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2-methyl-N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
2-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]phenol
3-(1-benzylpyrrolidin-3-yl)-1-(5-methanesulfonyl-2-methylphenyl)urea
5-chloro-N-[2-(2-hydroxyethoxy)ethyl]-7-methoxy-1-benzofuran-2-carboxamide
2-(dimethyl-1,2-oxazol-4-yl)-N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)acetamide
3-(dimethyl-1,2-oxazol-4-yl)-1-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
N-cyclopropyl-5-(2,3-dihydro-1-benzofuran-2-carbonyl)-1-[2-(4-methoxyphenyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-ethyl-N-{[7-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)butanamide
{1-[(1-ethyl-1H-pyrazol-3-yl)methyl]-3-propylpiperidin-3-yl}methanol
1-(but-2-yn-1-yl)-4-(1-butyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridine
4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-(pent-2-yn-1-yl)piperidine
4,7-dimethyl-2-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]quinazoline
1-(dimethylamino)-2-{4-[(2,5-dimethylphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}propan-2-ol
(3S,4S)-4-methyl-1-[1-(pyridine-2-carbonyl)piperidin-4-yl]piperidine-3,4-diol
2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]-4-(trimethylpyrimidin-4-yl)morpholine
(3R,4R)-3-cyclobutyl-1-(3,4-dihydro-2H-1-benzopyran-6-carbonyl)-4-methylpyrrolidin-3-ol
5-[1-(2-methyl-1,3-benzothiazole-5-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
6-(3-methoxyphenyl)-N-methyl-N-(pyridin-3-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-(piperidin-1-yl)-1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperidine-4-carboxamide
1-[(2E)-3-phenylprop-2-en-1-yl]-4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazole
1-{3-[3-(2,6-dimethylphenoxy)azetidin-1-yl]-3-oxopropyl}-1,2-dihydropyridin-2-one
N-cyclopropyl-N-({4-[3-(dimethylamino)propoxy]phenyl}methyl)-3-methylthiophene-2-carboxamide
N-[2-(1H-pyrazol-1-yl)ethyl]-3-(thiomorpholine-4-sulfonyl)benzamide
1-{7-[(4-acetylpiperazin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-(2-chlorophenoxy)ethan-1-one
(1r,4r)-4-({[2-(2-methoxyphenyl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}amino)cyclohexan-1-ol
1-[(5-methylthiophen-2-yl)methyl]-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
8-[2-(benzenesulfonyl)ethyl]-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
N-cyclopropyl-N-({3-[(2-fluorophenyl)methoxy]phenyl}methyl)-3-methylthiophene-2-carboxamide
1-{1-[(3-methylquinoxalin-2-yl)methyl]piperidin-3-yl}-2-phenylethan-1-one
ethyl 2-[({imidazo[1,2-a]pyridin-3-ylmethyl}(methyl)amino)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxylate
2-(4-{5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-6-yl}piperidin-1-yl)pyridine-3-carbonitrile
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-benzyl-N,N-dimethylpyrrolidine-2-carboxamide
7-[(2,4-dimethylphenyl)methyl]-3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
4-[1-(5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carbonyl)piperidin-4-yl]morpholine
N-{3-[4-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)piperidin-1-yl]phenyl}pyridine-4-carboxamide
{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}[(3,5-dimethoxyphenyl)methyl]amine
1-[(4aR,8aR)-6-(thiophen-3-ylmethyl)-decahydro-1,6-naphthyridin-1-yl]-2-(4-chlorophenoxy)ethan-1-one
methyl 5-[(4-hydroxy-4-methylpentan-2-yl)amino]-3-(4-methoxybenzamido)-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
ethyl 5-[2-(cyclohex-1-en-1-yl)acetyl]-1-(2-methoxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-{1-[1-(4-chlorophenyl)-3-hydroxypropan-2-yl]-1H-1,2,3-triazol-4-yl}benzonitrile
N-(2-chloropyridin-3-yl)-4,4-difluoropiperidine-1-carboxamide
1,3-dimethyl-N,N-bis(pyridin-4-ylmethyl)-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
methyl 3-({7-oxo-4-[(2E)-3-(thiophen-2-yl)prop-2-enoyl]-1,4-diazepan-1-yl}methyl)benzoate
4-{[4-(3,4-dimethylphenoxy)phenyl]methyl}piperazine-1-sulfonamide
N-[2-(dimethylamino)ethyl]-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)-3-(1H-pyrazol-1-yl)propanamide
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-2,7-dimethylimidazo[1,2-a]pyridine-3-carboxamide
1-(azepan-1-yl)-3-[3-({[2-(pyridin-4-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
1-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-2-(2-methoxyphenoxy)ethan-1-one
N-ethyl-N-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-1,2,5-oxadiazole-3-carboxamide
[(2-butyl-1H-imidazol-4-yl)methyl]({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(2-methoxyethyl)amine