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5-[3,5-dimethyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1-(2-methanesulfonylethyl)-4-phenyl-1H-imidazole
2-fluoro-6-{[(furan-2-ylmethyl)(thiophen-3-ylmethyl)amino]methyl}phenol
8-{[3-methoxy-4-(pyrrolidin-1-yl)phenyl]methyl}-2,8-diazaspiro[4.5]decan-3-one
2-(5-ethyl-1H-pyrrole-2-carbonyl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
1-{[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(3-methoxypropyl)piperidine
4-{[4-(cyclohexylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]methyl}phenol
N-[(4-methoxyphenyl)methyl]-3-oxo-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
(2S,4R)-4-amino-N-ethyl-1-{2-[(4-methoxyphenyl)amino]-2-methylpropanoyl}pyrrolidine-2-carboxamide
1-benzyl-N,N-dimethyl-5-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(4-fluorophenyl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}methanesulfonamide
2-{4-[(1-benzyl-1H-indol-6-yl)methyl]morpholin-3-yl}acetic acid
4-[5-({spiro[indene-1,4'-piperidine]-1'-yl}carbonyl)-1H-pyrazol-3-yl]phenol
1-[4-(4-chlorophenoxy)piperidin-1-yl]-2-(methylamino)ethan-1-one
4-[3-(2-hydroxyethyl)-4-(2-methylpropyl)piperazin-1-yl]-5-methylthieno[2,3-d]pyrimidine-6-carboxylic acid
(1S,6R)-3-{[5-(4-chlorophenyl)furan-2-yl]methyl}-3,9-diazabicyclo[4.2.1]nonane
3-(3-methylbutyl)-8-[3-(morpholin-4-yl)butanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-({[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)amino)-2-methylbutan-2-ol
1-(3-cyano-4-methoxyphenyl)-3-[(2-propyl-1,3-thiazol-4-yl)methyl]urea
(2S)-2-({1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)butan-1-ol
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-(2-phenylethyl)-N-(pyridin-2-ylmethyl)acetamide
{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}[(2,3-difluorophenyl)methyl]amine
2-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidine-1-carbonyl}-N,N-dimethylaniline
1-[(2,3-difluorophenyl)methyl]-3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidine
(3S,4R)-1-(2-methoxy-5-methylbenzoyl)-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
ethyl 1-[5-(2-methoxy-4-methylphenoxymethyl)-1,2-oxazole-3-carbonyl]piperidine-2-carboxylate
4-[4-(1-ethoxyethyl)phenyl]-2-methyl-1H-imidazole
3-chloro-5-[1-(cyclohexylmethyl)-3-(furan-2-yl)-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
2-(1H-pyrazol-1-yl)-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]benzamide
4-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)-3-(4-fluorophenyl)piperazin-2-one
1-{4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidine-1-carbonyl]phenyl}-3,5-dimethyl-1H-pyrazole
N-({3,5-dimethoxy-4-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]-2-(1H-pyrazol-1-yl)acetamide
{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}[2-(1H-imidazol-4-yl)ethyl]amine
1-[3-(4-methylphenoxymethyl)piperidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
1-(4-ethylpiperazin-1-yl)-3-{1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-4-yl}propan-1-one
N-[2-({3-[(2-methylphenyl)sulfamoyl]-5-[(naphthalen-2-ylmethyl)amino]phenyl}formamido)ethyl]acetamide
(1S,5R)-6-(2,5-dimethoxybenzoyl)-3-methyl-3,6-diazabicyclo[3.2.2]nonane
3-(1,2-oxazinan-2-yl)-N-[3-(pyridin-3-yloxy)propyl]propanamide
5-{[3-(3-fluoro-4-methoxybenzoyl)piperidin-1-yl]methyl}-N,N-dimethyl-1,3-thiazol-2-amine
2-methyl-4-[4-({[(3-methylthiophen-2-yl)methyl](pyridin-2-ylmethyl)amino}methyl)phenyl]but-3-yn-2-ol
ethyl 4-[(4-methoxyphenyl)methyl]-1-[2-(5-oxopyrrolidin-2-yl)acetyl]piperidine-4-carboxylate
6-(benzyloxy)-1-cyclohexyl-4-[3-(2-oxoimidazolidin-1-yl)benzoyl]-1,4-diazepan-2-one
methyl 4-(8-methoxy-2-methylquinolin-5-yl)pyridine-2-carboxylate
3-(1,2-oxazinan-2-yl)-1-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}propan-1-one
2-(3,4-dimethoxyphenyl)-1-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]ethan-1-one
(3R,4R)-4-(azepan-1-yl)-1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-3-ol
1-(piperidin-1-yl)-3-(4-{[4-(pyrazin-2-yl)piperazin-1-yl]methyl}phenoxy)propan-2-ol
(2,1,3-benzoxadiazol-4-ylmethyl)(methyl)[1-(pyrimidin-4-yl)ethyl]amine
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(pyrazin-2-yl)acetamide
1-[(1R,3S)-1-hydroxy-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-7-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one