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1-[(2R,3R,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(propan-2-yloxy)ethan-1-one
2-[4-(1-benzothiophen-3-yl)-2-(morpholin-4-ylmethyl)phenoxy]-N-[(3,5-dimethoxyphenyl)methyl]acetamide
2-{5-[(5-ethyl-1-benzofuran-3-yl)methyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
4-({1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}methyl)-5-methyl-2-(3-methylphenyl)-1,3-oxazole
N-(5-methanesulfonyl-2-methylphenyl)-4-(pyridin-4-yl)piperazine-1-carboxamide
4-[(2-methoxyphenyl)methyl]-11-{[3-(methylsulfanyl)propyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-chloro-N-({1-[2-(morpholin-4-yl)-2-oxoethyl]piperidin-3-yl}methyl)benzamide
[(3R,4R)-1-[(2-fluorophenyl)methyl]-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
(1r,4r)-4-[({3-[3-(azepan-1-yl)-2-hydroxypropoxy]phenyl}methyl)amino]cyclohexan-1-ol
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-(4-{[(5-methylfuran-2-yl)methyl]amino}piperidin-1-yl)benzamide
2-[2-fluoro-3-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-4-carbonitrile
(1S,5R)-3-({2-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonane
{3-[(3-chlorophenyl)methyl]-1-[2-(morpholin-4-yl)benzoyl]piperidin-3-yl}methanol
5-benzyl-5-{1-[1-(4-methoxyphenyl)cyclopentanecarbonyl]piperidin-4-yl}imidazolidine-2,4-dione
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(6-methylpyridine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-[(3-fluorophenyl)methyl]-1-(2-phenylethyl)piperidine-3,5-dicarboxamide
N-[2-methyl-2-(morpholin-4-yl)propyl]-6-phenylimidazo[2,1-b][1,3]thiazole-3-carboxamide
2-[(1-cyclobutanecarbonylpiperidin-4-yl)formamido]-3-(1H-imidazol-4-yl)propanoic acid
4-(1H-imidazol-4-ylmethyl)-9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(1R,5S,6R)-3-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
[(5-ethylpyridin-2-yl)methyl](methyl){[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}amine
2-{2-[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]-1H-imidazol-1-yl}-N-methylacetamide
N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-2-(2-oxopyrrolidin-1-yl)propanamide
(1R,5R)-6-[3-(benzyloxy)propyl]-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-(4-methylphenyl)-4-{[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}pyrrolidin-2-one
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(1H-pyrazol-4-yl)propanamide
1-[(3-methylphenyl)methyl]-4-[(1R,2S,3S,4R,5S)-tricyclo[3.2.1.02,4]octane-3-carbonyl]piperazine
N-ethyl-N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-2,6-dimethylquinoline-4-carboxamide
(4aR,7aS)-1-(3-methylbut-2-en-1-yl)-4-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-({1-[(3,5-dimethylphenyl)methyl]piperidin-4-yl}methyl)-2-hydroxy-2-methylpropanamide
2-(dimethylamino)-2-(3-fluorophenyl)-1-[4-(2-methoxyethyl)piperazin-1-yl]ethan-1-one
1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-[(4-fluorophenyl)methyl]-1,4-diazepan-5-one
N-({7-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-phenylacetamide
methyl (2S)-2-({[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]carbamoyl}amino)propanoate
[(1R)-1-(3-methoxyphenyl)ethyl]({3-methyl-1-[2-(thiomorpholin-4-yl)ethyl]-1H-pyrazol-4-yl}methyl)amine
1-benzyl-8-(2,3-dihydro-1H-inden-2-yl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N3-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-N5-tert-butyl-1-cyclohexyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-phenyl-6-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
2-[(2R,3S,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-3-carboxylic acid
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-1-(propan-2-yl)piperidine-4-carboxamide
(2R,6R)-1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
N-(but-2-yn-1-yl)-N-(furan-2-ylmethyl)-2-{4-[2-(phenylsulfanyl)acetamido]-1H-pyrazol-1-yl}acetamide
2-{2-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]-2-oxoethyl}-5,6-dimethyl-2,3-dihydropyridazin-3-one
2-(4-{2-[3-(1H-1,2,3,4-tetrazol-1-yl)phenoxy]acetyl}morpholin-3-yl)acetic acid
3-(2-methylpropyl)-2-oxo-1-[2-(piperidin-1-yl)ethyl]-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
methyl 7-oxo-3-(pyridin-4-ylmethyl)-9-(thiophen-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(1S,5R)-N-benzyl-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
1-(2-methylphenyl)-3-{1-[1-(5-methylthiophene-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-(2-methylphenyl)piperidine
5-{2-[2-(5-methylfuran-2-yl)-1H-imidazol-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione