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N-(2-fluorophenyl)-3-[3-(trifluoromethyl)benzoyl]piperidine-1-carboxamide
3-{5-[1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1H-1,2,3-triazol-4-yl]thiophen-3-yl}prop-2-yn-1-ol
methyl (2S,4R)-1-benzyl-4-(4-methylbenzamido)pyrrolidine-2-carboxylate
(3S,4R)-1-[4-(4-fluorophenyl)-4-oxobutanoyl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
5,6-dimethyl-3-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-1,2-dihydropyridin-2-one
N-[(4-ethylphenyl)methyl]-2-(3-hydroxyphenyl)-N-(2-methoxyethyl)acetamide
{[5,8-dimethoxy-2-(2-methoxyphenyl)quinolin-3-yl]methyl}dimethylamine
N-[2-(4-hydroxyphenyl)-2-oxoethyl]-N-methyl-1H-1,3-benzodiazole-2-carboxamide
1-{[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}-N-(6-phenoxypyridin-3-yl)piperidine-2-carboxamide
1-benzyl-2-methyl-5-(2-methylpropanamido)-N-(oxan-4-ylmethyl)-1H-1,3-benzodiazole-7-carboxamide
2-{4-[(2-ethoxyphenyl)methyl]-1-(propan-2-yl)piperazin-2-yl}ethan-1-ol
6-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
1-(4-benzylpiperazin-1-yl)-3-{1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-3-yl}propan-1-one
(5-{[2-(butylsulfanyl)pyrimidin-5-yl]methyl}-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)methanol
2-amino-6-{4-[(5-chlorofuran-2-yl)methyl]piperazin-1-yl}-3,4-dihydropyrimidin-4-one
N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]-1-[(2-methylpyrimidin-5-yl)methyl]piperidine-3-carboxamide
1-cycloheptyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-6-oxopiperidine-3-carboxamide
N-(1-{1-[(2E)-3-(3-chlorophenyl)prop-2-enoyl]piperidin-4-yl}-2-phenylethyl)-N,1-dimethyl-1H-pyrazole-3-carboxamide
1-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(1H-pyrazol-1-yl)propan-1-one
(3aR,5R,6S,7aS)-2-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-octahydro-1H-isoindole-5,6-diol
3-({4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-1-yl}methyl)benzoic acid
5-{1-[(2E)-3-(4-chlorophenyl)prop-2-enoyl]piperidin-4-yl}-3-[2-(dimethylamino)ethyl]-5-(3-methylbutyl)imidazolidine-2,4-dione
(2R,3R,6R)-5-(1-ethyl-1H-pyrazole-3-carbonyl)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-(5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
9-(3-hydroxy-2-methylbenzoyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)azepan-4-amine
2-methyl-5-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,3-benzothiazole
3-{2-[3-(3-fluorophenoxymethyl)piperidin-1-yl]-2-oxoethyl}-3-(3-methoxyphenyl)-1-methylpyrrolidine-2,5-dione
4-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-[(3-methyl-1H-pyrazol-4-yl)methyl]piperazine
1-[(1S,5R)-6-[4-(difluoromethoxy)benzenesulfonyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
3-butyl-1-methyl-4-[(1-propyl-1H-imidazol-2-yl)methyl]piperazin-2-one
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-(2-hydroxyethyl)-N-(propan-2-yl)acetamide
3-(1-methyl-1H-pyrrol-2-yl)-N-[(2-methylphenyl)(pyridin-4-yl)methyl]-1H-pyrazole-5-carboxamide
3-{5-[2-(methylsulfanyl)benzoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
N-{[2-(quinolin-3-yl)phenyl]methyl}propanamide
4-(4-chlorophenyl)-N-[2-(1,3-thiazol-4-yl)ethyl]butanamide
5-{1-[(3,5-dimethoxyphenyl)methyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
1-(3-chloro-5-fluorophenyl)-3-[(2S)-pyrrolidin-2-ylmethyl]urea
4-[1-(furan-2-ylmethyl)piperidine-3-amido]oxane-4-carboxylic acid
3-[2-(4-acetyl-1,4-diazepan-1-yl)-2-oxoethyl]-4-(naphthalen-2-ylmethyl)piperazin-2-one
5-cyclopropyl-N-methyl-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-N-[(1-methylpiperidin-3-yl)methyl]-1H-pyrazole-4-carboxamide
[(2-butyl-1H-imidazol-4-yl)methyl](2-methylpropyl)(pyridin-2-ylmethyl)amine
N-(2-{4-[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]-1H-1,2,3-triazol-1-yl}ethyl)-N-methylmethanesulfonamide
N-(3-cyclopentylpropyl)-5-(2,6-dimethylphenoxymethyl)-N-methyl-1,2-oxazole-3-carboxamide
3-[1-(1-benzothiophene-2-carbonyl)piperidin-3-yl]-1-(4-methylpiperazin-1-yl)propan-1-one
(4S)-4-(methoxymethyl)-3,3-dimethyl-1-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]piperidin-4-ol
5-ethyl-2-{1-[1-(furan-2-yl)ethyl]-1H-imidazol-2-yl}pyridine
2-{pyrazolo[1,5-a]pyridine-3-carbonyl}-1,2,3,4-tetrahydroisoquinolin-4-ol
N-cyclopentyl-2-{[(4-sulfamoylphenyl)methyl]amino}propanamide