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7-(1,3-benzothiazol-2-yl)-4-(1H-indol-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carbonyl}-4-methyl-1,2,3-thiadiazole
N-[2-(dimethylsulfamoyl)ethyl]-2-methyl-1,3-benzoxazole-6-carboxamide
5-methyl-2-(propylamino)-N-[1-(1H-1,2,4-triazol-5-yl)ethyl]benzamide
N-{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}-N,1-dimethylpiperidin-4-amine
3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-5-phenyl-1,2-oxazole
3-(cyclopropylmethyl)-5-[(4-fluorophenyl)methyl]-5-[1-(5-methylpyrazine-2-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
4-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
N-cyclopentyl-N-({4-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
3-phenyl-N-{[1-(pyridin-2-yl)piperidin-3-yl]methyl}-1H-pyrazole-4-carboxamide
4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)-1-(furan-2-carbonyl)piperidine
1-(2-ethoxyethyl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]-N-(prop-2-en-1-yl)acetamide
(4aS,7aR)-1-[(1-propyl-1H-imidazol-2-yl)methyl]-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(5-methylfuran-2-yl)methyl]piperidine
5-(2-methoxyphenoxymethyl)-N-(2-oxopyrrolidin-3-yl)-1H-pyrazole-3-carboxamide
N-{2-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]ethyl}-1-cyclohexyl-1H-1,2,3-triazole-4-carboxamide
5-(7-methoxy-2H-1,3-benzodioxol-5-yl)-1H,5H,6H,7H,8H-pyrido[3,2-f]indazol-7-one
3-{1-[2-(methylamino)-1,3-thiazole-4-carbonyl]piperidin-4-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
[(1-ethyl-1H-pyrazol-4-yl)methyl]({[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl})methylamine
4-(3-acetylbenzoyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
2-(2-methyl-1,3-thiazol-4-yl)-N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}acetamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetamide
(3S,4R)-3-benzyl-1-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-4-methylpiperidin-4-ol
5-cyclopropanecarbonyl-1'-(4,6-dimethylpyridine-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-{2-[1-(4-ethylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-oxoethyl}-1,3-thiazolidine-2,4-dione
2-[3-(2-fluorophenoxymethyl)piperidin-1-yl]-1,3-thiazole-4-carboxamide
2-(1-{[2-(butylsulfanyl)pyrimidin-5-yl]methyl}pyrrolidin-2-yl)-1H-1,3-benzodiazole
N-[(3R,4S)-4-cyclopropyl-1-(2-hydroxyethyl)pyrrolidin-3-yl]-2-methyl-5-(trifluoromethyl)benzamide
(4aS,7aR)-1-(2,1,3-benzothiadiazol-5-ylmethyl)-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[(3R,4S)-1-(4-chloro-1-methyl-1H-pyrrole-2-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
N-({2-[3-(4-methoxybenzenesulfonamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-4-methylbenzamide
4-{[(2,3-dimethoxyphenyl)methyl]amino}-N-(2-hydroxy-2-phenylethyl)-N,5-dimethylthieno[2,3-d]pyrimidine-6-carboxamide
6-[2-(6-methylpyridin-2-yl)ethyl]-5,6-dihydro-1,6-naphthyridin-5-one
N-{[1-(6-cyanopyridin-2-yl)piperidin-3-yl]methyl}-2,3-dimethoxybenzamide
2-{[1-(4-fluoro-3-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}pyridine
[1-(1H-imidazol-1-yl)propan-2-yl][(5-methoxy-1H-indol-2-yl)methyl]amine
(3R,4R)-3-cyclobutyl-4-methyl-1-(thiophene-3-carbonyl)pyrrolidin-3-ol
2-(pyridin-4-ylmethyl)-8-(pyrimidin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
(5-{[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]methyl}furan-2-yl)methanol
N-(2H-1,3-benzodioxol-5-yl)-1-[(6-methylpyridin-2-yl)methyl]piperidin-3-amine
2-amino-4-[2-(dimethylamino)pyrimidin-5-yl]-6-(4-hydroxyphenyl)-5-methylpyridine-3-carbonitrile
2-methoxy-1-(1'-{spiro[2.5]octane-1-carbonyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)ethan-1-one
3-[(1S,5S)-6-methyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-4-phenyl-1H-pyrazol-5-amine
N-{[5-methyl-2-(2-phenylmethanesulfonamidophenyl)-1,3-oxazol-4-yl]methyl}-2-(thiophen-2-yl)acetamide
1-[2-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)ethyl]-1H-1,2,3,4-tetrazole
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-[2-(1H-imidazol-1-yl)ethyl]-5-methylpiperidin-2-one
7-(3,4-dihydronaphthalen-2-yl)-4-(1H-pyrazol-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-[(4-ethoxyphenyl)methyl]-3-[2-(4-hydroxypiperidin-1-yl)-2-oxoethyl]piperazin-2-one
2-(dimethyl-1,2-oxazol-4-yl)-1-[3-(morpholine-4-carbonyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethan-1-one