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(1R,9aR)-1-{[4-hydroxy-4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]methyl}-octahydro-1H-quinolizin-1-ol
1-[2-(piperidin-1-yl)ethyl]-6-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}-3-(pyridin-4-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-4-(piperidin-1-ylmethyl)benzamide
3-(3-{7-methylthieno[3,2-d]pyrimidin-4-yl}phenyl)-1H-pyrazole
3-[(1-ethyl-1H-1,3-benzodiazol-2-yl)sulfanyl]-1-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]propan-1-one
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]piperazine
4-(1,3-thiazol-2-ylmethyl)-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
(3aS,6aR)-5-[(5-methylfuran-2-yl)methyl]-3-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
(2R,3S,6R)-5-[1-(methoxymethyl)cyclobutanecarbonyl]-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(2S,4R)-N,N-diethyl-4-[2-(propan-2-yloxy)acetamido]-1-(1H-pyrazole-3-carbonyl)pyrrolidine-2-carboxamide
5-{4-[(4-cyclopentyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}-1H-indole
2-(2-hydroxyphenyl)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}acetamide
1-{2-[4-(1-methylpiperidin-4-yl)morpholin-2-yl]ethyl}-3-(propan-2-yl)urea
1-(4-chlorophenyl)-N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]cyclopropane-1-carboxamide
5-(2-chloro-3-methylbenzoyl)-1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-[1-(2-chlorophenyl)ethyl]propanamide
4-{[3-(3,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}-1-methylpiperazine-2-carboxylic acid
3-{2-[(2-fluoro-5-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-(pyridin-3-ylmethyl)propanamide
3-[(2-{1-[1-(propan-2-yl)-1H-pyrrole-2-carbonyl]piperidin-3-yl}-1H-imidazol-1-yl)methyl]pyridine
1-[(2-fluorophenyl)methyl]-4-{[2-(2-methoxyethyl)pyrimidin-5-yl]methyl}-1,4-diazepane
4-{2,2-dimethyl-3-[2-(1,3-thiazol-2-yl)piperidin-1-yl]propyl}morpholine
1-(2-fluorophenyl)-4-[1-(4-methoxy-3-methylbenzoyl)piperidin-3-yl]piperazine
[1-(1-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)ethyl]dimethylamine
N-[(2-fluorophenyl)methyl]-3-{1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}propanamide
9-[(2S)-2-aminobutanoyl]-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrol-1-ylmethyl]-6-methylimidazo[1,2-a]pyridine
N-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-1-methyl-N-(pyridin-4-ylmethyl)piperidin-4-amine
2-{[2-(dimethyl-1,3-thiazol-5-yl)acetamido]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
N-[(4-methyl-1H-imidazol-2-yl)methyl]-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
(4aR,7aS)-N,N-dimethyl-6,6-dioxo-4-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
3-{1,2-dihydrospiro[indole-3,4'-piperidine]-1'-ylmethyl}pyridin-2-amine
1-(1-{1-[(2-chloro-6-fluoro-3-methoxyphenyl)methyl]piperidin-4-yl}ethyl)-4-methylpiperazine
ethyl 1-benzyl-5-[(4-hydroxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-{4-[(1H-indol-2-ylmethyl)amino]piperidin-1-yl}benzamide
N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2,3-dihydro-1-benzofuran-7-carboxamide
5-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenoxy]-1-azabicyclo[3.2.1]octane
1-cyclohexanecarbonyl-N-(furan-2-ylmethyl)-N-(1-hydroxy-2-methylpropan-2-yl)pyrrolidine-2-carboxamide
2-({4-[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl]-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)ethan-1-ol
[(3R,4S)-1-[(2-ethylphenyl)methyl]-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
3-{[2-(dimethylamino)-2-(4-methylphenyl)acetamido]methyl}-1,2,4-oxadiazole-5-carboxamide
N-({8-benzyl-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-3-chloro-4-fluorobenzamide
1-(cyclopropylmethyl)-N-methyl-5-(quinoline-2-carbonyl)-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-({6-oxo-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-7-yl}methyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonitrile
[5-(1-{[4-(hydroxymethyl)phenyl]methyl}-4-phenyl-1H-imidazol-5-yl)furan-2-yl]methanol
1-ethyl-8-{[2-(furan-2-yl)phenyl]methyl}-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(3-methylbutyl)-3-(2-oxo-2-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-yl}ethyl)piperazin-2-one
1-(cyclohex-3-en-1-ylmethyl)-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
2-({[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}(benzyl)amino)ethan-1-ol
6-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}pyrazine-2-carboxamide
N-ethyl-3-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]-N-[(2E)-3-phenylprop-2-en-1-yl]propanamide