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1-(2H-1,3-benzodioxol-5-yl)-5-[(4,5-dimethyl-1H-imidazol-1-yl)methyl]-1H-1,2,4-triazole
4-({2-[1-(4-methoxybenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
4-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
N,N-diethyl-1-{3-[2-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-2-yl]propanoyl}piperidine-3-carboxamide
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-2-hydroxy-2-phenylpropanamide
1-{4-[7-(1,3-benzothiazol-2-yl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]piperidin-1-yl}ethan-1-one
8-(2-fluoro-3-methoxyphenyl)-2-(morpholin-4-yl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
N-({8-[(5-chloro-2-hydroxyphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-1,3-dimethyl-1H-pyrazole-5-carboxamide
1-[9-methoxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-(2-methylpropyl)-4-[(naphthalen-1-ylmethyl)amino]pyrrolidine-2-carboxamide
methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl][(1-methyl-1H-indol-2-yl)methyl]amine
3-chloro-N-[2-(dimethylamino)ethyl]-4-({1-[3-(1-methylcyclopropyl)propanoyl]piperidin-4-yl}oxy)benzamide
N-{[2-fluoro-3-(trifluoromethyl)phenyl]methyl}-1-(methoxymethyl)cyclopropane-1-carboxamide
4-{4-[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]butyl}morpholine
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}acetamide
4-(hydroxymethyl)-1-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)piperidin-4-ol
methyl 8-(1-benzofuran-2-ylmethyl)-1-(2-methoxyethoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
1,9-dimethyl-4-[(3-phenylphenyl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[2-(1-benzylpiperidin-4-yl)ethyl]-6-(methoxymethyl)pyrimidin-4-amine
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(3-fluorophenoxymethyl)piperidine
1-(4-{[4-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
5-(cyclopentylamino)-1-ethyl-N-(furan-3-ylmethyl)-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-{[(1-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)oxy]methyl}pyridine
2-methyl-N-(1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-1H-1,3-benzodiazole-5-carboxamide
N-cyclopropyl-1-[2-(4-methoxyphenyl)ethyl]-5-(pyridine-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(2R,3R,6R)-3-(3-methoxyphenyl)-5-(3-methylbenzoyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-methyl-5-{4-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
1-{3-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]propyl}-1,2,3,4-tetrahydroquinoline
2-tert-butyl-4-hydroxy-N-methyl-N-{[2-(2-methylpropoxy)phenyl]methyl}pyrimidine-5-carboxamide
1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-cyclopentylpropan-1-one
2-methyl-4-{3-[4-(6-methylpyridin-2-yl)piperazine-1-carbonyl]phenyl}butan-2-ol
10-[3-(butan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraen-9-one
2-(4-chloro-3-methyl-1H-pyrazol-1-yl)-N-methyl-N-(quinolin-5-ylmethyl)acetamide
1-(5-chloropyridin-2-yl)-4-{3-[(3-methoxyphenyl)methyl]-1,2-oxazole-5-carbonyl}piperazine
7-[(2-butyl-1H-imidazol-4-yl)methyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}[4-(pyridin-2-yl)butyl]amine
1-(2-{[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]amino}-4-methylpyrimidin-5-yl)ethan-1-one
1,9-dimethyl-4-(2-phenylpyrimidine-5-carbonyl)-1,4,9-triazaspiro[5.5]undecane
(3S)-N-tert-butyl-2-{[2-(methylamino)-1,3-thiazol-4-yl]methyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
5-oxo-1-(pyridin-4-ylmethyl)-N-[(1r,4r)-4-hydroxycyclohexyl]pyrrolidine-3-carboxamide
N-methyl-N-[2-(morpholin-4-yl)ethyl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
3-(4-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}piperazin-1-yl)-1λ6-thiolane-1,1-dione
ethyl 2-{1-[5-(3,4-difluorophenoxymethyl)-1,2-oxazole-3-amido]cyclohexyl}acetate
2-[4-(4-methylphenyl)-3-oxopiperazine-1-carbonyl]thiophene-3-sulfonamide
N-(1,4-dioxan-2-ylmethyl)-1-(6-fluoro-4-methylquinazolin-2-yl)piperidine-4-carboxamide
8-[2-(4-methylphenoxymethyl)furan-3-carbonyl]-5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine
(2S,4R)-N-[2-(2-fluorophenyl)ethyl]-1-(2-methylpropyl)-4-{[(5-methylthiophen-2-yl)methyl]amino}pyrrolidine-2-carboxamide
4-(2-chlorobenzoyl)-2-[(4-methoxyphenyl)methyl]morpholine
2-amino-4-[2-(dimethylamino)-1,3-thiazol-5-yl]-6-(2,5-dimethylthiophen-3-yl)pyridine-3-carbonitrile
2-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carbonyl]pyridin-4-amine