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N-[(8-{[4-(propan-2-yl)phenyl]methyl}-1-oxa-8-azaspiro[4.5]decan-2-yl)methyl]benzamide
1-(2-methylpropyl)-4-{4-[(pyrimidin-2-yl)amino]piperidine-1-carbonyl}pyrrolidin-2-one
1,3-dimethyl-4-(2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carbonyl)piperazin-2-one
1-[(3,5-dimethylphenyl)methyl]-4-{2-[4-(hydroxymethyl)phenyl]acetyl}piperazin-2-one
4-({4-methyl-5-[1-(4-methylpyrimidine-5-carbonyl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
N-[(3-chlorophenyl)methyl]-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
(2S)-2-[(5-methylhexan-2-yl)amino]-3-phenylpropan-1-ol
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-3,5-dimethyl-N-(oxolan-2-ylmethyl)furan-2-carboxamide
1-[2-(2H-1,3-benzodioxol-5-ylmethyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]piperidine-3-carboxamide
2-methoxy-4-{6-oxo-7-propyl-2,7-diazaspiro[4.5]decan-2-yl}pyridine-3-carbonitrile
7-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2,4-dimethylquinoline
2-methyl-6-{4-oxo-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl}-2,3-dihydropyridazin-3-one
1-(5-propyl-1,2-oxazole-3-carbonyl)-4-(thian-4-yl)piperazine
2-{1-[(2-fluorophenyl)methyl]-4-(propan-2-yl)piperazin-2-yl}ethan-1-ol
2-phenyl-1-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-{thieno[3,2-d]pyrimidin-4-yl}piperidin-3-ol
1-[4-(2-methylbutyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]-2-phenylethan-1-ol
2-[({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(oxolan-2-ylmethyl)amino]acetic acid
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]acetamide
3-ethyl-8-[(1-methyl-1H-indol-3-yl)methyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(cyclohexylmethyl)-2-methanesulfonyl-5-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}-1H-imidazole
3-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-4,5,6,7-tetrahydro-1,2-benzoxazole
(3R,4R)-1-(8-chloroquinoline-2-carbonyl)-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
1-(2-chloro-4-fluorobenzenesulfonyl)-3-(2-methoxybenzoyl)piperidine
N,N-dimethyl-5-{[4-(thiomorpholin-4-yl)piperidin-1-yl]methyl}pyridin-2-amine
N-(2-hydroxy-1-phenylethyl)-1-(methoxymethyl)cyclobutane-1-carboxamide
N-{3-[methyl(phenyl)amino]propyl}-2-(pyrrolidin-3-yl)acetamide
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
1-{2-[3-(2-chlorophenoxy)azetidin-1-yl]-2-oxoethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
1-{[4-(hydroxymethyl)oxan-4-yl]methyl}-1-methyl-3-[3-(2-methyl-1,3-thiazol-4-yl)phenyl]urea
ethyl 1-(5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-4-(3-phenylpropyl)piperidine-4-carboxylate
4-(5-fluoropyrimidin-2-yl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]pyrazolo[1,5-a]pyridine-7-carboxamide
3-(2-methylphenyl)-N-(5-oxo-1-propylpyrrolidin-3-yl)propanamide
1-[(3-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}-1,2-oxazol-5-yl)methyl]piperidin-4-ol
4-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
6-methyl-3-[1-(1H-pyrazol-1-yl)propan-2-yl]-3,4-dihydroquinazolin-4-one
2-(2,3-dihydro-1H-inden-1-yl)-N-[(3-hydroxy-4-methoxyphenyl)methyl]-N-methylacetamide
1-[2-(dimethyl-1,2-oxazol-4-yl)ethyl]-2-(3-methoxyphenyl)piperidine
2-(4-ethoxyphenyl)-1-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-1H-imidazole
2,3-dimethyl-7-{[3-(pyrimidin-2-yloxy)phenyl]methyl}-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
[(3-methoxyphenyl)methyl](prop-2-en-1-yl){[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}amine
N-methyl-3-(1-methyl-1H-pyrazol-5-yl)-N-[2-(1H-pyrazol-1-yl)ethyl]propanamide
6-methoxy-3-methyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-1-benzofuran-2-carboxamide
3-(3,4-dimethoxybenzoyl)-1-(1-methyl-1H-pyrazole-5-carbonyl)piperidine
(5S,9aS,9bS)-2-cyclopentyl-5-(3,5-dimethylphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-methyl-N-(pyrimidin-4-ylmethyl)-6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-amino-6-(2-amino-5-methyl-1,3-thiazol-4-yl)-4-(2,5-difluorophenyl)pyridine-3-carbonitrile