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2-amino-4-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-6-(propan-2-yl)pyridine-3-carbonitrile
1-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]-4-(2-phenylethyl)piperazine
1-methyl-N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
2-amino-N-(2,1,3-benzothiadiazol-5-ylmethyl)-N,4-dimethyl-1,3-benzothiazole-6-carboxamide
N-cyclohexyl-2-(1H-imidazol-2-yl)benzamide
(1R,3S,5S)-8-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-8-azabicyclo[3.2.1]octan-3-ol
5-[4-(5-chloropyridin-2-yl)piperazine-1-carbonyl]-N-ethylpyrimidin-2-amine
N-{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}thian-4-amine
2-ethyl-4-methyl-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-1,3-thiazole-5-carboxamide
4-[5,6-dimethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-1,4-oxazepan-6-ol
1-[2-(piperidin-2-yl)ethyl]-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1H-1,2,3-triazole-4-carboxamide
2-{[(1-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-4-yl)oxy]methyl}pyridine
1-methyl-5-[3-(pentan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1H-1,2,3-benzotriazole
(2E)-3-(2-chlorophenyl)-N-{2-[4-(2-fluorophenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]ethyl}prop-2-enamide
2-methyl-4-(4-{[3-(pyrrolidin-1-yl)pyrrolidin-1-yl]methyl}phenyl)butan-2-ol
6-(benzyloxy)-1-(2-methylpropyl)-4-(pyridine-3-carbonyl)-1,4-diazepan-2-one
N-(1,4-dioxan-2-ylmethyl)-N-methyl-1-(4-methylquinazolin-2-yl)piperidine-4-carboxamide
2-[2-({[(3-methylthiophen-2-yl)methyl](pyridin-2-ylmethyl)amino}methyl)phenoxy]acetic acid
N-(3-chloro-4-fluorophenyl)-3-[1-(3-methylfuran-2-carbonyl)piperidin-4-yl]propanamide
5-(5-chloro-2-methoxyphenyl)-2-fluorobenzamide
N-[(3R,4S)-4-cyclopropyl-1-[(2-fluoro-4-methoxyphenyl)methyl]pyrrolidin-3-yl]-3-methoxypropanamide
4-(isoquinolin-1-yl)-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-(piperidin-4-yl)-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-6-phenylimidazo[2,1-b][1,3]thiazole-3-carboxamide
4-[3-(azepane-1-carbonyl)piperidin-1-yl]-2-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}piperidin-4-yl)propanamide
1-[3-(furan-2-yl)phenyl]-3-methyl-3-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)urea
(4aS,8aR)-6-(1-aminocyclopropanecarbonyl)-1-(2-phenylethyl)-decahydro-1,6-naphthyridin-2-one
3-{1-[1-(3-fluorobenzoyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}pyridine
N-{[7-(cyclopent-1-ene-1-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(thiophen-3-yl)acetamide
6-(3-fluoro-4-methoxyphenyl)-N-(3-methylbutyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
5-(1-{[4-(diethylamino)phenyl]methyl}piperidin-4-yl)-5-(2-phenylethyl)imidazolidine-2,4-dione
2-methoxy-4-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
1-[(3R,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-3-(pyridin-3-yl)propan-1-one
(1R,5R)-N-(2-methylphenyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
(1S,5R)-6-propyl-3-{2-[4-(trifluoromethyl)phenyl]acetyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
2-({1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}oxy)-4-methoxy-N-(2-methoxyethyl)benzamide
2-(6-hydroxy-1,4-oxazepan-4-yl)-N-[(2-methylphenyl)methyl]acetamide
N-(4-{[({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)amino]methyl}phenyl)acetamide
N-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]benzamide
3-(2-{1-[2-(dimethylamino)ethyl]-5-oxopyrrolidin-2-yl}ethyl)-1-[2-(propan-2-yl)phenyl]urea
N3-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-N1,N1-dimethylpiperidine-1,3-dicarboxamide
(1S,6R)-9-[2-(1,1,2,2-tetrafluoroethoxy)benzoyl]-3,9-diazabicyclo[4.2.1]nonane
8-(2,4-difluorobenzoyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
4-{1-[(2-chloro-4-fluorophenyl)methyl]piperidin-4-yl}-2-methylpyrimidine
N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-5-(1H-imidazol-1-ylmethyl)furan-2-carboxamide
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-7-fluoro-3-methyl-1-benzofuran-2-carboxamide
4-ethyl-3-({1-[2-(1H-1,2,4-triazol-1-yl)propanoyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-4-[3-(1H-pyrazol-1-yl)propyl]-1,4-diazepane
N-(pyridin-3-ylmethyl)-4-[(1S,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]pyridine-2-carboxamide