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2-[1-cyclopentyl-3-(3-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-N-methylacetamide
2-fluoro-N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-5-sulfamoylbenzamide
6-[(3-methoxyphenyl)methoxy]-4-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]-1-(2-phenylethyl)-1,4-diazepan-2-one
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]propanamide
N-[(5-fluoro-2-methylphenyl)methyl]-3-{5-[methoxy(phenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
[(5-methylthiophen-2-yl)methyl](prop-2-en-1-yl){[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}amine
2-{1-[(2-methyl-1H-imidazol-4-yl)methyl]piperidin-4-yl}-1,2,3,4-tetrahydroisoquinoline
4-[1-(1-benzothiophene-2-sulfonyl)piperidin-3-yl]morpholine
2-[2-({methyl[1-(1,3-thiazol-2-yl)ethyl]amino}methyl)-4-phenylphenoxy]-1-(piperidin-1-yl)ethan-1-one
{[5-(methoxymethyl)furan-2-yl]methyl}(methyl)({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine
N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-1-(2-methylpropyl)-5-oxopyrrolidine-3-carboxamide
1-ethyl-3-(3-hydroxyazetidine-1-carbonyl)-4,6-dimethyl-1,2-dihydropyridin-2-one
N-(3,4-dimethoxyphenyl)-1-[3-(morpholin-4-yl)benzoyl]piperidin-3-amine
3-(1-propyl-1H-pyrazole-5-carbonyl)-3,9-diazaspiro[5.5]undecane
methyl({[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}){[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}amine
N-[2-(7-{[4-(trifluoromethyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]oxolane-2-carboxamide
N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-3-(piperidin-4-ylmethyl)benzamide
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)-3-(pyrazin-2-yl)propanamide
4-(4-methanesulfonyl-1,4-diazepane-1-carbonyl)-6-methyl-1,2-dihydroquinolin-2-one
4-{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methoxy}-1H-indole
N-{4-[4-({1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}(methyl)amino)piperidin-1-yl]phenyl}-2-phenoxyacetamide
(1R,4S)-2-{2-[4-(trifluoromethoxy)phenyl]pyridine-3-carbonyl}-2-azabicyclo[2.2.1]heptane
5-(2-{[(3-methoxyphenyl)methyl]amino}ethyl)-1-(2-phenylpropyl)pyrrolidin-2-one
4-[(4-{2-[1-(2,3-dimethyl-1H-indole-5-carbonyl)piperidin-2-yl]ethoxy}phenyl)methyl]piperazine-1-carbaldehyde
2-{1-[(4-ethoxyphenyl)methyl]-4-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperazin-2-yl}ethan-1-ol
3-[2-(3-methoxyphenyl)ethyl]-1-[(2-methyl-1H-imidazol-4-yl)methyl]piperidine
4-(3,4-dimethylphenyl)-1-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-1H-1,2,3-triazole
3-(1,2-oxazolidin-2-yl)-N-[3-(3-phenylpropanamido)phenyl]propanamide
3-{5-[(2E)-but-2-en-1-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1-(4-hydroxypiperidin-1-yl)propan-1-one
ethyl 3-[(3-methoxyphenyl)methyl]-1-[2-(pyridin-4-ylsulfanyl)acetyl]piperidine-3-carboxylate
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]acetamide
1-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]-3-(3-hydroxy-1,2-oxazol-5-yl)propan-1-one
3-[N-benzyl-1-(1-cyclopentanecarbonylpiperidin-4-yl)formamido]propanamide
2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(quinolin-5-ylmethyl)acetamide
(1R,5R)-6-(3-acetylbenzoyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-4-(4-phenyl-1H-pyrazol-5-yl)piperidine
9-[(3-fluoro-2,4-dimethylphenyl)methyl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
N-benzyl-N-(cyclobutylmethyl)-1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
(2S)-N-{[5-methyl-7-(2-methylquinolin-6-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-oxopyrrolidine-2-carboxamide
[(4-ethynylphenyl)methyl](methyl)[1-(4-methylpyridin-2-yl)propan-2-yl]amine
(4aR,7aS)-1-(2-hydroxyethyl)-4-(3-methoxy-2-methylbenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[1-(2-hydroxyethyl)-1H-1,2,4-triazol-5-yl]-1-methyl-1,2-dihydroquinolin-2-one
N-[5-(6-methyl-9H-purin-9-yl)pyridin-2-yl]methanesulfonamide
methyl 6-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-2-(methylsulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-(4-chlorophenyl)-5-[1-(methoxymethyl)cyclobutanecarbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-(4-{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1,4-diazepan-1-yl)ethan-1-one
2-ethyl-4-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
2-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}-5-propylpyrimidine
{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})amine