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4-(benzyloxy)-1-[1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperidine
(2S)-2-amino-1-[4-(2-aminopyrimidin-4-yl)piperidin-1-yl]-3-hydroxypropan-1-one
N-(3,5-dimethoxyphenyl)-3-{1-[3-(pyridin-3-yl)propanoyl]piperidin-3-yl}propanamide
1-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-2-(3-hydroxypiperidin-1-yl)ethan-1-one
5-(2H-1,3-benzodioxol-5-yl)-N-[3-(1H-imidazol-1-yl)-1-phenylpropyl]-1,2,4-triazin-3-amine
1-cyclopropyl-3-(4-methoxyphenyl)-3-{2-[4-(4-methoxyphenyl)piperazin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
ethyl 1-[(3-acetylphenyl)methyl]-4-[(4-chlorophenyl)methyl]piperidine-4-carboxylate
N-[(5-methylthiophen-2-yl)methyl]-6-oxo-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-2-hydroxypropanamide
2-(1,2-benzoxazol-3-yl)-N-{3-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}acetamide
2-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-yl]-N-(5-methyl-1,2-oxazol-3-yl)acetamide
2-{[({3-methoxy-2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amino]methyl}-3,4-dihydroquinazolin-4-one
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
3-benzyl-4-[5-(3-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]piperazin-2-one
3-(azocan-1-yl)-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]propanamide
1-(2,3-dihydro-1H-inden-2-yl)-4-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-1,4-diazepane
8-[(2-chlorophenyl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
5-(2-{3-oxo-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-4-yl}ethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-{[7-(4-fluorobenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}propane-1-sulfonamide
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2,2-dimethylpropanamide
(2S,4S)-4-amino-N-ethyl-1-[4-(1H-pyrazol-1-yl)benzenesulfonyl]pyrrolidine-2-carboxamide
7-(3-chlorophenyl)-4-[3-(pyridin-3-yl)propyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-{4-[(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]piperidine-1-carbonyl}-6-(propan-2-yl)-1,2-dihydropyridin-2-one
2-[3-oxo-9-(1,3-thiazole-4-carbonyl)-2,9-diazaspiro[5.5]undecan-2-yl]propanoic acid
4-(5-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl)morpholine
N-cyclopropyl-5-[(2-hydroxy-7-methylquinolin-3-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
2-cyclopropyl-5-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]pyrimidine
1-(diethylamino)-3-[5-({[3-(1H-imidazol-1-yl)propyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
5-oxo-1-[2-(pyridin-4-ylformamido)ethyl]pyrrolidine-3-carboxylic acid
N-(1-ethyl-1H-1,2,3-triazol-4-yl)-2-{4-[4-(1H-imidazol-1-ylmethyl)phenyl]-1H-pyrazol-1-yl}acetamide
5-benzenesulfonamido-N-(1,4-dioxan-2-ylmethyl)-1-ethyl-2-methyl-1H-1,3-benzodiazole-7-carboxamide
{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(1-methylpiperidin-3-yl)methyl]amine
2-(2,3-dihydro-1H-isoindol-2-yl)-1-[6-hydroxy-4-(2-hydroxyethyl)-1,4-diazepan-1-yl]ethan-1-one
N-benzyl-3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carboxamide
N-{[5,8-dimethoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-2-methyl-1,3-thiazole-4-carboxamide
1-ethyl-4-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidine-1-carbonyl]-1,2-dihydropyridin-2-one
N-[1-(4-chlorophenyl)-3-hydroxypropan-2-yl]-3-(4-hydroxyphenyl)-1H-pyrazole-5-carboxamide
2-{4-[(2,6-dimethoxyphenyl)methyl]-1-(3-methylbutyl)piperazin-2-yl}ethan-1-ol
5-{2-[2-(cyclopropylmethyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-[(4-{[1-(4-methylbenzoyl)piperidin-3-yl]methoxy}phenyl)methyl]morpholine
(1S,6R)-9-{1-methyl-3-phenyl-1H-thieno[2,3-c]pyrazole-5-carbonyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
N-[(3R,4S)-4-cyclopropyl-1-(furan-2-carbonyl)pyrrolidin-3-yl]-2-(5-methyl-1H-pyrazol-1-yl)acetamide
2-(4-fluorophenyl)-N-(3-methyl-1,2,4-thiadiazol-5-yl)-3-oxopiperazine-1-carboxamide
methyl 3-ethanesulfonamido-5-({imidazo[1,2-a]pyridin-2-ylformamido}methyl)benzoate
methyl (2S)-1-{2-[1-(3-methoxypropyl)-2,5-dioxo-3-phenylpyrrolidin-3-yl]acetyl}pyrrolidine-2-carboxylate
2-[4-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl]ethan-1-ol
N-[3-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)propyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
4-(4-hydroxybenzoyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-cyclopropyl-1-[(2-methoxyphenyl)methyl]-6-methyl-3-[4-(pyridin-2-yl)piperazine-1-carbonyl]-1,4-dihydropyridin-4-one