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2-({4-[(4-cyclopentyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}methyl)-6-methylpyridine
N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-{[(5-methylpyrazin-2-yl)methyl]amino}pyridine-3-carboxamide
1-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]-3-phenoxypropan-1-one
N-methyl-3-(2-methylpyrrolidine-1-carbonyl)-N-(pyrazin-2-ylmethyl)benzene-1-sulfonamide
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[(3R,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]ethan-1-one
{[3-(1H-1,3-benzodiazol-5-yl)-1,2,4-oxadiazol-5-yl](2-fluorophenyl)methyl}dimethylamine
6-methoxy-3-{[4-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}-1H-indazole
N-(2,3-dihydro-1H-inden-4-yl)-3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.5]decane-7-carboxamide
2-({4-[(4-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)-6-methoxyphenol
3-(2-{4-[hydroxy(phenyl)methyl]piperidin-1-yl}-2-oxoethyl)-1-(3-methoxypropyl)-3-(2-methylphenyl)pyrrolidine-2,5-dione
2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-(1-methoxypropan-2-yl)acetamide
2-(2-methyl-1,3-thiazol-4-yl)-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]acetamide
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-1-methyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
1-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrol-1-yl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
4-(1H-imidazol-2-ylmethyl)-1-[(4-methoxyphenyl)methyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
(1R,3S)-N3-ethyl-1,2,2-trimethyl-N1-{2-[(3-methylpyridin-2-yl)amino]ethyl}cyclopentane-1,3-dicarboxamide
1-(2-methoxyethyl)-N-methyl-N-[(5-methyl-1H-indol-3-yl)methyl]pyrrolidine-3-carboxamide
N-{[4-(cyclopentyloxy)phenyl]methyl}-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-cyclopentyl-5-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-(3-methoxy-2-methylbenzoyl)-1-(2-methoxyphenyl)piperazin-2-one
5-{1-[2-(2-methylphenyl)acetyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-(pyridin-3-yl)imidazolidine-2,4-dione
1-({2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)-4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidine
(2S,4R)-N-[2-(2-fluorophenyl)ethyl]-1-(2-methylpropyl)-4-{[(3-phenoxyphenyl)methyl]amino}pyrrolidine-2-carboxamide
2-ethyl-1-(propan-2-yl)-4-[2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]piperazine
N-(1-{1-[4-(piperidin-1-yl)benzoyl]piperidin-4-yl}-1H-pyrazol-5-yl)acetamide
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-N-[(2-methylphenyl)methyl]-N-(prop-2-en-1-yl)propanamide
5-{[2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]methyl}-2-(pyridin-2-yl)pyrimidine
1-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-5,5-diphenylpiperidin-2-one
4-(2-chlorophenoxy)-1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)piperidine
8-[(3,5-dimethoxyphenyl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidine-1-carbonyl)pyridine
2-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}pyridine-3-carboxamide
N-{[6,7-dimethoxy-2-(3-methoxyphenyl)quinolin-3-yl]methyl}-2-methyl-N-(oxolan-2-ylmethyl)-1,3-thiazole-4-carboxamide
1-({1-[6-(cyclopentylamino)pyridine-3-carbonyl]piperidin-4-yl}methyl)pyrrolidin-2-one
1-(3,5-dimethylphenyl)-N-[(3-ethoxy-4-methoxyphenyl)methyl]-4,5,6,7-tetrahydro-1H-indazol-4-amine
8-(5-methylpyrazine-2-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
6-(4-methylpiperazin-1-yl)-N4-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}pyrimidine-2,4-diamine
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-2-[methyl(piperidin-4-yl)amino]acetamide
5-(2-methoxyacetamido)-N,1-dimethyl-2-(pyridin-4-yl)-N-[1-(1,3-thiazol-2-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
1-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-2-(2-methyl-1H-imidazol-1-yl)propan-1-one
3-cyclopropyl-1-[4-(furan-2-ylmethoxy)phenyl]-3-[(1-methyl-1H-pyrazol-4-yl)methyl]urea
N-[2-(2-methoxyphenyl)ethyl]-2-(4-{4-[methyl(1H-pyrazol-5-ylmethyl)amino]piperidin-1-yl}phenyl)acetamide
N-[3-(dimethylamino)propyl]-N-methyl-1-(4-methylbenzenesulfonyl)piperidin-3-amine
{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}(thiophen-2-ylmethyl)amine
3-(2H-1,3-benzodioxol-5-yl)-N-methyl-N-[(5-methylfuran-2-yl)methyl]-3-phenylpropanamide
2-({4-[(2-fluorophenyl)methyl]piperidin-1-yl}methyl)pyridine
2-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}-1-(piperidin-1-yl)ethan-1-one
2-[(5-methylfuran-2-yl)methyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-{4-[2-(dimethylamino)-2-(4-fluorophenyl)acetyl]-2-oxopiperazin-1-yl}benzonitrile
1-phenyl-4-(1-propylpiperidin-4-yl)piperazine