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1-{3-[(dimethylsulfamoyl)amino]phenyl}-3-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]urea
1-{3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
1-cyclopropyl-4-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]pyrrolidin-2-one
1-(4-methyl-1H-imidazole-2-carbonyl)-3-{[4-(pyrrolidin-1-ylmethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
2-(dimethylamino)-2-(4-fluorophenyl)-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]acetamide
N-{1-[1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperidin-4-yl]-2-phenylethyl}-N-methyl-2-(1H-pyrazol-1-yl)acetamide
(2R,6R)-4-[3-(1-methylpiperidin-4-yl)propanoyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
5-{4-[(4-fluorophenyl)methyl]piperidine-1-carbonyl}-N,4-dimethyl-1,3-thiazol-2-amine
N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
4-(4-{1-[3-(trifluoromethyl)phenyl]-1H-imidazol-2-yl}-1H-1,2,3-triazol-1-yl)piperidine
3-[(3-ethoxyphenyl)methyl]-9-methoxy-N-methyl-7-oxo-N-(1,3-thiazol-4-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
4-[4-(cyclohexylmethyl)-1H-1,2,3-triazol-1-yl]-1-(1H-imidazole-4-carbonyl)piperidine
N-{[5-chloro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-(morpholin-4-yl)cyclohexane-1-carboxamide
1-[(2-methoxypyrimidin-5-yl)methyl]spiro[azepane-4,2'-chromene]
4-cyclopropyl-1-[(3,4-dimethoxypyridin-2-yl)methyl]-4-methylpyrrolidin-2-one
5-{[3-cyclopropyl-1-(1,1-dioxo-1λ6-thiolan-3-yl)-1H-1,2,4-triazol-5-yl]methyl}-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[(5-methylfuran-2-yl)methyl]amine
(3aS,6aS)-2-[2-(1H-1,2,4-triazol-1-yl)benzoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(4-ethoxyphenyl)-1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
1-{1-[2-(2-ethoxyethoxy)benzoyl]piperidin-4-yl}piperidin-3-ol
N-[3-(1H-imidazol-1-yl)propyl]-3-(1H-indol-2-ylmethyl)-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
[4-({4-[2-(1H-pyrazol-1-ylmethyl)phenyl]-1H-1,2,3-triazol-1-yl}methyl)phenyl]methanol
2-(2-{imidazo[2,1-b][1,3]thiazol-6-ylformamido}ethyl)-4-methyl-1,3-thiazole-5-carboxylic acid
N-(4-methoxy-2-methylphenyl)-3-(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-3-yl)propanamide
1-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}cyclopropane-1-carboxamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-5-(2,4-dimethoxyphenyl)-N-methyl-1,2,4-triazin-3-amine
2-[1-butyl-3-(ethoxymethyl)-1H-1,2,4-triazol-5-yl]-1-methylazepane
2-{4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-1-[(4-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
(4aS,7aR)-1-(2,5-dimethylfuran-3-carbonyl)-4-methanesulfonyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{1-[5-(4-methoxyphenyl)furan-2-carbonyl]piperidin-2-yl}pyridine
N-cyclopropyl-N-{[4-methoxy-3-(pyridin-4-ylmethoxy)phenyl]methyl}oxolane-2-carboxamide
methyl 3-[1-(4-chlorophenyl)cyclopropaneamido]-5-{[3-(3-methyl-1H-pyrazol-1-yl)propanamido]methyl}benzoate
methyl 1-[6-(2-methylphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]piperidine-4-carboxylate
6-{1-[3-(1H-1,3-benzodiazol-1-yl)propanoyl]piperidin-3-yl}-3,4-dihydropyrimidin-4-one
1-{4-[(1,3-dihydroxypropan-2-yl)amino]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]-4-sulfamoylbutanamide
1-[(4aS,8aR)-1-[3-(methylsulfanyl)propyl]-2-oxo-decahydro-1,6-naphthyridine-6-carbonyl]cyclopropane-1-carbonitrile
1-butyl-3-(thiophen-2-ylmethyl)-5-(1H-1,2,3-triazol-5-yl)-1H-1,2,4-triazole
N-(3-hydroxypropyl)-1-{1-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
3-(2-ethoxypropyl)-3-methyl-1-(quinolin-6-yl)urea
N-{[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}-4-sulfamoylbenzamide
2-[1-(2,6-dimethylquinoline-4-carbonyl)-3-oxopiperazin-2-yl]-N-methylacetamide
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-(5-oxo-5-phenylpentanoyl)pyrrolidin-3-yl]acetamide
2,4-dimethyl-N-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]pyrimidine-5-carboxamide
2-[2-({[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl](methyl)carbamoyl}amino)phenyl]-N,N-dimethylacetamide
1,3-dimethyl-N-(1,2-oxazol-5-ylmethyl)-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
ethyl 1-[(3-methyl-1H-pyrazol-5-yl)methyl]-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylate
1-[5-(3,4-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]-4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridine
2-[1-cyclopentyl-3-(2-fluorophenyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-{[2-(trifluoromethyl)phenyl]methyl}acetamide
4-[1-(pyridine-3-sulfonyl)azetidin-3-yl]pyridine