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1-(4-methoxyphenyl)-6,6-dimethyl-4-(3-methylbenzoyl)piperazin-2-one
N-({7-[(4-phenyl-1,3-thiazol-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzamide
1-(2-methyl-5-propylpyrimidin-4-yl)-1,4-diazepan-5-one
2-ethyl-4-methyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-1,3-oxazole-5-carboxamide
4-{4-[(2,2-dimethylpyrrolidin-1-yl)methyl]-1H-1,2,3-triazol-1-yl}-1-(3-methylbut-2-en-1-yl)piperidine
2-(2-methyl-1,3-thiazol-4-yl)-1-[1-(pyridin-3-yl)-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl]ethan-1-one
1-[(3S,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]-2-(1H-indol-1-yl)ethan-1-one
1-[2-(naphthalen-1-ylmethyl)morpholin-4-yl]-3-(1H-pyrazol-4-yl)propan-1-one
2-cyclopropyl-N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-1,3-benzoxazole-6-carboxamide
(2,1,3-benzoxadiazol-4-ylmethyl)[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](2-methoxyethyl)amine
methyl 2-({1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazol-4-yl}formamido)-4-(methylsulfanyl)butanoate
N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carboxamide
2-(4-chloro-2-{[(3S,4S)-3-(dimethylamino)-4-hydroxypyrrolidin-1-yl]methyl}phenoxy)acetic acid
{4-[(2-chlorophenyl)methyl]-1-[(2-fluoro-5-methoxyphenyl)methyl]piperidin-4-yl}methanol
1-(3-chlorophenyl)-4-{1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carbonyl}piperazine
2-(3-hydroxyphenyl)-1-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}ethan-1-one
N-[2-methoxy-5-({[(3-methyloxetan-3-yl)methyl]carbamoyl}amino)phenyl]acetamide
(2S,4R)-4-amino-1-[(8-chloroquinolin-2-yl)methyl]-N-ethylpyrrolidine-2-carboxamide
(3S,4S)-4-(pyridin-2-yl)-1-(quinoline-8-carbonyl)pyrrolidine-3-carboxylic acid
1-{2-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-2-oxoethyl}pyrrolidin-2-one
2-(dimethyl-1,2-oxazol-4-yl)-2-{8-methoxy-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}acetic acid
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N-methyl-1-(pyrrolidin-1-yl)cyclopentane-1-carboxamide
N-[3-chloro-2-(4-ethylpiperazin-1-yl)phenyl]-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-1-[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]ethan-1-one
4-(3-fluorophenoxy)-1-[(2S)-oxolane-2-carbonyl]piperidine-4-carboxylic acid
1-{2-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
[4-(4-methoxyphenyl)butan-2-yl](methyl){2-[4-(4-methylpiperazine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}amine
N-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-chlorobenzamide
N-methyl-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
{4-[(3-methoxyphenyl)methyl]-1-(pyrimidin-2-yl)piperidin-4-yl}methanol
ethyl 3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carboxylate
1-[(2,6-difluorophenyl)methyl]-N-(3-ethoxypropyl)-1H-1,2,3-triazole-4-carboxamide
1-(3-{3-[hydroxy(phenyl)methyl]-4H-1,2,4-triazol-4-yl}phenyl)ethan-1-one
1-[(4aS,8aR)-4a-(hydroxymethyl)-decahydro-1,6-naphthyridin-6-yl]-4-(3,5-dimethyl-1H-pyrazol-1-yl)butan-1-one
2-{1-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1H-1,2,3-triazol-4-yl}quinoline
7-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-2,3-dimethyl-1H-indole
propan-2-yl 4-chloro-3-[2-(propan-2-yloxy)acetamido]benzoate
2-{1,3-dimethyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-6-ethoxyphenol
N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-5-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
4-[(2-methylphenyl)methyl]-1-[3-(1H-pyrazol-1-yl)benzoyl]-1,4-diazepan-5-one
ethyl 4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
2-[1-(1H-indole-2-carbonyl)piperidin-3-yl]-4-methyl-1H-1,3-benzodiazole
4-{[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}thiomorpholine
4-(3,3-diphenylpiperidine-1-carbonyl)-1-methylimidazolidin-2-one
(1-methyl-4-{[5-(2-methylpropyl)thiophen-2-yl]methyl}piperazin-2-yl)methanol
1-{6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carbonyl}-3-(hydroxymethyl)piperidin-3-ol
N-(2-{6-[(2-fluorophenyl)methoxy]-4-(2-methylpropyl)-3-oxo-1,4-diazepan-1-yl}-2-oxoethyl)acetamide
[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amine
3-(3-methoxybenzoyl)-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-1-[(3S)-3-ethylmorpholin-4-yl]ethan-1-one