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3-[1-(5-acetylthiophene-3-carbonyl)piperidin-3-yl]-N-(3-chloro-4-methoxyphenyl)propanamide
4-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)-1λ6-thiane-1,1-dione
4-{2-methyl-6-[1-(pent-2-yn-1-yl)piperidin-4-yl]pyrimidin-4-yl}morpholine
3-(2H-1,3-benzodioxol-5-yl)-5-(thiomorpholine-4-sulfonyl)benzoic acid
1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
4-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-N-[2-(1-methylpyrrolidin-2-yl)ethyl]pyrimidin-2-amine
4-{1-[(4-chlorophenyl)methyl]pyrrolidin-3-yl}-1-(1-methyl-1H-pyrazole-5-carbonyl)piperidine
7-(3-chlorophenyl)-4-(cyclohex-3-ene-1-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
ethyl 1-ethyl-5-(furan-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-[5-(2-chloro-4-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]-1,2-oxazinane
propyl 8-(morpholine-4-sulfonyl)-1,2,3,4-tetrahydroisoquinoline-2-carboxylate
2-[1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)pyrrolidin-3-yl]benzoic acid
(3S,5R)-1-[2-(2-methylphenyl)acetyl]-5-(4-methylpiperazine-1-carbonyl)piperidine-3-carboxylic acid
3-[4-(2-amino-6-methylpyrimidin-4-yl)piperazine-1-carbonyl]piperidine-1-carboxamide
(3aR,6aR)-2-acetyl-5-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
6-{[4-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}quinoline
4-(furan-3-ylmethyl)-3-{2-[4-(2-methoxyphenoxy)piperidin-1-yl]-2-oxoethyl}piperazin-2-one
{[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-(1,2-oxazol-3-ylmethyl)piperidin-4-ol
N-[(4-fluorophenyl)methyl]-3-{1-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}propanamide
3-(2-amino-1,3-thiazol-4-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]propanamide
(2R)-1-{3-[(1,2-oxazol-3-ylmethyl)carbamoyl]benzenesulfonyl}pyrrolidine-2-carboxamide
N,4-dimethyl-N-{2-[4-({methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)phenoxy]ethyl}benzamide
6-methyl-2-{[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonan-3-yl]methyl}quinolin-4-ol
5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]-2-(pyridin-3-yl)pyridine
N-methyl-4-oxo-N-(pyridin-2-ylmethyl)-3,4-dihydrophthalazine-1-carboxamide
[(3S,5R)-5-[(dimethylamino)methyl]-1-[2-(pyridin-4-yl)-1,3-thiazole-4-carbonyl]piperidin-3-yl]methanol
1-{3-[2-(3-methoxyphenyl)ethyl]piperidin-1-yl}-3-(1,2-oxazinan-2-yl)propan-1-one
N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]-2-(pyrrolidin-1-yl)-6-(trifluoromethyl)pyrimidin-4-amine
5-(2-methylpropyl)-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
methyl 1-(2-methoxyethyl)-5-[(3-phenylbutyl)amino]-3-(3-phenylpropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}[(4-methylphenyl)(pyridin-4-yl)methyl]amine
(1S,5R)-3-(pyridin-2-ylmethyl)-6-(pyrrolidine-1-sulfonyl)-3,6-diazabicyclo[3.2.2]nonane
2-[3-({spiro[indene-1,4'-piperidine]-1'-yl}carbonyl)pyrazolo[1,5-a]pyrimidin-6-yl]ethan-1-ol
1-(cyclohexylmethyl)-N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
(2R,3R)-3-{methyl[3-(3-methylphenoxy)propyl]amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl){[5-(oxolan-2-yl)thiophen-2-yl]methyl}amine
1-(oxan-4-ylmethyl)-6-(pyridin-3-ylmethoxy)-4-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-1,4-diazepan-2-one
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2,3-difluoro-4-methoxybenzamide
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(morpholin-4-yl)benzamide
5-methyl-4-[(oxolan-2-ylmethyl)amino]-N-[(4-phenyloxan-4-yl)methyl]thieno[2,3-d]pyrimidine-6-carboxamide
1-[2-(3-fluorophenyl)ethyl]-N-(3-hydroxy-2,2-dimethylpropyl)-6-oxopiperidine-3-carboxamide
N-(6-methoxy-1,3-benzothiazol-2-yl)-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propanamide
N-(6-cyanopyridin-3-yl)-4-{[methyl(oxan-2-ylmethyl)amino]methyl}benzamide
7-(2-methoxyphenyl)-N-(2-methylphenyl)-4-oxo-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepine-2-carboxamide
1-[2-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-oxoethyl]imidazolidine-2,4-dione
(3S,4R)-4-(4-fluorophenyl)-1-(2-methanesulfonylethyl)pyrrolidine-3-carboxylic acid
N-(1-benzylpiperidin-4-yl)-1-[2-(dimethylamino)ethyl]-6-oxopiperidine-3-carboxamide
1-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-2-(4-methyl-1,4-diazepan-1-yl)ethan-1-one
1-[1-(4-fluorophenyl)piperidin-4-yl]-N-phenylpiperidin-3-amine