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(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-[2-(2-oxo-1,2-dihydropyridin-1-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[1-(4-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-5-methyl-1,2-oxazole
N4-(thiophen-2-ylmethyl)-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine
1-(4,4-difluoropiperidin-1-yl)-2-(dimethylamino)-2-(2-fluorophenyl)ethan-1-one
2-{2-[4-(3,5-dimethyladamantane-1-carbonyl)piperazin-1-yl]ethoxy}ethan-1-ol
2-(phenoxymethyl)-N-[2-(pyrazin-2-yl)ethyl]-1,3-oxazole-4-carboxamide
(2S)-N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-2-acetamidopropanamide
N-methyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
2-methoxy-1-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
N-{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-N-[(trimethyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
3-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-1-{4-[2-(pyridin-2-yl)ethoxy]phenyl}urea
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-(furan-2-yl)-N-[3-(pyrrolidin-1-ylmethyl)phenyl]-1H-pyrazole-4-carboxamide
8-(3,6-dimethyl-1-benzofuran-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(5-chloro-6-methyl-1-benzofuran-3-yl)-N-[(5-methylpyrazin-2-yl)methyl]acetamide
4-{4-[1-(4-methylpiperazin-1-yl)ethyl]piperidine-1-carbonyl}phenol
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-(1H-imidazol-2-ylmethyl)piperidine-4-carboxamide
1-{3-[2-(pyridin-2-yl)-1H-imidazol-1-yl]phenyl}propan-1-one
1-cyclopropanecarbonyl-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]piperidine-4-carboxamide
(3S,4R)-1-(1H-indole-6-carbonyl)-N,N-dimethyl-4-propylpyrrolidin-3-amine
5-{1-[(2S)-1-acetylpyrrolidine-2-carbonyl]piperidin-4-yl}-5-(2-methylpropyl)-3-(thiophen-2-ylmethyl)imidazolidine-2,4-dione
1-[(4aS,8aS)-7-(5,6-dimethoxypyrazine-2-carbonyl)-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]ethan-1-one
(5R)-5-[1-(5-chloro-2-methoxyphenyl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]pyrrolidin-2-one
N,N-dimethyl-5-(quinolin-6-yl)thiophene-2-carboxamide
1-(2-cyclopentylacetyl)-N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]piperidine-2-carboxamide
2-phenyl-7-(5-phenylpentanoyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-{1-[7-(quinolin-5-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}furan-2-carboxamide
(4aS,7aR)-1-(3-methyl-1H-pyrazole-5-carbonyl)-4-(3-methylbutanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(1R,3R)-3-aminocyclopentyl]-2-(pyridin-3-yloxy)acetamide
(3aS,6aS)-2-benzyl-5-[(2-methyl-1,3-thiazol-4-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-N-[3-(oxolan-3-yl)propyl]piperidin-4-amine
2,4-dimethoxy-6-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-1,3,5-triazine
3-[3-(6-methoxynaphthalene-2-carbonyl)piperidine-1-carbonyl]pyridin-1-ium-1-olate
N-(2-hydroxy-1-phenylethyl)-1-oxo-1,2-dihydroisoquinoline-4-carboxamide
N-cyclobutyl-2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}acetamide
1-[1-(4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)piperidin-4-yl]propan-1-ol
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]propanamide
2-{1-[(2-cyclohexylpyrimidin-5-yl)methyl]piperidin-2-yl}acetic acid
3-{1-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]piperidin-4-yl}-N-phenylpropanamide
N-methyl-N-[2-(morpholin-4-yl)ethyl]-2-[4-(trifluoromethyl)phenyl]-1,3-benzoxazole-5-carboxamide
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-N-[2-(diethylamino)ethyl]-1H-pyrazole-4-carboxamide
(2R,3R,6R)-5-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-{[4-(4-methoxypyrimidin-2-yl)piperazin-1-yl]methyl}-N-propylpyrimidin-2-amine
6-[(diethylamino)methyl]-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
6-[4-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]quinoxaline
7-{[4-(benzyloxy)piperidin-1-yl]methyl}-4-(1-ethylpiperidine-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(1-{5H,6H-benzo[h]quinazolin-2-yl}-5-(furan-2-yl)-1H-pyrazole-4-carbonyl)-4-ethylpiperazine
8-(butan-2-yl)-3-[(4-methoxyphenyl)methyl]-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-[1-(2,3-dimethoxybenzoyl)piperidin-4-yl]-3-(oxolan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
3-{[(2S)-oxolan-2-ylmethyl]sulfamoyl}-N-[2-(1,3-thiazol-4-yl)ethyl]benzamide