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2-benzyl-5-formamido-N,1-dimethyl-N-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
(1S,9S)-11-{2-methylimidazo[1,2-a]pyridine-6-carbonyl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
2-{1-[(5-methylfuran-2-yl)methyl]-4-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-methyl-N-[2-(oxan-4-yl)ethyl]-1H-pyrazole-3-carboxamide
5-{1-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]pyrrolidin-2-yl}-N-ethylthiophene-2-carboxamide
N'-({1-[(2-methoxy-3,5-dimethylphenyl)methyl]piperidin-3-yl}methyl)ethanediamide
3-{5-[2-methyl-2-(1H-pyrrol-1-yl)propanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
N-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]-2-propyl-1,3-thiazole-4-carboxamide
N-[4-(3-fluorophenyl)phenyl]-1-(3-methoxypropanoyl)piperidine-3-carboxamide
3-(3-fluorophenyl)-6-(oxane-4-carbonyl)-1-[2-(piperidin-1-yl)ethyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}-1-[4-(morpholine-4-carbonyl)phenyl]piperidin-4-amine
N-phenyl-3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
5-[1-(2,3-difluorobenzoyl)piperidin-4-yl]-5-ethyl-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]imidazolidine-2,4-dione
N-[2-(2-methoxyphenyl)ethyl]-3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
2-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-methyl-N-(naphthalen-1-ylmethyl)-1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
(1S,4S)-2-(5-chloro-2-methoxyphenyl)-5-(3-fluorobenzoyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
6-ethyl-N-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-2-(piperidin-1-yl)pyrimidin-4-amine
1-[5-(methoxymethyl)furan-2-carbonyl]-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
2-({[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)amino}methyl)pyridine-3-carboxylic acid
(1S,5R)-3-{2-[(cyclopropylmethyl)sulfanyl]acetyl}-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(2,1,3-benzoxadiazol-5-ylmethyl)(methyl)({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)amine
3-[(6-amino-2-{[(2-methylphenyl)methyl]sulfanyl}pyrimidin-4-yl)(methyl)amino]propanamide
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
2-amino-6-(furan-2-yl)-4-(isoquinolin-5-yl)pyridine-3-carbonitrile
4-[3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-N-methylpyridin-2-amine
8-[2-(adamantan-1-yl)acetyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
6-({4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]piperidin-1-yl}methyl)pyridine-2-carboxylic acid
N,N-dimethyl-7-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-2-(phenylamino)pyrimidine-5-carboxamide
methyl 3-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)-7-oxo-9-(3-phenylpropoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-(4-phenyl-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}piperidin-4-yl)ethan-1-one
(4aR,7aS)-1-(2-hydroxyethyl)-4-[(6-methylquinolin-5-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
9-methoxy-N-[(3-methoxyphenyl)methyl]-3-(2-methyl-4-oxopentanoyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
6-(4-oxo-4H-chromene-2-carbonyl)-N-phenyl-6-azaspiro[2.5]octane-1-carboxamide
(2S,4S)-4-amino-1-(4-chloro-1-methyl-1H-indole-2-carbonyl)-N,N-diethylpyrrolidine-2-carboxamide
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one
2-{4-[3-(hydroxymethyl)piperidin-1-yl]piperidin-1-yl}-6-(2-methoxyphenyl)-N-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]pyridine-3-carboxamide
3-methyl-1-(1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)butan-1-ol
N-{2-[(2-chlorophenyl)formamido]ethyl}-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamide
3-(1-{[4-chloro-2-(dimethylamino)-1,3-thiazol-5-yl]methyl}piperidin-3-yl)-N-cyclopropylpropanamide
N-[(5-chlorothiophen-2-yl)methyl]-2-ethyl-4-methyl-1,3-oxazole-5-carboxamide
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-(pentan-3-yl)piperazin-2-yl}ethan-1-ol
N-methyl-N-{1-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]-2-phenylethyl}pyridine-2-carboxamide
N-[2-(3-fluorophenyl)ethyl]-3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
1-(2,3-dimethylphenyl)-3-methyl-3-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]urea
2-methyl-9-[(4-methyl-6-phenylpyrimidin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-4,6-dimethyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
2-(methylsulfanyl)-N-({5-[4-(methylsulfanyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)acetamide
2-(2,3-dimethylbenzamido)-N-[2-methyl-2-(morpholin-4-yl)propyl]-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide