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1-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one
5-(2-methoxyacetamido)-1-(2-phenylethyl)-N-[2-(pyridin-3-yloxy)propyl]-1H-1,3-benzodiazole-7-carboxamide
3-[(3R,4S)-4-(morpholin-4-yl)-1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}piperidin-3-yl]propan-1-ol
4-cyclopropanecarbonyl-6-[(3-methoxyphenyl)methoxy]-1-(2-phenylethyl)-1,4-diazepan-2-one
N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]-2-[(2-fluorophenyl)methyl]-1,3-benzoxazole-6-carboxamide
2-[3-(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)-1H-indol-1-yl]acetamide
[3-(2-phenylethyl)-1-{thieno[2,3-d]pyrimidin-4-yl}piperidin-3-yl]methanol
1-[3-(5-methylfuran-2-yl)butyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-6-(morpholine-4-carbonyl)pyrazin-2-amine
methyl 4-{4-[(1-propyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}benzoate
{[(3R,4S)-4-cyclopropyl-1-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}pyrrolidin-3-yl]sulfamoyl}dimethylamine
N-({2,3-dimethylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
N,N-dimethyl-5-{[4-(pyrrolidin-3-yl)piperazin-1-yl]methyl}pyridin-2-amine
methyl 9-[2-(2-fluorophenyl)ethoxy]-7-oxo-3-[(2E)-3-phenylprop-2-en-1-yl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-[4-(4-fluorophenyl)oxane-4-carbonyl]-3-(1-methyl-1H-imidazol-2-yl)piperidine
4-[benzyl({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amino]butan-1-ol
N-(2H-1,3-benzodioxol-5-yl)-5-{1H-pyrazolo[3,4-b]pyridin-1-yl}furan-2-carboxamide
3-ethyl-1-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidine-3-carboxylic acid
4-(2,6,8-trimethylquinoline-4-carbonyl)-1,4-oxazepan-6-ol
ethyl 2-{[(4-{3-[cyclohexyl(methyl)amino]-2-hydroxypropoxy}-3-methoxyphenyl)methyl](methyl)amino}acetate
1-[3-(2-hydroxypropan-2-yl)pyrrolidin-1-yl]-3-(pyridin-3-yl)propan-1-one
({3-[2-(4-cyclobutanecarbonylpiperazin-1-yl)ethoxy]phenyl}methyl)(methyl)(naphthalen-1-ylmethyl)amine
1-[2-(4-fluorophenyl)benzoyl]-3-(3-methoxypropyl)piperidine
2-(4-amino-1H-pyrazol-1-yl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]acetamide
(1R,5S)-N-[4-ethoxy-3-(1H-pyrrol-1-yl)phenyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
methyl 3-(2-methoxy-2-phenylacetamido)-6-{[methyl(2-methylpropyl)amino]methyl}thieno[2,3-b]pyridine-2-carboxylate
7-(3-ethyl-1,2-oxazole-5-carbonyl)-N,N-dimethyl-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-[5-(1-benzyl-1H-imidazol-5-yl)-1-methyl-1H,4H-pyrazolo[3,4-d]imidazol-3-yl]pyridine
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-{2-[4-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-oxoethyl}-4-(propan-2-yl)piperazin-2-one
N-[2-(dimethylamino)ethyl]-4-(methoxymethyl)-5-methyl-N-[(5-methylthiophen-2-yl)methyl]-1,2-oxazole-3-carboxamide
1-[(4-methoxyphenyl)methyl]-4-[2-(morpholin-2-yl)acetyl]piperazin-2-one
methyl(oxan-4-ylmethyl){[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}amine
6-[(3-fluorophenyl)methoxy]-1-(2-methylpropyl)-4-(quinoxaline-5-carbonyl)-1,4-diazepan-2-one
3-[2-(azetidin-1-yl)-2-oxoethyl]-1-benzyl-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
1-[4-(4-{[2-(4-methylphenyl)ethyl]amino}piperidin-1-yl)benzoyl]piperidin-3-ol
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(5-methoxyfuran-2-carbonyl)piperidine
N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}-2-(1-methyl-3-oxopiperazin-2-yl)acetamide
2-{4-[(3-fluoro-2-methylphenyl)methyl]morpholin-3-yl}acetic acid
5-[(2-fluorophenyl)methyl]-5-(1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)imidazolidine-2,4-dione
4-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
5-{[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]methyl}quinoxaline
{[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}[2-(piperidin-1-yl)ethyl]amine
2-(3-{[1-(4-fluoro-3-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}phenoxy)ethan-1-ol
2-{2-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethoxy}ethan-1-ol
6-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-(2-{1-[(2S)-oxolan-2-ylmethyl]-1H-imidazol-2-yl}quinolin-6-yl)acetamide
N-[(3S,5S)-1-benzyl-5-(ethylcarbamoyl)pyrrolidin-3-yl]-5-hydroxypyrazine-2-carboxamide
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-(2,3-dimethoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[2-(2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-4-(methylsulfanyl)benzamide