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N-(3-cyanophenyl)-8-(2-methoxyethyl)-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide
1-cyclopropanecarbonyl-N-{[3-(methylcarbamoyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-4-carboxamide
methyl 5-[(1-hydroxypropan-2-yl)amino]-1-(2-methylpropyl)-3-(2-phenylacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(1R,3S)-3-{[3-(hydroxymethyl)phenyl]carbamoyl}cyclopentyl]imidazo[1,2-b]pyridazine-3-carboxamide
N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}-3-(1H-pyrazol-4-yl)propanamide
3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-[2-(methylsulfanyl)ethyl]benzamide
5-chloro-N-[(4-methoxyphenyl)(pyridin-4-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
2-methyl-N-(1H-1,2,4-triazol-5-ylmethyl)-1-benzofuran-5-carboxamide
2-{[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]amino}-1-(6-methyl-1,2,3,4-tetrahydroquinolin-1-yl)ethan-1-one
7-[2-(methylamino)-1,3-thiazole-4-carbonyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
3-methyl-N-({5-methyl-2-[4-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)benzamide
11-{[(3,4-difluorophenyl)methyl]amino}-4-(2,3-dihydro-1H-inden-2-yl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-[1'-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
N-[(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]-4-(morpholin-4-yl)pentanamide
2,3,5-trimethyl-N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
5-{1-[(3-chloro-4-hydroxyphenyl)methyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
2-methyl-N,N-bis(propan-2-yl)-4-(pyrrolidin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carboxamide
(3S,4S)-1-[6-(morpholin-4-yl)pyrimidin-4-yl]-4-(naphthalen-2-yl)piperidin-3-ol
1-(2-aminoethyl)-N-cyclopentyl-N-[(2-methoxyphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
2-{3-[(7-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]phenoxy}ethan-1-ol
1-[5-(1-cyclobutanecarbonylpyrrolidin-2-yl)thiophene-2-carbonyl]-3,3-difluoropiperidine
N-[(3R,4S)-1-[3-(dimethylamino)pyrazin-2-yl]-4-(propan-2-yl)pyrrolidin-3-yl]propane-1-sulfonamide
4-(3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanoyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-one
6-{3-[1-(1,4-dioxan-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}-N,N-dimethylpyridazin-3-amine
3-[4-(methylsulfanyl)benzoyl]-1-[3-(1H-pyrazol-1-yl)propyl]piperidine
1-cyclopentyl-5-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)piperidin-2-one
1-cyclobutanecarbonyl-4-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]-1,4-diazepane
5-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrole-1-sulfonyl]-1,3-dimethyl-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-N-ethyl-3-(piperidin-3-yl)benzamide
5-(2-chloro-4-methoxyphenoxymethyl)-N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-1,2-oxazole-3-carboxamide
3-{1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]piperidin-3-yl}-N-(2-fluorophenyl)propanamide
2-{[4-(2,3-dimethylphenyl)piperazin-1-yl]methyl}-4-(3,6-dimethylpyrazin-2-yl)phenol
6-cyclopentyl-1-methyl-N-[2-(4-methyl-1,3-thiazol-2-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(3S,9aR)-3-benzyl-8-(4-chlorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-chloro-4-fluoro-N-{2-[(pyridin-3-yl)amino]ethyl}-1-benzothiophene-2-carboxamide
N-methyl-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}-4-(1H-pyrazol-4-yl)butanamide
9-(2-methoxyethyl)-1-methyl-4-(1H-pyrrole-3-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
[(4-methoxyphenyl)methyl](methyl){[4-(oxolan-2-ylmethyl)-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}amine
2-{5-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1H-1,2,4-triazol-3-yl}pyridine
4-({5-[(1-propylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-3-yl}methyl)morpholine
2-amino-6-methyl-N-{2-[(pyridin-3-yl)amino]ethyl}pyrimidine-4-carboxamide
2-[(3,5-difluorophenyl)methyl]-8-(2-ethylbutanoyl)-2,8-diazaspiro[4.5]decan-3-one
(1R,3S)-7-[(2-ethylphenyl)methyl]-7-azaspiro[3.5]nonane-1,3-diol
[(3R,4R)-1-[(3,5-dichloropyridin-4-yl)methyl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
(1S,5R)-6-benzyl-3-(4-fluorobutyl)-3,6-diazabicyclo[3.2.2]nonane
methyl (2S,4S,5R)-1,2-dimethyl-4-{methyl[(3-methylpyridin-4-yl)methyl]carbamoyl}-5-(2-methylphenyl)pyrrolidine-2-carboxylate
5-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-N-methyl-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
[3-(2-methyl-1H-imidazol-1-yl)propyl]({[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
methyl[(1-phenylpyrrolidin-3-yl)methyl](pyridin-3-ylmethyl)amine
5-chloro-4-[1-(cyclohex-3-en-1-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1,3-dimethyl-1H-pyrazole