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N-[2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)ethyl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-(1-carbamoylethyl)piperidine-4-carboxamide
5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-[2-(1H-pyrazol-1-yl)ethyl]pyridin-2-amine
2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(pyrazin-2-ylmethyl)acetamide
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1-[(4-fluorophenyl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
1-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-methyl-3-(1H-1,2,4-triazol-1-yl)propan-1-one
1-[2-(4-methoxyphenyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)piperidine-3-carboxamide
2-({4-[4-(morpholin-4-yl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)ethan-1-ol
4-(1H-imidazol-1-yl)-1-(3-methoxypyrazin-2-yl)piperidine-4-carboxylic acid
benzyl (1R,5R)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxylate
1-(pyrimidine-4-carbonyl)spiro[azepane-4,2'-chromene]
6-(3-chlorothiophene-2-carbonyl)-1-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-6-azaspiro[2.5]octane
2-({[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(2-hydroxyethyl)amino)ethan-1-ol
2-(2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}phenoxy)propanamide
N,N-diethyl-1-(2-{1-ethyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}acetyl)piperidine-3-carboxamide
N5-tert-butyl-N3-[(3-methoxyphenyl)methyl]-N3-methyl-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
9-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-3-(1,2-oxazole-5-carbonyl)-3-azaspiro[5.5]undecane
(5-{[({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)amino]methyl}furan-2-yl)methanol
3-{3-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propanoic acid
2-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-oxo-N-(propan-2-yl)acetamide
4-{[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(3S,5S)-1-cycloheptanecarbonyl-5-(ethylcarbamoyl)pyrrolidin-3-yl]-1H-pyrrole-3-carboxamide
2-(morpholin-2-yl)-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}acetamide
2-benzyl-8-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
3-(1-butyl-1H-imidazol-2-yl)-N-(4-ethoxyphenyl)piperidine-1-carboxamide
(1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-[(4-methoxyphenyl)methyl]piperidin-4-yl)methanol
N-[2-(methylsulfanyl)phenyl]-4-[4-(pyridin-2-yl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
N-(2-methoxyethyl)-3-({1-[(2,4,5-trimethylphenyl)methyl]piperidin-4-yl}oxy)benzamide
4-(1H-pyrazol-1-ylmethyl)-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-1-carboxamide
(2R,3S,6R)-5-(3-ethyl-1H-pyrazole-4-carbonyl)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-ethoxy-N-{2-[4-(hydroxymethyl)piperidin-1-yl]-5,6,7,8-tetrahydroquinazolin-5-yl}propanamide
3-[3-(3-chlorophenyl)pyrrolidin-1-yl]-5-(2-fluorophenyl)-1,2,4-triazine
1-{4-[(2-fluorophenyl)methyl]-1,4-diazepan-1-yl}-2-(3-hydroxypiperidin-1-yl)ethan-1-one
1-(furan-2-ylmethyl)-N-[2-(pyridin-4-yl)ethyl]piperidine-4-carboxamide
3-hydroxy-N-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]piperidine-1-carboxamide
1-{[(3R,4R)-4-(hydroxymethyl)-1-[2-(methylsulfanyl)pyridine-3-carbonyl]pyrrolidin-3-yl]methyl}piperidin-4-ol
methyl[(3-methyl-1H-indol-2-yl)methyl]{[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}amine
3-{2-[4-(1-hydroxypropyl)piperidin-1-yl]-2-oxoethyl}-3-(4-methoxyphenyl)-1-(3-methylbutyl)pyrrolidine-2,5-dione
N-{[3-(difluoromethoxy)phenyl]methyl}-4-(pyridin-3-yl)pyrimidin-2-amine
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-1H-indole-6-carboxamide
1-{[4-(difluoromethoxy)phenyl]methyl}-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
9-[(2S)-2-amino-2-cyclopropylacetyl]-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
7-cyclohexyl-2-(5-propyl-1,3,4-thiadiazol-2-yl)-2,7-diazaspiro[4.5]decan-6-one
2-{2-[1-(2-methylpropanoyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
4-(morpholin-4-yl)-N-{[4-(oxolan-2-ylmethoxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)benzamide
8-fluoro-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]quinoline-2-carboxamide
N-methyl-N-{1-[3-(prop-2-en-1-yloxy)benzoyl]pyrrolidin-3-yl}acetamide
N-cyclopropyl-1-[(3-methoxyphenyl)methyl]-5-(quinolin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]-1,2-oxazole-3-carboxamide
3-[(3R,4S)-4-(morpholin-4-yl)-1-(quinoline-3-carbonyl)piperidin-3-yl]propan-1-ol