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1-benzyl-3-(4-ethyl-1,3-dimethyl-1H-pyrazol-5-yl)-1-(2-hydroxyethyl)urea
1-[5-({5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-1H-pyrazol-3-yl]ethan-1-one
1-(pyrrolidin-1-yl)-4-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butan-1-one
2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-1-[4-(thiophene-2-carbonyl)piperazin-1-yl]ethan-1-one
3-{5-[(3-methoxyphenyl)carbamoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
1-butyl-3-methyl-5-{2-methylimidazo[1,2-a]pyrimidin-3-yl}-1H-1,2,4-triazole
2-(2-{1-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
N,2-dimethyl-N-(2-phenyl-1-{1-[(2E)-3-(pyridin-4-yl)prop-2-enoyl]piperidin-4-yl}ethyl)furan-3-carboxamide
N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-(propan-2-yl)acetamide
(1R,5R)-N,N-dimethyl-6-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
methyl 4-{[(1-{4-[(benzylcarbamoyl)methyl]phenyl}piperidin-4-yl)amino]methyl}benzoate
(3R,5R)-N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
6-(4-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}piperazin-1-yl)-9H-purine
8-chloro-2-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}quinoline
2-[(6-{[(4-fluorophenyl)methyl](methyl)amino}pyridazin-3-yl)oxy]-1-[4-(4-methyl-1,2,5-oxadiazol-3-yl)piperazin-1-yl]ethan-1-one
9-ethyl-1-methyl-4-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[(2R,3R)-2-methoxy-1'-(3-phenylprop-2-yn-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
methyl 2-[1-(2-methoxyethyl)-2,4-dioxo-8-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
2-chloro-4-[6-(propan-2-yloxy)pyridazin-3-yl]benzamide
1-cyclobutanecarbonyl-4-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]-1,4-diazepane
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-({methyl[2-(pyrrolidin-1-yl)ethyl]amino}methyl)piperidin-2-one
2-{2-[(2,6-dimethylquinolin-4-yl)formamido]ethyl}-4-methyl-1,3-thiazole-5-carboxylic acid
[(1-methyl-1H-pyrazol-4-yl)methyl](propan-2-yl)({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)amine
N-(2-methoxy-2-methylpropyl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-[1-(2-phenylethyl)piperidin-3-yl]-1-benzofuran-2-carboxamide
2-(4,6-dimethyl-1-benzofuran-3-yl)-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}acetamide
8-[5-(hydroxymethyl)furan-2-carbonyl]-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
3-(pyridin-4-yl)-1-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]propan-1-one
2-cyclopropyl-N-[4-(methylamino)butyl]pyrimidine-5-carboxamide
3-{1-methyl-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-5-yl}-2-(methylsulfanyl)pyridine
N-(2-fluorophenyl)-3-[1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)piperidin-3-yl]propanamide
1-{2-[1-(1-benzofuran-5-carbonyl)piperidin-4-yl]ethyl}pyrrolidin-2-one
1-[4-(1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-5-methyl-1H-pyrazole-4-carbonyl)piperazin-1-yl]ethan-1-one
4-(2,6-difluorobenzoyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
4-[(2-fluoro-4-methoxyphenyl)methyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-one
1-[2-(4-{2-[(4-fluorophenyl)methyl]-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)-2-oxoethyl]-4-phenylpyrrolidin-2-one
1-(1-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}azetidin-3-yl)piperidine
N-benzyl-N-[(4-methyl-1,3-thiazol-5-yl)methyl]-2-[4-(propan-2-yl)morpholin-2-yl]acetamide
4-{[2-(2,3-dihydro-1-benzofuran-5-yl)phenyl]methyl}morpholine
2-[3-({4-[(2-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenoxy]ethan-1-ol
[3-(2-phenylethyl)-1-[1-(pyridin-2-ylmethyl)piperidin-4-yl]piperidin-3-yl]methanol
1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-2-carboxamide
5-ethyl-4-{[4-ethyl-5-oxo-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]methyl}furan-2-carboxamide
ethyl 4-[({4-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]phenyl}carbamoyl)amino]piperidine-1-carboxylate
3-{2-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]ethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[5-(1-methyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]acetic acid
methyl 4-(5-{[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoate
1-{5-[(4-methoxyphenyl)methyl]-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperidin-4-ol
1-(2-chlorophenyl)-3-{1-[1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-6-methoxy-N-methylpyrimidin-4-amine