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2-{4-[4-(2-chlorophenyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}pyridine-3-carboxamide
6-(1,3-benzothiazol-6-yl)-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
5-[1-(thiophen-3-ylmethyl)-1H-imidazol-2-yl]-2,1,3-benzoxadiazole
2-{4-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]morpholin-3-yl}-N-[3-(hydroxymethyl)phenyl]acetamide
2-{[2-(2,5-dimethylphenyl)ethyl]amino}-N-(2-fluoro-5-methylphenyl)acetamide
N-[2-(1H-imidazol-1-yl)ethyl]-N,2,6-trimethylquinoline-3-carboxamide
1-(5-fluoro-2-methylphenyl)-2-(oxolan-3-yl)-1H-imidazole
2-(2,5-dioxoimidazolidin-1-yl)-N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}acetamide
1-(4-ethylpiperazin-1-yl)-3-[1-(oxolane-3-carbonyl)piperidin-4-yl]propan-1-one
5-(4-fluorophenyl)-2-methyl-4-{1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}pyrimidine
2-(butylsulfanyl)-6-[3-(2-fluorophenoxy)azetidin-1-yl]pyrimidin-4-amine
{[2-methanesulfonyl-1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}(methyl)[1-(trimethyl-1H-pyrazol-4-yl)ethyl]amine
5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-2-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}pyridine
methyl 2-({1-[4-(cyclopentylcarbamoyl)phenyl]piperidin-4-yl}amino)acetate
1-{5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperidin-4-ol
1-(4-{7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decane-2-carbonyl}thiophen-2-yl)ethan-1-one
9-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one
2,6-dihydroxy-N-methyl-N-{[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}benzamide
(1R,5S)-3-[1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]-3,8-diazabicyclo[3.2.1]octane
2-{[(3R,5S)-5-[4-(adamantan-2-yl)piperazine-1-carbonyl]-1-[(4-methylphenyl)methyl]pyrrolidin-3-yl]sulfanyl}pyrimidine
(1S,6R)-9-{2-[(2-methylphenyl)sulfanyl]acetyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
5-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
2-[(2-chlorophenyl)methyl]-4-[(1-ethyl-1H-imidazol-2-yl)methyl]morpholine
N-[(5-fluoro-2-methylphenyl)methyl]-1-[(2-methoxyphenyl)methyl]-6-oxopiperidine-3-carboxamide
1-{3-[1-(6-methylpyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-oxopropyl}piperidin-2-one
N-[(4,6-dimethylpyridin-2-yl)methyl]-2-(2-fluorophenoxymethyl)-N-methyl-1,3-oxazole-4-carboxamide
2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]-1-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine
1-(3-oxo-3-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}propyl)azepan-2-one
3-methyl-5-propyl-N-(2,2,2-trifluoroethyl)-1-benzofuran-2-carboxamide
1-(4-phenylphenyl)-N-[2-(pyridin-4-yl)ethyl]piperidin-4-amine
2-[methyl(2-phenylethyl)amino]-N-(pyridin-3-ylmethyl)-2,3-dihydro-1H-indene-2-carboxamide
N-butyl-N-[(4-fluorophenyl)methyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
3-{2-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonan-3-yl]-2-oxoethyl}-3,4-dihydroquinazolin-4-one
3-(2,3-dihydro-1-benzofuran-5-ylmethyl)-9-methoxy-10-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
(3S,5R)-N3-(6-methylpyridin-3-yl)-N5-(pyrimidin-4-ylmethyl)piperidine-3,5-dicarboxamide
(2S,4R)-4-amino-N,N-diethyl-1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]pyrrolidine-2-carboxamide
4-[6-(1-cycloheptanecarbonylpiperidin-3-yl)pyrimidin-4-yl]morpholine
N-butyl-4-{[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N-(but-2-yn-1-yl)-1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-(furan-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-[(3-chlorophenyl)methyl]-N-[1-(naphthalen-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
(3aS,6aS)-2-cyclopentanecarbonyl-5-[2-(4H-1,2,4-triazol-4-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-[(4-hydroxyquinolin-2-yl)methyl]piperazine-1-sulfonamide
(1S,5R)-6-(2,5-dimethylbenzenesulfonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N-methyl-1-(propan-2-yl)piperidine-4-carboxamide
2-methyl-6-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-4H-pyran-4-one
N-[1-(2-{4-[(3-fluorophenyl)methyl]-3-oxopiperazin-1-yl}-2-oxoethyl)-1H-pyrazol-4-yl]pyridine-2-carboxamide
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-({[(3-methyl-1H-pyrazol-5-yl)methyl]amino}methyl)piperidin-2-one
N-[3-(1H-imidazol-1-yl)butyl]-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
3-{[4-({1,9-dioxaspiro[5.5]undecan-4-yl}amino)piperidin-1-yl]methyl}phenol
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-2-(2-propyl-1H-1,3-benzodiazol-1-yl)propanamide