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9-[(3,5-difluorophenyl)methyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-[5-amino-3-(furan-2-yl)-1H-1,2,4-triazol-1-yl]-5-[(propan-2-yl)sulfamoyl]benzoic acid
3-(2-methylpropyl)-N-{[1-(pyridin-2-yl)piperidin-3-yl]methyl}-1,2-oxazole-5-carboxamide
2-{1-[1-methyl-3-(thiophen-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-yl}benzoic acid
N-ethyl-3-[2-(furan-2-yl)-2-oxoacetamido]-N-phenylbenzamide
2-(2-{[1-(furan-2-ylmethyl)piperidin-3-yl]formamido}ethyl)-4-methyl-1,3-thiazole-5-carboxylic acid
2-{4-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-1-(thiophen-3-ylmethyl)piperazin-2-yl}ethan-1-ol
N-[2-hydroxy-3-(3-methoxyphenoxy)propyl]-5-methyl-4-{[2-(pyridin-2-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
5-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-3,4-dihydropyrimidin-4-one
2-{2-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoethyl}cyclopentan-1-one
3-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1-{3-[(trifluoromethyl)sulfanyl]phenyl}urea
3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}-3-{[(pyridin-4-ylmethyl)amino]methyl}piperidin-2-one
N-[3-(azepan-1-yl)propyl]-5-fluoro-N-methylquinazolin-4-amine
3-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-1-{[1,2,4]triazolo[4,3-a]pyridin-8-yl}urea
2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}-N-(propan-2-yl)acetamide
4-[(1-ethyl-1H-pyrazol-3-yl)methyl]-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
1-[2-(1H-imidazol-1-yl)-1-phenylethyl]-2-(2-methoxyphenyl)-1H-imidazole
N-benzyl-4-oxo-N-(1,3-thiazol-2-ylmethyl)-1,4-dihydroquinoline-2-carboxamide
N-[4-({4-[2-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)phenyl]acetamide
(3aS,6aS)-5-{[3-(4-methoxyphenoxy)phenyl]methyl}-1-methyl-octahydropyrrolo[3,4-b]pyrrole
N-(2,4-dimethoxyphenyl)-3-[2-(pyridin-3-yl)piperidin-1-yl]propanamide
5-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-N-methylpyrimidin-2-amine
N-methyl-5-[(4-methylpiperazin-1-yl)methyl]-N-{[3-(methylsulfanyl)phenyl]methyl}furan-2-carboxamide
2-[5-(1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}piperidin-4-yl)-1H-pyrazol-3-yl]acetic acid
N-({3-methyl-7-[2-(pyrimidin-2-ylsulfanyl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(methylsulfanyl)benzamide
3-{2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-2-oxoethyl}-2,3-dihydro-1H-isoindol-1-one
2-acetyl-8-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-(8-methoxy-2-methylquinolin-5-yl)-1-methyl-6-(thiolan-3-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-[(4aR,8aR)-6-(3-methoxybenzoyl)-decahydro-1,6-naphthyridin-1-yl]-2-phenylethane-1,2-dione
6-(3,6-dimethyl-1-benzofuran-2-carbonyl)-2,3-dimethyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
ethyl 4-{[1-(5-propylpyrimidin-4-yl)piperidin-4-yl]amino}piperidine-1-carboxylate
N,2-dimethyl-N-(2-phenylethyl)-6-(piperidin-3-yl)pyrimidin-4-amine
1-cyclopentanecarbonyl-N-[2-(1H-imidazol-4-yl)ethyl]piperidine-4-carboxamide
3-benzyl-1-(3-methoxypropyl)-8-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(thiophen-3-yl)acetamide
6-ethyl-N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-2-methylquinoline-4-carboxamide
1-{2-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-5-(trifluoromethyl)-1,2-dihydropyridin-2-one
N-[2-(3-methoxyphenyl)ethyl]-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl](ethyl)[(3-methyl-1,2-oxazol-5-yl)methyl]amine
3-(1-butyl-1H-imidazol-2-yl)-1-(2,4-dimethylbenzoyl)piperidine
3-(1H-1,3-benzodiazol-1-yl)-1-{3-[benzyl(methyl)amino]piperidin-1-yl}propan-1-one
methyl 3-[(naphthalen-1-ylformamido)methyl]-5-[2-(1H-pyrazol-1-yl)acetamido]benzoate
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
N-[(3S,5S)-5-(diethylcarbamoyl)-1-propylpyrrolidin-3-yl]-6-(methoxymethyl)pyridine-2-carboxamide
1-[(4aR,8aR)-7-[(4-chloro-2-fluorophenyl)methyl]-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]ethan-1-one
3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-1-(furan-3-ylmethyl)-1-methylurea
[3-(2-methylpropyl)-1-{[(1s,4s)-4-aminocyclohexyl]methyl}piperidin-3-yl]methanol
2-(4-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperazin-1-yl)-1,3-benzothiazole
(2-phenylethyl)({[6-(thiophen-3-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl})amine
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[4-(3-phenylpropyl)piperidin-1-yl]ethan-1-one