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N-{4-oxo-4-[4-oxo-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]butyl}acetamide
4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-methyl-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
2-[1,3-dimethyl-4-(3-propoxypiperidin-1-yl)-1H-pyrazolo[3,4-d]pyrimidin-6-yl]pyridine
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-5-(3-methoxyphenyl)-1,2,4-triazin-3-amine
2-{2-[1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
1-({4-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)-2,4-dimethyl-1,4-diazepane
N3-{3-azaspiro[5.5]undecan-9-yl}-N1-(pyridin-3-yl)propane-1,3-diamine
(2S,4S)-1-(2,3-dihydro-1H-inden-2-yl)-N-methyl-4-{[(3-methylphenyl)methyl]amino}pyrrolidine-2-carboxamide
N-cyclopropyl-3-[1-(thiophene-3-carbonyl)piperidin-4-yl]propanamide
N-[(7-{[3-(trifluoromethyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]benzenesulfonamide
6-{[5-(2-chlorophenyl)furan-2-yl]methyl}-N-methyl-N-(1,3-thiazol-4-ylmethyl)-6-azaspiro[2.5]octane-1-carboxamide
(5S,9aS,9bS)-2-(2,3-dihydro-1H-inden-2-yl)-5-[3-(1H-pyrazol-1-yl)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[2-(2-chlorophenyl)-1-{1-[(2,3-dimethoxyphenyl)methyl]piperidin-4-yl}ethyl]-N-methylfuran-2-carboxamide
N-[(4-methoxyphenyl)methyl]-N-(2-methylpropyl)furan-3-carboxamide
4-(1H-imidazol-1-yl)-N-[(3R,4S)-1-(oxan-4-yl)-4-propylpyrrolidin-3-yl]butanamide
[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
[(3R,4R)-1-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
(1S,9S)-11-(3-{2-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-2-yl}propanoyl)-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
N-(2-{4-[(4-phenylpiperidin-1-yl)methyl]phenoxy}propyl)-2H-1,3-benzodioxole-5-carboxamide
(3R,4R)-1-[(6-chloro-2H-chromen-3-yl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-ol
N,N-dimethyl-6-(3-{1-[(3-methylpyridin-2-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyridine-3-carboxamide
5-{4-[(2-fluorophenyl)methyl]piperidine-1-carbonyl}pyridin-2-amine
3-(4-{2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl}piperazin-1-yl)-1,2-dihydropyrazin-2-one
5-(4-fluorophenyl)-N-[2-(pyrrolidin-1-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-(6-hydroxy-1,4-oxazepan-4-yl)-2-(4-phenylpiperidin-1-yl)ethan-1-one
N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1-[2-(methylsulfanyl)pyrimidin-4-yl]piperidin-4-amine
4-[(2,3-dimethoxyphenyl)methyl]-3-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]piperazin-2-one
N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
5-{1-[3-(2-chlorophenyl)propanoyl]piperidin-4-yl}-3-(furan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
3-{2-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-2-oxoethyl}-4-(propan-2-yl)piperazin-2-one
1-(4-methoxy-3-methylbenzoyl)-N-phenylpiperidin-3-amine
6-(azepan-1-yl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
6-[(4-benzylpiperidin-1-yl)methyl]-N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[2-(dimethylamino)ethyl]-4-(5-fluoro-2-methylphenyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
2-{[4-(4-fluorophenyl)-4-hydroxypiperidin-1-yl]methyl}pyridine-3-carboxylic acid
4-[1-(3-fluorophenyl)-1H-1,2,4-triazol-5-yl]azepane
1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-(2-fluorophenyl)piperazine
(2S,4R)-N,N-diethyl-1-methyl-4-(1-phenylcyclopentaneamido)pyrrolidine-2-carboxamide
3-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N-(propan-2-yl)propanamide
(2S,4R)-N-cycloheptyl-1-[(2-fluoro-4-methoxyphenyl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
9-[2-(piperidin-1-yl)acetyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-{5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}phenol
N-{[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-2-(1-propylpiperidin-4-yl)acetamide
N-(2,3-dihydro-1H-inden-5-yl)-2-[4-(4-fluorophenyl)-2-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]acetamide
N-[1-(morpholin-4-ylmethyl)cyclopentyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
2-(1,2-benzoxazol-3-yl)-1-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]benzamide
8-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decane
[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl](methyl){spiro[2.3]hexan-1-ylmethyl}amine
[(2S,4R)-1-methyl-4-[(1-{thieno[3,2-d]pyrimidin-4-yl}piperidin-4-yl)amino]pyrrolidin-2-yl]methanol