N-[(4-fluorophenyl)(pyridin-4-yl)methyl]-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}acetamide
2-[1-(7-methyl-1-benzofuran-2-carbonyl)azetidin-3-yl]pyridine
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2,3-dimethylquinoxaline-6-carboxamide
(3S,4S)-4-[(4-cyclobutyl-6-methylpyrimidin-2-yl)amino]-1-(propan-2-yl)pyrrolidin-3-ol
1-(3,5-dimethylphenyl)-4-[3-(1-methylpiperidin-3-yl)propanoyl]piperazin-2-one
N-methyl-2-(4-oxo-1,4-dihydroquinolin-1-yl)-N-[1-(pyridin-3-yl)ethyl]acetamide
2-methyl-6-[3-(1-methylpiperidin-3-yl)propanoyl]-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}pyrrolidin-3-yl]methanol
N-(1-{7-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)pyridine-3-carboxamide
3-phenyl-1-[2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]piperazine
(3R,5S)-5-(morpholin-4-ylmethyl)-N-(oxolan-2-ylmethyl)-1-(2-phenylethyl)piperidine-3-carboxamide
2-(1-benzyl-1H-pyrazol-4-yl)-7-methoxy-N,N-dimethylquinoline-4-carboxamide
9-methoxy-7-oxo-3-[4-(propan-2-yloxy)benzoyl]-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-[(3-methoxyphenyl)methyl]-1-(3-methylbutyl)-8-(oxan-4-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-methyl-2-oxo-8-(quinolin-2-ylmethyl)-1,8-diazaspiro[4.5]decane-4-carboxylic acid
5-{3-[2-(1,3-benzothiazol-2-yl)pyrrolidin-1-yl]-3-oxopropyl}-5-(furan-2-ylmethyl)pyrrolidin-2-one
2-[(furan-2-ylmethyl)(methyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
1-methyl-4-{[(3R,5R)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-5-(pyrrolidine-1-carbonyl)piperidin-3-yl]methyl}piperazine
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(2-{[(3-cyclopentylpropyl)amino]methyl}-5-methoxyphenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
4-methyl-2-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenol
N-[4-({[(1-cyclohexylpiperidin-3-yl)methyl](pyridin-3-ylmethyl)amino}methyl)phenyl]acetamide
4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)-N-[2-(propan-2-yl)phenyl]piperidine-1-carboxamide
N-[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
3-(2,3-dihydro-1H-inden-2-yl)-8-[(2-hydroxy-3-methoxyphenyl)methyl]-1-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-{[3-(1H-pyrazol-5-yl)piperidin-1-yl]methyl}-2-(pyridin-2-yl)pyrimidine