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1-[(1R,5R)-6-[(2,4-dichlorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
3-(4-methoxyphenyl)-3-phenyl-1-(thiomorpholin-4-yl)propan-1-one
2-[(2,6-dichlorophenyl)methyl]-5-(2,3-dihydro-1H-isoindole-2-carbonyl)pyrimidin-4-ol
1-(1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-1,2,3,6-tetrahydropyridin-4-yl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-(2-chlorophenyl)-3-{1-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
N-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-1-(pyridin-3-ylmethyl)piperidin-4-amine
2-methyl-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
1-[3-({[(3,5-dimethoxyphenyl)methyl]amino}methyl)pyridin-2-yl]piperidin-3-ol
3-[1-(cyclopropylmethyl)-1H-pyrazol-5-yl]-1-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]urea
5-[2-(4-methylpiperazin-1-yl)propanoyl]-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
2-phenyl-1-(1-{[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)ethan-1-ol
1-{3-[ethyl(pyridin-4-ylmethyl)amino]piperidin-1-yl}but-2-yn-1-one
[2-(1H-imidazol-1-yl)ethyl]({[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
1-[(1S,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-[(trifluoromethyl)sulfanyl]ethan-1-one
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-oxo-4-phenylbutanamide
(1S,2R)-N1-[2-(4-hydroxyphenyl)ethyl]-N2-propylcyclohexane-1,2-dicarboxamide
(2R,3R)-3-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-1'-methyl-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-(cyclopentylmethyl)-6-methyl-1-(pyridin-3-ylmethyl)-3-{1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl}-1,4-dihydropyridin-4-one
7-(3-chlorophenyl)-4-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N,N-diethyl-1-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}piperidine-3-carboxamide
3-{1-ethyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}pyridine
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-2-(2-phenyl-1H-imidazol-1-yl)acetamide
N-{1-[1-(2,3,4-trimethoxybenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopropanecarboxamide
1-{5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(pyridin-4-ylsulfanyl)ethan-1-one
2-[4-(4,6-dimethylpyrimidin-2-yl)-1H-pyrazol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
2-cyclopropyl-4-phenyl-9-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecane
(3aR,6aS)-2-ethyl-5-(4-fluorobenzenesulfonyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-{[(5-fluoro-1H-indol-2-yl)methyl]carbamoyl}pyridin-1-ium-1-olate
ethyl 2-(1-{2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetyl}piperidin-2-yl)acetate
2-methyl-5-({5-[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-4-phenyl-1H-imidazol-1-yl}methyl)pyrazine
2-cyclopentyl-N-(3-{4-[3-(methoxymethyl)piperidin-1-yl]piperidin-1-yl}phenyl)acetamide
3,5-dimethyl-4-{2-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]ethyl}-1H-pyrazole
1-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-3-[4-methyl-3-(2-oxopyrrolidin-1-yl)phenyl]urea
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-N,1,7-trimethyl-1H-indole-2-carboxamide
N,N-dimethyl-2-[(1S,5R)-3-(3-methylthiophene-2-carbonyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
N-[3-(6-methyl-1,3-benzoxazol-2-yl)propyl]-2-(4-methyl-1,4-diazepan-1-yl)acetamide
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]propanamide
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N,4-dimethyl-1,2,5-oxadiazole-3-carboxamide
5-ethyl-N-(1-methoxypropan-2-yl)-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
8-(2-butoxyacetyl)-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-2-[2-(thiophen-2-yl)ethyl]piperidine
4-[(3-fluorophenyl)methyl]-1-[(2E)-3-(4-methoxyphenyl)prop-2-enoyl]-1,4-diazepan-5-one
2-(5-{2-amino-6-[(4-methylphenyl)sulfanyl]pyrimidin-4-yl}-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl)ethan-1-ol
3-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1-[7-(1H-imidazol-1-yl)-2,3-dihydro-1,4-benzodioxin-6-yl]-3-methylurea
methyl 2-[ethyl(2-methylprop-2-en-1-yl)sulfamoyl]-6-(1H-indol-2-ylmethyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
6-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-[(7S,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(6-chloropyridin-3-yl)urea
3-{5-[(2-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}-1-[2-(1,3-thiazol-2-yl)ethyl]urea
5-ethyl-2-methyl-N-[1-(morpholin-4-ylmethyl)cyclopentyl]pyrimidin-4-amine
(5S,9aS,9bS)-5-(1,5-dimethyl-1H-pyrazol-4-yl)-2-[(2-methylphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one