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(2S)-2-(8-fluoro-4-oxo-3,4-dihydroquinazolin-3-yl)-3-methylbutanamide
2-(2H-1,3-benzodioxol-5-yloxy)-1-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}ethan-1-one
6-methyl-3-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
N,N-dimethyl-4-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperazine-1-sulfonamide
N-{1-oxa-8-azaspiro[4.5]decan-3-yl}pyrazine-2-carboxamide
2-(2,5-dimethylphenyl)-N-(1-methylpiperidin-4-yl)-N-(pyridin-3-ylmethyl)acetamide
1-[2-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-oxoethyl]imidazolidine-2,4-dione
6-{2-methyl-2,8-diazaspiro[4.5]decane-8-carbonyl}-1,2-dihydropyridin-2-one
3-hexyl-8-(6-methylpyridine-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-methanesulfonamido-5-({[(4-methoxynaphthalen-1-yl)methyl]amino}methyl)-N-phenylbenzamide
4-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1-(pyridin-4-ylmethyl)pyrrolidin-2-one
3-(2,3-dihydro-1H-inden-2-yl)-5-methyl-5-{1-[(2,4,5-trimethoxyphenyl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
(2S,4S)-4-(4,5,6,7-tetrahydro-1-benzothiophene-2-amido)pyrrolidine-2-carboxylic acid
2-(2-methoxyphenyl)-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]acetamide
2-{4-[3-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}-2-oxoacetamide
N-[(2,4-difluorophenyl)methyl]-1-[(4-fluorophenyl)methyl]-5-(2-methoxyacetamido)-1H-1,3-benzodiazole-7-carboxamide
4-fluoro-N-({1-[(5-methylfuran-2-yl)methyl]piperidin-3-yl}methyl)benzamide
4-{3-[(2,5-dimethylphenyl)methyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl}piperazin-2-one
N-(2-methoxyethyl)-N-[(5-methylthiophen-2-yl)methyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
N-[1-(furan-2-yl)ethyl]-9-methoxy-3-[2-(2-methoxyphenyl)acetyl]-N-methyl-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-{1-[(5-methylthiophen-2-yl)methyl]pyrrolidin-2-yl}-1,3-thiazole
1-[2-oxo-2-(3-propoxypiperidin-1-yl)ethyl]-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
5-[4-(4-methoxybenzoyl)piperazine-1-carbonyl]-2-methylpyrimidine
4-[1-(propane-2-sulfonyl)piperidin-3-yl]benzoic acid
2-(dimethylamino)-2-(2-fluorophenyl)-1-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}ethan-1-one
4-[(4-{[2-(hydroxymethyl)phenyl]methyl}piperazin-1-yl)methyl]benzoic acid
2-[4-(4-hydroxyphenyl)piperazine-1-carbonyl]-3,4-dihydroquinazolin-4-one
N-ethyl-4-({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)piperidine-1-carboxamide
N-(2-methyl-4-{5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-6-yl}phenyl)furan-2-carboxamide
ethyl 1-[(5-chlorothiophen-2-yl)methyl]-3-(2-methoxyethyl)piperidine-3-carboxylate
1-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(pyridin-2-ylsulfanyl)ethan-1-one
(3R,4R)-4-cyclobutyl-N-[(3-fluorophenyl)methyl]-4-hydroxy-3-methylpiperidine-1-carboxamide
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2,5-dimethyl-1,3-thiazole-4-carboxamide
2-(4-{4-azaspiro[2.5]octan-4-ylmethyl}phenyl)-6-[2-(1H-pyrazol-1-yl)ethyl]-3,4-dihydropyrimidin-4-one
N-[(4-chlorophenyl)methyl]-1-(1-cyclopropanecarbonylpiperidin-4-yl)piperidine-3-carboxamide
N,N-dimethyl-5-{[methyl({[4-(1H-pyrazol-1-yl)phenyl]methyl})amino]methyl}pyrimidin-2-amine
2-chloro-4-fluoro-N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)benzamide
1-[2-(dimethylamino)ethyl]-5-[4-(2-ethylphenyl)piperazine-1-carbonyl]piperidin-2-one
1-[2-(dimethylamino)ethyl]-5-(4-methyl-1H-imidazole-5-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
methyl 2-[1-(5,6-dimethylpyrimidin-4-yl)pyrrolidin-3-yl]acetate
4-(1-methyl-1H-pyrazole-4-carbonyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(4-ethylphenyl)methyl]-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
2-cyclopropyl-N-[1-(4-fluorophenyl)piperidin-4-yl]-1,3-benzoxazole-6-carboxamide
1-[(4-chlorophenyl)methyl]-N-[2-(1H-indol-1-yl)ethyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
N-[(1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}piperidin-3-yl)methyl]-1-phenylmethanesulfonamide
3-[3-(thiophen-3-yl)-1,2,4-oxadiazol-5-yl]-1H-indazole
2-ethyl-4-phenyl-9-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecane
4-benzyl-3-ethyl-1-(1-methyl-1H-pyrazole-5-carbonyl)-1,4-diazepan-5-one
2-amino-6-(1,3-dimethyl-1H-pyrazol-4-yl)-4-[4-(1H-pyrazol-1-ylmethyl)phenyl]pyridine-3-carbonitrile
N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-4-(quinoxalin-2-yl)morpholine-2-carboxamide