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N-(furan-2-ylmethyl)-N-(2-hydroxyethyl)-1-methyl-5-phenyl-1H-pyrazole-3-carboxamide
ethyl 1-[(2,3-difluorophenyl)methyl]-3-(2-methoxyethyl)piperidine-3-carboxylate
4-[3-(prop-2-en-1-yloxy)benzoyl]-7-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
N,N-diethyl-1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]piperidine-3-carboxamide
1-[2-(2-chlorophenyl)ethyl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
1-cyclopentyl-3-{2-[4-(2,4-dimethylphenyl)piperazin-1-yl]-2-oxoethyl}-3-(3-fluorophenyl)pyrrolidine-2,5-dione
(3R,4R)-N-benzyl-3-hydroxy-N,4-dimethyl-3-(propan-2-yl)pyrrolidine-1-sulfonamide
4-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-3-methyl-1-[(3-methylphenyl)methyl]piperazin-2-one
4-[(1-ethylpiperidin-4-yl)amino]-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-2-one
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]-1,4-diazepan-5-one
N-[(4-methylpyridin-2-yl)methyl]-2-(2,2,6,6-tetramethylpiperidin-4-yl)acetamide
2-[(1S,5R)-3-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
3-(methylsulfanyl)-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-1H-indole-2-carboxamide
5-[4-(adamantan-1-yl)piperazine-1-carbonyl]-1H-1,2,3-benzotriazole
3-[5-(5-acetylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]-N-methyl-N-(2-phenylethyl)propanamide
N-{4-[3-(4-{[methyl(naphthalen-1-ylmethyl)amino]methyl}phenoxymethyl)piperidine-1-carbonyl]phenyl}acetamide
2-{4-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]phenyl}acetamide
(5S,9aS,9bS)-5-[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]-2-[(5-methylfuran-2-yl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-{[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]methyl}benzonitrile
3-[({[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}amino)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-5-methylpyrimidin-2-amine
N-[(3R,4S)-1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]cyclopropanesulfonamide
3-[(dimethylamino)methyl]-1-(2-methoxypyridine-4-carbonyl)pyrrolidin-3-ol
6-(2,5-dimethylphenyl)-N-methyl-N-(oxolan-3-yl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-amino-6-methyl-N-[2-(pyridin-3-yloxy)propyl]pyrimidine-4-carboxamide
N-(5-chloro-2-methoxyphenyl)-3-{1-[3-(pyridin-4-yl)propanoyl]piperidin-3-yl}propanamide
2-[4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)piperidine-1-carbonyl]pyrazine
N-[2-(3,4-dimethylphenoxy)ethyl]-3-propyl-1H-pyrazole-5-carboxamide
2-[1-cyclopentyl-3-(2-fluorophenyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-(propan-2-yl)acetamide
1-[4-chloro-2-(trifluoromethyl)phenyl]-3-{2-[5-(hydroxymethyl)-1,2,4-oxadiazol-3-yl]ethyl}urea
2-ethyl-N-[3-(1H-1,2,3-triazol-1-yl)propyl]pyrimidine-5-carboxamide
5-{1H-pyrazolo[3,4-b]pyridin-1-yl}pyridin-2-ol
(1-{[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}-3-[(4-fluorophenyl)methyl]piperidin-3-yl)methanol
1-{4-[2-(2H-1,3-benzodioxol-5-yl)-5-fluoro-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one
N4,N4,5-trimethyl-N2-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}pyrimidine-2,4-diamine
N-{[5-(2,6-difluorophenyl)-1,2,4-oxadiazol-3-yl]methyl}-2-methylimidazo[1,2-a]pyridine-6-carboxamide
2-{[1-ethyl-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1H-indole
2-(2,5-dimethoxyphenyl)-N-[2-(dimethylamino)ethyl]-N-{[2-(4-methoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}acetamide
6-methoxy-3-[4-(piperazin-1-yl)phenyl]quinoline
1-(2H-1,3-benzodioxol-5-yl)-2-(4-methyl-1H-imidazol-5-yl)-1H-imidazole
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]pyrrolidine-3-carboxylic acid
2-[methyl({[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl})amino]acetic acid
N-(2,3-dihydro-1H-inden-2-yl)-1-propyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-(1-{7-[(4-hydroxy-2-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)methanesulfonamide
N-({1-[(4-acetamidophenyl)methyl]piperidin-3-yl}methyl)-1H-indole-2-carboxamide
N,N-diethyl-2-{[2-oxo-1-(2-phenylethyl)-4-(1,2,3-thiadiazole-4-carbonyl)-1,4-diazepan-6-yl]oxy}acetamide
2-(3-{3-[4-(dimethylamino)-5-methylpyrimidin-2-yl]phenyl}-1H-pyrazol-1-yl)-N,N-dimethylacetamide
2-{[(5-methylpyrazin-2-yl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
5-methyl-N-[3-(5-methyl-4-{[4-(1H-1,2,4-triazol-1-yl)butanamido]methyl}-1,3-oxazol-2-yl)phenyl]thiophene-2-carboxamide