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ethyl 1-[(4-methoxyphenyl)methyl]-5-(5-oxopyrrolidine-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-(2-fluorophenyl)-1-[4-(pyrrolidine-1-sulfonyl)-1,4-diazepan-1-yl]ethan-1-one
5-butyl-4-(1,2-oxazole-3-carbonyl)-1-(3-phenylphenyl)piperazin-2-one
(3aS,6aR)-5-[(3-ethenylphenyl)methyl]-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N,6-dimethyl-N-[3-(oxolan-2-yl)propyl]imidazo[1,2-a]pyridine-2-carboxamide
2-ethyl-N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-4-methyl-1,3-thiazole-5-carboxamide
1-(4-{[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}piperidin-1-yl)ethan-1-one
2-(2-ethyl-1H-imidazol-1-yl)-1-[(3R,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]ethan-1-one
2-amino-4-(4-hydroxy-2-methoxyphenyl)-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
4-(4-ethoxy-3-methylphenyl)-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-4-oxobutanamide
{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[1-(4-methyl-1,3-thiazol-2-yl)ethyl]amine
4-(1,3-benzothiazol-2-yl)-2-({[2-(3-chlorophenyl)ethyl]amino}methyl)phenol
2-[2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-methylacetamido]acetic acid
3-cyano-N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylbenzamide
5-(2,4-dimethoxypyrimidin-5-yl)-2,3-dihydro-1H-inden-1-one
5-[4-(benzyloxy)piperidine-1-carbonyl]-1-[(3-methoxyphenyl)methyl]piperidin-2-one
2-[(2-ethoxyphenyl)methyl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-(1,3-dimethyl-1H-pyrazol-4-yl)-3-({methyl[(2-methylphenyl)methyl]amino}methyl)benzamide
4-(2,4-dimethoxybenzoyl)-2-(2-phenylethyl)morpholine
N-[2-(1H-pyrazol-4-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-[1-cyclopentyl-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carbonyl]-1-phenylpiperazin-2-one
4-methoxy-N-(2-{7-[(4-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
propan-2-yl 2-cyclopropyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecane-9-carboxylate
(3aR,6aR)-2-cyclopentyl-N-[2-(4-hydroxypiperidin-1-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
5-[(3-hydroxypiperidin-1-yl)methyl]-N-[2-(2-methylphenyl)ethyl]-1,2-oxazole-3-carboxamide
4-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(2-{[benzyl(methyl)amino]methyl}phenoxy)-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]acetamide
3-(3-fluorophenyl)-3-{2-oxo-2-[4-(propan-2-yl)piperazin-1-yl]ethyl}-1-(pyridin-3-ylmethyl)pyrrolidine-2,5-dione
2-({[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}(oxolan-2-ylmethyl)amino)acetamide
6-ethyl-N2,N2,N4-trimethyl-N4-(1H-pyrazol-5-ylmethyl)pyrimidine-2,4-diamine
1-[(3,4-difluorophenyl)methyl]-3-[(dimethylamino)methyl]-3-hydroxypiperidin-2-one
4,4-difluoro-N-(trimethyl-1H-pyrazol-4-yl)piperidine-1-carboxamide
2-oxo-8-[2-(thiophen-3-yl)acetyl]-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-(1,2-benzoxazol-3-yl)-N-{1-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
5-[1-(3-chlorothiophene-2-carbonyl)piperidin-4-yl]-5-ethyl-3-(2-methylprop-2-en-1-yl)imidazolidine-2,4-dione
4-fluoro-N-(2-{7-[(4-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
6-methyl-5-(5-{6-[2-(pyrrolidin-1-yl)ethyl]pyridin-3-yl}-1,2,4-oxadiazol-3-yl)-1,2,3,4-tetrahydro-2,7-naphthyridine
3-[2-(dimethylamino)ethyl]-5-(1-{2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl}piperidin-4-yl)-5-(3-methylbutyl)imidazolidine-2,4-dione
methyl (2S,4R)-1-methyl-4-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzamido]pyrrolidine-2-carboxylate
N-(2-methoxyethyl)-2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
3-{1-[(3-ethyl-1,2-oxazol-5-yl)methyl]piperidin-4-yl}-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
(3S,4R)-1-{[3-(2-aminoethyl)phenyl]methyl}-4-(2H-1,3-benzodioxol-5-yl)pyrrolidine-3-carboxylic acid
N-cyclopropyl-3-[1-(2-{[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}acetyl)piperidin-4-yl]propanamide
2,5-dichloro-N-{2-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-oxoethyl}benzamide
N-[(1S)-2-hydroxy-1-phenylethyl]-3-[(2-methylprop-2-en-1-yl)oxy]benzamide
1-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]-1H-imidazole-4-sulfonamide
2-[2-(1H-imidazol-4-yl)ethyl]-8-(4-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
5-amino-N-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-4-phenyl-1H-pyrazole-3-carboxamide
2-(1,2-benzoxazol-3-yl)-N-{[3-(pyrazin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}acetamide