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7-(cyclobutylmethyl)-2-[1-(propan-2-yl)-1H-pyrrole-2-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
N-{[2-(3-chlorophenyl)-7-fluoroquinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]oxolane-2-carboxamide
N-phenyl-5-(4H-1,2,4-triazol-4-yl)pyridin-2-amine
N-[1-(2,4-difluorophenyl)ethyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-(4-{3-[(2-methylprop-2-en-1-yl)oxy]benzoyl}morpholin-3-yl)acetic acid
4-[(1-benzyl-1H-imidazol-2-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
5-(2-chloro-6-fluoro-3-methoxyphenyl)-1-(1-cyclopropylethyl)-1H,4H-pyrazolo[3,4-d]imidazole
N-(pyridin-3-ylmethyl)-3-[(thiolan-3-yl)sulfamoyl]benzamide
N-(2-methylpropyl)-N-[(3-methylthiophen-2-yl)methyl]-1,4-dioxane-2-carboxamide
3-(3-hydroxy-3-methylbutyl)-N-[1-(1,3-thiazol-5-yl)propan-2-yl]benzamide
N-[1-(cyclohexylmethyl)piperidin-3-yl]-1H-indole-5-carboxamide
N-(propan-2-yl)-1-[(1s,4s)-4-(3,4-dimethoxybenzenesulfonamido)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
4,6-dimethyl-2-oxo-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-1,2,3,4-tetrahydropyrimidine-5-carboxamide
1-(2-methyl-4-{[1-(2-propoxyphenyl)ethyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
3-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}-N-ethylbenzamide
4-[3-(7-fluoro-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)phenyl]-2-methylbutan-2-ol
3-{2-[3-(4-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-1-methyl-3-(4-phenylphenyl)pyrrolidine-2,5-dione
N-(2-methoxy-4-{2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamido}phenyl)-2,2-dimethylpropanamide
(2S)-2-[({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amino]-3-phenylpropanamide
[(3R,4R)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}-1-(2-methylbenzoyl)pyrrolidin-3-yl]methanol
6-(benzyloxy)-1-cyclohexyl-4-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-1,4-diazepan-2-one
1-(2-chloro-4-fluorobenzoyl)-3-(2,5-difluorobenzoyl)piperidine
1-(1-benzyl-1H-pyrazole-4-carbonyl)-3-(3,4-dimethoxybenzoyl)piperidine
1,4,6-trimethyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-oxo-1,2-dihydropyridine-3-carboxamide
4-hydroxy-N-methyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2-phenylpyrimidine-5-carboxamide
N-{[7-chloro-2-(3-methylphenyl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)-2H-1,3-benzodioxole-5-carboxamide
N-cyclopropyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(phenylamino)pyrimidine-5-carboxamide
6-{4-[3-(trifluoromethyl)phenoxy]piperidin-1-yl}pyrimidine-2,4-diamine
N-[2-(2-oxo-1,3-oxazolidin-3-yl)phenyl]thiomorpholine-4-carboxamide
5-(1-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-1H-1,2,3-triazol-4-yl)pyrimidine
8-(1,3-benzothiazol-2-ylmethyl)-1-ethyl-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]-1-(2-methylphenyl)piperazin-2-one
4-{1-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]piperidin-3-yl}morpholine
N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-3-{4-[2-(3-methylphenyl)acetamido]-1H-pyrazol-1-yl}benzamide
N-[1-(hydroxymethyl)cyclopropyl]-2-[4-methyl-6-(morpholine-4-carbonyl)-3,4-dihydro-2H-1,4-benzoxazin-3-yl]acetamide
4-(5-methyl-1-propyl-1H-pyrazol-4-yl)-N-[1-(pyridin-4-yl)propyl]pyrimidin-2-amine
N-methyl-2-(morpholin-3-yl)-N-[(4-phenoxyphenyl)methyl]acetamide
1-(2-oxo-2-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}ethyl)-1,4-dihydroquinolin-4-one
3-(1-benzyl-1H-imidazol-2-yl)-1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidine
7-(oxan-4-yl)-2-[2-(2-oxopyrrolidin-1-yl)ethyl]-2,7-diazaspiro[4.5]decan-6-one
3-[2-(methylsulfanyl)benzoyl]-1-(3-phenylprop-2-yn-1-yl)piperidine
2-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidine-1-carbonyl]pyridin-3-ol
ethyl 2-[4-({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)morpholin-3-yl]acetate
4-(4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazine-2-carbonyl)morpholine
2-(4-{5-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-3-yl}phenyl)ethan-1-ol
methyl 5-[(cyclohexylmethyl)amino]-1-methyl-3-(2-phenoxyacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-{1-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-ethyl-1H-1,2,4-triazol-5-yl]propyl}morpholine
8-benzyl-1-(3-methylbutyl)-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{6-[3-(propan-2-yloxy)phenyl]pyridin-2-yl}piperazine
1-(3-carbamoylpyridin-2-yl)-4-(4-fluorophenoxy)piperidine-4-carboxylic acid