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2-(2,6-dimethoxy-4-methylphenyl)-2-[methyl(pyrazin-2-ylmethyl)amino]acetic acid
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-5-(4-methylphenyl)-1H-pyrazole-3-carboxamide
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-[2-(furan-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-[2-(3-methoxyphenyl)ethyl]-1-(1,3-thiazol-2-yl)piperidine
8-methoxy-3-(piperidin-4-yl)-3,4-dihydroquinazolin-4-one
6-(aminomethyl)-2-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}pyrimidin-4-amine
2-amino-3-ethyl-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-methyl-3-{[2-(phenylamino)pyrimidin-5-yl]formamido}propanoic acid
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2H-1,3-benzodioxole-5-carboxamide
3-{1-[(7-chloro-3-methyl-1H-indol-2-yl)methyl]piperidin-4-yl}-1-(morpholin-4-yl)propan-1-one
methyl 5-{[1-(2-fluorophenyl)propan-2-yl]amino}-1-[2-(1H-indol-3-yl)ethyl]-3-(3-methoxypropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-({[1-(pyrimidin-2-yl)piperidin-4-yl]amino}methyl)benzene-1-sulfonamide
1-(1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)-2-methylpropan-1-ol
(1R,5R)-6-(cyclobutylmethyl)-3-[4-(propan-2-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
4-(5-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecane-11-carbonyl}-1H-pyrazol-3-yl)phenol
(3R)-1-({1-[1-(5-ethylthiophene-3-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)pyrrolidin-3-amine
2-{3-[(2,4-difluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}pyridine-3-carbonitrile
2-(propan-2-yl)-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1,3-benzoxazole-5-carboxamide
N-methyl-3-(methylsulfanyl)-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]propanamide
methyl (2S,4R)-4-(5-chloro-3-phenyl-1H-indole-2-amido)-1-(2-methylpropyl)pyrrolidine-2-carboxylate
1-{5H,6H-benzo[h]quinazolin-2-yl}-N-(2-methoxyethyl)-5-methyl-N-(propan-2-yl)-1H-pyrazole-4-carboxamide
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperazine
1-[2-methoxy-5-({[2-(methylsulfanyl)ethyl]amino}methyl)phenoxy]-3-(4-methyl-1,4-diazepan-1-yl)propan-2-ol
1-[(2-methoxyphenyl)methyl]-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
2-(2-chloro-6-methoxy-4-{[2-(methoxymethyl)piperidin-1-yl]methyl}phenoxy)acetamide
3-methanesulfonamido-N-[(4-methoxyphenyl)methyl]-N-propylpropanamide
3-{5-[(2S)-1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]pyrrolidin-2-yl]-1,2,4-oxadiazol-3-yl}pyridine
6-[(3-methoxyphenyl)methoxy]-4-(oxane-4-carbonyl)-1-(2-phenylethyl)-1,4-diazepan-2-one
3-chloro-2-methyl-N-{[4-(2-methylphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}benzene-1-sulfonamide
1-benzyl-8-(9H-fluoren-2-ylmethyl)-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(carbamoylmethyl)-N-[(5-chloro-1H-indol-2-yl)methyl]piperidine-4-carboxamide
N-cyclopropyl-3-{1-[1-(pyridin-2-yl)piperidine-3-carbonyl]piperidin-4-yl}propanamide
1-methyl-1'-{[2-(propylamino)pyrimidin-5-yl]methyl}-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
N-(furan-2-ylmethyl)-1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carboxamide
2-methoxy-1-{4-[4-(4-methylphenoxy)piperidine-1-carbonyl]piperidin-1-yl}ethan-1-one
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
2-(4-fluorophenyl)-N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-hydroxy-N-methylacetamide
N-[1-(4-fluorophenyl)-2-methylpropan-2-yl]-2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]acetamide
(2S)-2-amino-3-hydroxy-1-{6-[(4-methylpiperazin-1-yl)sulfonyl]-1,2,3,4-tetrahydroisoquinolin-2-yl}propan-1-one
1-[4-({3-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)piperazin-1-yl]ethan-1-one
1-[4-(2H-1,3-benzodioxol-4-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]-3-phenylpropan-1-ol
6-[3-(4-chlorobenzoyl)piperidine-1-carbonyl]-2-methyl-2,3-dihydropyridazin-3-one
1-(2-methoxyethyl)-6-oxo-N-[3-(pyridin-3-yl)propyl]piperidine-3-carboxamide
3-[(3aS,6aS)-1-(pyridine-3-carbonyl)-octahydropyrrolo[2,3-c]pyrrole-5-carbonyl]-1-methyl-4,5,6,7-tetrahydro-1H-indazole
3-(but-2-yn-1-yl)-5-[1-(but-2-ynoyl)piperidin-4-yl]-5-(2-phenylethyl)imidazolidine-2,4-dione
3-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}-1-(oxan-4-yl)piperidine
N-[(5-oxopyrrolidin-2-yl)methyl]-N-(propan-2-yl)-2-(4-propanoylphenoxy)acetamide
1-{5-[(diethylamino)methyl]-2-methylfuran-3-carbonyl}-3-ethylpiperidine-3-carboxylic acid
N-cyclopropyl-N-({4-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-4-(4-methylphenyl)benzamide
N,N-dimethyl-4-[1-(2-phenylethyl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]piperidine-1-carboxamide