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N-[(3S,4R)-1-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
N-{[7-({4-[methyl(phenyl)amino]phenyl}methyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}acetamide
N-(4-methoxyphenyl)-5-(4-methyl-1H-pyrazol-1-yl)furan-2-carboxamide
4-benzyl-2-[(1-cyclohexyl-3-methyl-1H-1,2,4-triazol-5-yl)methyl]morpholine
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-(1-methyl-1H-pyrazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(cyclohex-1-en-1-ylmethyl)-5-oxo-1-(propan-2-yl)pyrrolidine-3-carboxamide
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
7-[(3-chlorophenyl)methyl]-3-(oxolan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
N-cyclopentyl-N-ethyl-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
3-{[1-(2H-1,3-benzodioxole-5-carbonyl)pyrrolidin-3-yl]methyl}benzamide
N-(prop-2-en-1-yl)-2-[4-(pyrimidin-2-yloxy)piperidine-1-carbonyl]aniline
1-methyl-N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(2,5-dimethylphenyl)-1-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
2,7,8-trimethyl-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]quinoline-4-carboxamide
2-(dimethylamino)-N-[3-({[1-(6-methylpyridin-3-yl)ethyl]carbamoyl}amino)phenyl]acetamide
4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(oxan-4-yl)piperidine
1-cyclohexyl-N-[(2-methylphenyl)(pyridin-4-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
1-(3,5-dimethoxybenzoyl)-4-(pyrimidin-2-yl)piperazine-2-carboxylic acid
ethyl 1-[(3-hydroxy-4-methoxyphenyl)methyl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
N-(oxan-4-ylmethyl)-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propanamide
3-(2-phenylphenyl)-1,2,4,5,10,11-hexaazatricyclo[7.3.0.02,6]dodeca-3,5,7,9,11-pentaene
N-(3-{[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}phenyl)pentanamide
N-{[7-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
methyl 3-(2-methylpropanamido)-6-[(4-phenylpiperidin-1-yl)methyl]thieno[2,3-b]pyridine-2-carboxylate
4-methyl-2-{[methyl(quinolin-5-ylmethyl)amino]methyl}phenol
6-methyl-N-[3-(4-methylbenzenesulfonamido)propyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
3-[(3R,4S)-4-(dimethylamino)-1-[2-(2,4,7-trimethyl-1H-indol-3-yl)acetyl]piperidin-3-yl]propanoic acid
3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[1-(1H-indol-1-yl)propan-2-yl]propanamide
4-(3-ethoxyphenyl)-2-methyl-5H,6H,7H-cyclopenta[d]pyrimidine
(1R,5R)-6-benzyl-3-(dimethyl-1,3-thiazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-{2-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(carbamoylmethyl)-N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]piperidine-4-carboxamide
8-(2-methoxypyridine-3-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2,5-dimethoxy-N-{[4-(2-methylpropyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}benzamide
methyl 5-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
N,5-dimethyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
N-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
1-[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
(3S,9aR)-3-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-(3-methylphenyl)-5-{3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]propyl}-1,2,4-oxadiazole
(2R,3S,6R)-3-phenyl-5-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}-1,5-diazatricyclo[5.2.2.02,6]undecane
3-{[(1R,5S,8S)-8-(dimethylamino)-3-azabicyclo[3.2.1]octan-3-yl]methyl}benzoic acid
N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-3-methyl-N-(oxolan-2-ylmethyl)thiophene-2-carboxamide
1-[(3-fluorophenyl)methyl]-4-(3-phenyl-1,2-oxazole-4-carbonyl)piperazin-2-one
N-methyl-3-(5-methylthiophen-2-yl)-N-(quinolin-4-ylmethyl)-1H-pyrazole-5-carboxamide
3-(5-hydroxy-1,2-dimethyl-1H-indole-3-carbonyl)-3,9-diazaspiro[5.6]dodecan-10-one
1-benzyl-3-(2-methoxyethyl)-8-[(4-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(cyclohex-3-en-1-ylmethyl)-4-[2-(methoxymethyl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidine
2-(4-chloro-2-methylphenoxy)-N-{[8-(3-methylbutanoyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}propanamide
(1S,5R)-6-(5-methylthiophene-3-carbonyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane