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(3R)-1-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-ol
5-[2,2-bis(prop-2-en-1-yl)pyrrolidine-1-carbonyl]-1-(pyridin-2-ylmethyl)piperidin-2-one
1-(cyclohexylmethyl)-N-(2-methoxyethyl)-6-oxo-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-ethyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]acetamide
2-(4-chloro-1-methyl-1H-pyrrole-2-carbonyl)-7-(cyclobutylmethyl)-2,7-diazaspiro[4.5]decan-6-one
1-[4-(4-methoxyphenoxy)piperidin-1-yl]-3-(2-methyl-1H-imidazol-1-yl)propan-1-one
N-[(2-chloro-6-fluorophenyl)methyl]-N-cyclopropyl-5,6,7,8-tetrahydroquinoline-3-carboxamide
1-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}-2-methoxyethan-1-one
(1S,5R)-6-(cyclobutylmethyl)-3-[(3,4-dimethoxypyridin-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-(2-methoxyethyl)-N-methyl-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
methyl 3-[(2,5-dimethylphenyl)methyl]-7-oxo-9-(pyridin-4-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-(2,3-dihydro-1H-isoindol-2-ylmethyl)-7-methoxy-1,2-dihydroquinolin-2-one
1-[2-(4-chlorophenyl)ethyl]-6-oxo-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-[(3S,4R)-1-(2-ethylpyrimidine-5-carbonyl)-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
(3S,5S)-5-[(4-fluorophenyl)carbamoyl]-1-(3,3,3-trifluoropropyl)piperidine-3-carboxylic acid
(3aS,6aS)-2-(ethanesulfonyl)-5-[(4-ethoxyphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3,5-dimethyl-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1H-indole-2-carboxamide
N-({3-methoxy-4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)-3-(3-methyl-1H-pyrazol-1-yl)-N-[(3S)-2-oxoazepan-3-yl]propanamide
1-(3-methoxypropyl)-4-[6-(4H-1,2,4-triazol-4-yl)pyridine-2-carbonyl]piperazine
3-{2-[4-(3-chlorophenoxy)piperidin-1-yl]-2-oxoethyl}-3-(2-fluorophenyl)-1-methylpyrrolidine-2,5-dione
1-[(2R,3R)-3-[butyl(methyl)amino]-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-2-hydroxy-2-methylpropan-1-one
4-[(4-fluorophenyl)methyl]-1-[(2-methyl-1,3-oxazol-4-yl)methyl]piperidine
1-(1-methyl-1H-pyrrol-2-yl)-2-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethane-1,2-dione
(1S,4S)-2-{3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}-2-azabicyclo[2.2.1]heptane
2-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]benzonitrile
(2S,4R)-1-[(2-aminopyridin-3-yl)methyl]-N-methyl-4-[2-(2-oxo-1,3-oxazolidin-3-yl)acetamido]pyrrolidine-2-carboxamide
3-(1H-pyrazol-5-yl)-1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidine
N-[2-(1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)ethyl]acetamide
1-(cyclopentylmethyl)-4-[(2,3,4-trimethoxyphenyl)methyl]piperazine
1-[(2,6-difluorophenyl)methyl]-N-[1-(2-methoxyphenyl)ethyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
4-(1-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}piperidin-3-yl)morpholine
2-[4-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)piperidin-1-yl]pyridine-4-carbonitrile
1-(furan-2-ylmethyl)-N-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]piperidine-3-carboxamide
N-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
2-[(3-chlorophenyl)methyl]-N-[2-(1H-pyrazol-4-yl)ethyl]-1,3-benzoxazole-6-carboxamide
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[2-(1H-imidazol-1-yl)-1-phenylethyl]acetamide
1-[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
5-chloro-N-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)furan-2-carboxamide
N-(6-methylpyridin-3-yl)-2,3-dihydro-1,4-benzodioxine-6-carboxamide
1-[4-({3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}methyl)thiophen-2-yl]ethan-1-one
7-(3,6-dimethylpyrazin-2-yl)-4-[(4-hydroxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-(2-fluorophenyl)-1-{9-methyl-3,9-diazaspiro[5.6]dodecan-3-yl}propan-1-one
2-(3-methoxyphenyl)-1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidine
(3R,4R)-3-hydroxy-N-(2-methylphenyl)-4-{[2-(morpholin-4-yl)ethyl]amino}pyrrolidine-1-carboxamide
methyl 5-(cyclobutylamino)-3-acetamido-1-[2-(1H-indol-3-yl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
5-[3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-3-(propan-2-yl)-1,2-oxazole
1-(2-phenoxyethyl)-4-[(2-phenyl-1H-imidazol-4-yl)methyl]piperazine
(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-7-{[(4-methoxyphenyl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}[1-(2-chlorophenyl)ethyl]amine
3-{2-[1-(2-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-oxoethyl}-1,3-oxazolidin-2-one