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3-(6-chloropyridazin-3-yl)-3,9-diazaspiro[5.5]undecane
1-(thiophene-3-carbonyl)-3-[3-(trifluoromethyl)benzoyl]piperidine
N-(morpholin-2-ylmethyl)-5-(propan-2-yl)-1,3-oxazole-4-carboxamide
3-[2-fluoro-3-(pyrrolidin-1-ylmethyl)phenoxy]-6-methylpyridazine
(2S,4R)-1-[(2-chlorophenyl)methyl]-4-(cyclooctylamino)-N,N-diethylpyrrolidine-2-carboxamide
methyl 2-[3-oxo-1-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)piperazin-2-yl]acetate
N,2,5-trimethyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
N-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-N-methylthian-4-amine
methyl[2-methyl-3-(pyrrolidin-1-yl)propyl]{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}amine
6-methyl-5-({4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}methyl)quinoline
1-{3-[3-(morpholin-4-yl)-3-oxopropyl]piperidin-1-yl}-5-phenylpentan-1-one
methyl 5-[(4-methylpentan-2-yl)amino]-3-(oxolane-2-amido)-1-(2-phenylethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-{[7-(3-cyclopentylpropanoyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}oxolane-3-carboxamide
1-(2-methylquinolin-8-yl)-3-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}urea
N3-{2-[(2-butyl-6-methylpyrimidin-4-yl)amino]ethyl}piperidine-1,3-dicarboxamide
2-cyclopropanecarbonyl-8-(4-fluorobenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-fluoro-N-[(1-{imidazo[1,2-a]pyridine-2-carbonyl}piperidin-3-yl)methyl]benzamide
1-(2-aminoethyl)-N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-[3-(1H-indol-2-yl)phenyl]-1-(pyridin-2-ylmethyl)piperidine-4-carboxamide
N-(1-{2-[cyclohexyl(methyl)amino]-4-methylpyrimidin-5-yl}ethyl)-2-(2,5-dioxoimidazolidin-1-yl)acetamide
N-cyclohexyl-4-(3-ethyl-4-methyl-1H-pyrazole-5-amido)piperidine-1-carboxamide
(1S,5R)-3-[(2-fluoro-4-methylphenyl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(1S,5R)-3-(1-benzofuran-5-ylmethyl)-6-methyl-3,6-diazabicyclo[3.2.2]nonane
N-{5-[4-(1,3-benzothiazol-2-yl)piperazine-1-carbonyl]-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl}propanamide
N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-4-(1H-pyrazol-3-yl)benzamide
5-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid
4-acetyl-N-[3-methoxy-5-(trifluoromethyl)phenyl]-1,4-diazepane-1-carboxamide
2-[1-(2-phenylethyl)-4-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl]ethan-1-ol
4-(2-{4-[3-(4-methylphenoxymethyl)piperidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}ethyl)morpholine
2-{[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]methyl}-N-[(4-methylphenyl)methyl]quinazolin-4-amine
{3-[(2,4-difluorophenyl)methyl]-1-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}methanol
1-cyclohexyl-N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
N-(2-methoxyethyl)-1-methyl-N-{2-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-amine
N-[(3S,4R)-1-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-4-propylpyrrolidin-3-yl]acetamide
2-(1H-1,3-benzodiazol-1-yl)benzamide
5-[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-4-yl]-5-propyl-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
3-phenoxy-N-(1-{1-[2-(pyridin-3-yl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)propanamide
5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-[(5-methyl-1,2-oxazol-3-yl)methyl]pyridin-2-amine
4-[(dipropylamino)methyl]-N-(oxolan-2-ylmethyl)benzamide
4-(1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-3-yl)pyrimidine
N-{[5-chloro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-(methylsulfanyl)benzamide
1-ethyl-N-[(2-fluorophenyl)methyl]-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(3-fluorophenyl)-N-[1-(3-methylbutyl)-1H-pyrazol-5-yl]-3-oxopiperazine-1-carboxamide
[(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl)methyl](methyl)(2-methylpropyl)amine
N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-4-hydroxy-2-(3-methylphenyl)pyrimidine-5-carboxamide
ethyl 4-{3-[(3,4-dimethoxyphenyl)amino]piperidin-1-yl}piperidine-1-carboxylate
2-(3-hydroxypropyl)-8-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
1-[4-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)piperidin-1-yl]ethan-1-one
N-[(3S,4R)-1-{[4-chloro-2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
N-(1-{1-[1-(4-methoxyphenyl)cyclopentanecarbonyl]piperidin-4-yl}-1H-pyrazol-5-yl)acetamide