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N-[(3S)-1-benzylpyrrolidin-3-yl]-4-ethyl-5-methylpyrimidin-2-amine
3-[1-(2,1,3-benzoxadiazol-4-ylmethyl)piperidin-4-yl]-N-(oxolan-2-ylmethyl)propanamide
N-({7-[2-(2-methoxyphenyl)acetyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)oxolane-3-carboxamide
1-(cyclohexylmethyl)-N-[1-(4-methylphenyl)propyl]-1H-1,2,3-triazole-4-carboxamide
1-({5-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3-dimethylurea
2-(1,2-oxazol-5-yl)-4-[2-(pyridin-2-yl)-1H-imidazol-1-yl]phenol
3-[2-(3-fluorophenyl)ethyl]-1-(propane-2-sulfonyl)piperidine
2-(1H-imidazol-1-yl)-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]propanamide
3-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-(furan-2-ylmethyl)propanamide
2-(5-{1-[2-(4-chloro-1H-pyrazol-1-yl)propanoyl]piperidin-4-yl}-1H-pyrazol-3-yl)acetic acid
3-propyl-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]-1H-pyrazole-5-carboxamide
2-[(cyclopropylmethyl)sulfanyl]-N-methyl-N-(quinolin-5-ylmethyl)acetamide
1-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-1,2,4-triazole
1-(4-fluorophenyl)-4-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}butane-1,4-dione
2-methyl-1-[4-(2-phenylethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]propan-1-ol
N-methyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
{4-[(3R,4S)-3-(dimethylamino)-4-propylpyrrolidine-1-carbonyl]phenyl}methanol
3-hydroxy-1-(3-phenylpropyl)-3-(thiomorpholin-4-ylmethyl)piperidin-2-one
1-[(2,6-difluorophenyl)methyl]-N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
7-({4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}methyl)-1H-indole
methyl 6-[3-(2-chlorophenyl)propanoyl]-2-(diethylsulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-(4-chlorobenzoyl)-1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)piperidine
(furan-2-ylmethyl)({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})[2-(morpholin-4-yl)ethyl]amine
(3aS,6aS)-5-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
methyl 3-{3-[(2-methoxyethyl)carbamoyl]-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}propanoate
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-3-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
6-(5-fluoro-2-methoxyphenyl)-1,3-benzothiazol-2-amine
N2-{2-cyclopentyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl}-N1-(pyridin-3-yl)ethane-1,2-diamine
N-methyl-N-(2-methylpropyl)-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
3-[(4aR,7aS)-4-(5-hydroxypyrazine-2-carbonyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
3-(4-methoxy-3,5-dimethylbenzoyl)-1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)piperidine
2-methyl-1-[1-(1-propyl-1H-pyrazole-5-carbonyl)azetidin-3-yl]piperidine
2-{[4-(2-methoxyethyl)piperazin-1-yl]methyl}-N-[2-(2-methoxyphenyl)ethyl]quinazolin-4-amine
1-(4-chlorophenyl)-5-methyl-4-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}piperazin-2-one
9-acetyl-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(1,1-dioxo-1λ6-thiolan-3-yl)-3,3-diphenylpiperidine-1-carboxamide
2-{4-[(4-fluorophenyl)methyl]-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl}-6-methylpyridine-3-carboxylic acid
9-[2-(methylsulfanyl)propanoyl]-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(4,7-dimethylquinazolin-2-yl)-N-[(3-fluoro-4-methylphenyl)methyl]piperidine-4-carboxamide
1-(3-{[6-(thiomorpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]amino}propyl)pyrrolidin-2-one
3-(2H-1,3-benzodioxol-5-ylmethyl)-N-[(1R,2S)-2-phenylcyclohexyl]-1,2-oxazole-5-carboxamide
4-[(2-methylphenyl)sulfanyl]-1-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}piperidine
4,6-dimethyl-2-{[2-(3,4,5-trimethoxyphenyl)-1H-imidazol-1-yl]methyl}pyrimidine
2-(2-methoxyethyl)-8-(5-methyl-1H-indazole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
[(2R)-1-(5-chloro-3-phenyl-1H-indole-2-carbonyl)pyrrolidin-2-yl]methanol
2-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-methyl-2-{2-methylimidazo[1,2-a]pyridin-3-yl}-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}acetamide
3-[(4-methoxypyridin-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-1-[(4-methylphenyl)amino]cyclopentane-1-carboxamide
2-{4-[6-fluoro-4-(4-methylpiperazine-1-carbonyl)quinolin-2-yl]-1H-pyrazol-1-yl}ethan-1-ol