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3-(4-methylpiperazin-1-yl)-6-{[1-(pyrrolidin-1-yl)hex-5-en-2-yl]oxy}pyridazine
N-[1-(4-methoxyphenyl)-4-(morpholin-4-yl)-1H-indazol-3-yl]-1-methylcyclopropane-1-carboxamide
3-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-[(4-methoxyphenyl)methyl]benzamide
1-{7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-(pyridin-2-ylsulfanyl)ethan-1-one
N-[(3-chlorophenyl)methyl]-1-(2-cyclopropyl-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl)piperidine-4-carboxamide
N5,N5-dimethyl-N6-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
4-(3-chlorobenzoyl)-7-(2,6-dimethoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(4-benzyl-2-oxopyrrolidin-1-yl)-N-methyl-N-(thian-4-yl)acetamide
2-(dimethylamino)-N-[2-methyl-3-({[2-(1-methyl-1H-pyrazol-5-yl)ethyl]carbamoyl}amino)phenyl]acetamide
7-{1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
4-[1-(4-fluorobenzoyl)piperidin-3-yl]-5-(4-fluorophenyl)-2-methylpyrimidine
2-[4-({2-[2-(dimethylamino)ethyl]piperidin-1-yl}methyl)phenyl]ethan-1-amine
(1R,3S)-3-{[(5-chloro-2-ethoxyphenyl)methyl](methyl)carbamoyl}cyclopentane-1-carboxylic acid
1-(2-chlorophenyl)-4-[2-(2-hydroxyphenoxy)acetyl]-5-methylpiperazin-2-one
1,5-dimethyl-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]-1H-indazole-3-carboxamide
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(1-ethyl-1H-imidazol-2-yl)methyl]acetamide
N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]cyclopentanecarboxamide
2-[4-(2H-1,3-benzodioxol-5-yl)-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-(cyclopropylmethyl)acetamide
N-({2-[2-(2-cyclopentylacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-4,5,6,7-tetrahydro-2-benzothiophene-1-carboxamide
(3aS,6aS)-2-cyclohexyl-5-[(dimethyl-4H-1,2,4-triazol-3-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
propan-2-yl 4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
5-[(3-methoxyphenyl)methyl]-3-methyl-5-[1-(naphthalen-2-ylmethyl)piperidin-4-yl]imidazolidine-2,4-dione
N-(propan-2-yl)-7-{[2-(pyridin-2-yl)ethyl]sulfamoyl}-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
4-(4-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}phenyl)-4H-1,2,4-triazole
({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl){[2-(2-methylphenyl)pyrimidin-5-yl]methyl}amine
(2S,4S)-4-amino-N-methyl-1-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanoyl]pyrrolidine-2-carboxamide
2-(1H-1,3-benzodiazol-1-yl)-N-{[5-methyl-7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
3-({2-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]acetamido}methyl)-4-methylbenzoic acid
methyl 2-({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}formamido)acetate
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-2-(methylamino)pyridine-4-carboxamide
2-(4-chlorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]ethan-1-one
4-{[4-(4,5-dimethyl-6-oxo-1,6-dihydropyrimidin-2-yl)phenyl]methyl}-N,N-dimethylpiperazine-1-carboxamide
1-{3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide
5-(1H-1,2,3-benzotriazole-5-carbonyl)-N-cyclopropyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]-1-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonan-3-yl]ethan-1-one
3-{[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-4-methyl-1,2,5-oxadiazole
1,3-dimethyl-N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-[2-(dimethylamino)ethyl]-8-fluoro-N-[(5-methylthiophen-2-yl)methyl]quinoline-2-carboxamide
3-(dimethylamino)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]benzamide
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
2-[(4S)-4-hydroxy-3,3,4-trimethylpiperidin-1-yl]-N-(1-methyl-1H-pyrazol-3-yl)acetamide
1-{7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-(1H-pyrazol-1-yl)ethan-1-one
N-[2-(1H-1,2,3-benzotriazol-1-yl)ethyl]-2,4-dimethylpyrimidine-5-carboxamide
6-methyl-N-[1-(morpholine-4-carbonyl)piperidin-4-yl]imidazo[1,2-a]pyridine-2-carboxamide
1-{3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}-2-{[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}ethan-1-one
1-(benzenesulfonyl)-4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-5-one
(4aS,8aR)-6-(1-methyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-1-(3-methylbutyl)-decahydro-1,6-naphthyridin-2-one
3-{[1-(2-fluoro-4-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-pyrazole