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1'-[(4-fluoro-3-methylphenyl)methyl]-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
6-methyl-N-[(4-phenylmorpholin-2-yl)methyl]imidazo[1,2-a]pyridine-2-carboxamide
3-(3-chloro-1H-1,2,4-triazol-5-yl)-N-methyl-N-(quinolin-5-ylmethyl)propanamide
1-benzyl-N3-[1-(4-chlorophenyl)ethyl]-4-oxo-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
1-ethyl-8-[(9-ethyl-9H-carbazol-3-yl)methyl]-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-methyl-1-(4-methylphenyl)-4-(thiophene-3-carbonyl)piperazin-2-one
N-[(1S,2S)-2-[(4-fluorophenyl)methyl]cyclopentyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
N-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-[4-(4-{[methyl(quinolin-6-ylmethyl)amino]methyl}phenoxy)piperidin-1-yl]-2-[3-(trifluoromethyl)phenyl]ethan-1-one
3-[4-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]quinoline
5-{1-[2-(3-fluorophenyl)acetyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-(pyridin-3-yl)imidazolidine-2,4-dione
(2S,4R)-N-ethyl-4-{[(9-ethyl-9H-carbazol-3-yl)methyl]amino}-1-(2-methylpropyl)pyrrolidine-2-carboxamide
N-[2-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]oxolane-3-carboxamide
1-{2-[2-(dimethylamino)ethyl]piperidin-1-yl}-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
methyl 3-(naphthalen-1-ylmethyl)-7-oxo-9-[3-(pyridin-3-yl)propoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-[1-(propan-2-yl)piperidin-4-yl]-1-{4-[2-(1H-pyrrol-1-yl)ethyl]piperazin-1-yl}ethan-1-one
2-chloro-N-{2-[(6-fluoro-2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)formamido]ethyl}benzamide
1-(1-cycloheptyl-1H-1,2,3-triazole-4-carbonyl)-4-[(2-methylphenyl)sulfanyl]piperidine
[(4-methanesulfonylmorpholin-2-yl)methyl]({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amine
3-{[(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-4-yl)oxy]methyl}pyridine
5-{1-[5-(2-methylpropyl)-1,2-oxazole-3-carbonyl]piperidin-4-yl}-5-(2-phenylethyl)imidazolidine-2,4-dione
6-(2,5-dimethylphenyl)-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-{[5-(1H-1,3-benzodiazol-1-ylmethyl)-1H-pyrazol-3-yl]formamido}-N-ethylpropanamide
N-benzyl-2-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}acetamide
(2S,4S)-4-(4-{2-[(2-methoxyphenyl)formamido]propan-2-yl}-1H-1,2,3-triazol-1-yl)-N-methylpyrrolidine-2-carboxamide
5-[(1-benzylpiperidin-4-yl)amino]-1-methyl-N-[(5-methylfuran-2-yl)methyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-{6-oxa-9-azaspiro[4.5]decane-9-carbonyl}-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-[(3-methyl-1H-pyrazol-5-yl)methyl]piperazin-2-yl}ethan-1-ol
N-{1-[(3-fluorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-2-(pyridin-4-ylsulfanyl)acetamide
(1-{5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyridin-2-yl}pyrrolidin-3-yl)methanol
6-(thiophen-3-yl)-9H-purin-2-amine
4-ethyl-5-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-1,3-thiazol-2-amine
(4aS,8aR)-6-(2,4-dimethylpyrimidine-5-carbonyl)-1-(3-hydroxypropyl)-decahydro-1,6-naphthyridin-2-one
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-(pyridin-3-yl)pyridine-3-carboxamide
N-ethyl-4-(4-methoxyphenyl)-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-4-oxobutanamide
3-fluoro-5-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
N-benzyl-N,1-dimethyl-5-{[2-(pyridin-2-yl)ethyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-{4-[3-(2,6-dimethylphenoxy)azetidin-1-yl]pyridine-2-carbonyl}morpholine
1-(oxolane-2-carbonyl)-4-{1H-pyrrolo[2,3-b]pyridin-6-yl}piperazine
4-({[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)-2-methylbutan-2-ol
4-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)-N-methyl-1,3-thiazol-2-amine
(2S,4S)-4-amino-N-methyl-1-[2-(pyridin-4-yl)ethanesulfonyl]pyrrolidine-2-carboxamide
N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
N-({7-[(2S)-2-acetamido-4-methylpentanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(methylsulfanyl)benzamide
4-(4-{[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl)benzamide
3-[3-(dimethylamino)propyl]-8-[(3-hydroxyphenyl)methyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{2-[7-(quinolin-6-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}cyclobutanecarboxamide
1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-N-(4-fluorophenyl)piperazine-2-carboxamide
N-[(3-methylphenyl)methyl]-6-oxo-1-(2-phenylethyl)piperidine-3-carboxamide
N-[2-(3-methoxyphenyl)phenyl]-1-[(4-methylphenyl)methyl]piperidine-4-carboxamide