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2-[({5-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]furan-2-yl}methyl)sulfanyl]pyrimidine
2,4-difluoro-6-[3-(1H-pyrazol-3-yl)phenyl]phenol
N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-1H-imidazole-2-carboxamide
N-(1-cycloheptylpiperidin-3-yl)-3,5-dimethylfuran-2-carboxamide
1-(4-{4-[(8-methoxyquinolin-2-yl)methyl]piperazin-1-yl}phenyl)ethan-1-one
1-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-2-(1H-imidazol-1-yl)ethan-1-one
4-[1-(2-cyclohexylethyl)-1H-1,2,3-triazole-4-carbonyl]-1-[(3,4-dimethylphenyl)methyl]piperazin-2-one
N-[(3S)-1-benzylpyrrolidin-3-yl]-N-methyl-2-(pyridin-4-yl)pyrimidine-5-carboxamide
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl](methyl)[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amine
3-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidine-1-carbonyl]-1H-indazole
(2E)-1-{3-[4-(3-chlorophenyl)piperazin-1-yl]piperidin-1-yl}-3-(pyridin-4-yl)prop-2-en-1-one
3-cyclopentyl-N-{[5-methyl-2-(2-phenylmethanesulfonamidophenyl)-1,3-oxazol-4-yl]methyl}propanamide
1-[3-(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)-3-oxopropyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-[1-(3-methylphenyl)-1H-pyrazol-4-yl]pyrimidin-2-amine
4,4-difluoro-N-[4-(propylsulfanyl)phenyl]piperidine-1-carboxamide
4-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]acetamido}-N-phenylpiperidine-1-carboxamide
N-({7-[(2,4-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-methoxybenzamide
6-methyl-5-[5-(4,5,6,7-tetrahydro-2-benzothiophen-1-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
3-[1-(2,6-dimethylquinolin-4-yl)-N-methylformamido]-3-phenylpropanoic acid
1-{5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperidin-3-ol
3-chloro-4-({1-[(2-hydroxy-6-methoxyphenyl)methyl]piperidin-4-yl}oxy)-N-(2-methoxyethyl)benzamide
2-[(5-methylpyrazin-2-yl)methyl]-8-[2-(morpholin-4-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-N'-phenylethanediamide
2-(methylsulfanyl)-N-[(3R,4S)-1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}-4-propylpyrrolidin-3-yl]acetamide
2-benzyl-N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methyl-1,3-thiazole-4-carboxamide
9-{[2-(difluoromethoxy)phenyl]methyl}-3,9-diazaspiro[5.6]dodecane
2-tert-butyl-6-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
2-({3-[4-(2-methylpropyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)-1H-indole
N-{1-[1-(3-methylphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]ethyl}methanesulfonamide
3-{2-[(2R,3R,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
2-(1H-imidazol-1-yl)-1-{5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethan-1-one
2-(3-methoxypropyl)-8-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2,5-dimethyl-N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)furan-3-carboxamide
2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-1-[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]ethan-1-one
(3R,4S)-1-{[5-(3-fluorophenyl)-1,3,4-oxadiazol-2-yl]methyl}-3,4-dimethylpiperidin-4-ol
ethyl 4-{1-[(5-chlorothiophen-2-yl)methyl]piperidin-3-yl}piperazine-1-carboxylate
3-[3-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)phenyl]-5-methyl-1,2,4-oxadiazole
1-{[5-(4-ethoxyphenyl)furan-2-yl]methyl}azepan-4-ol
1-(2,3-difluoro-6-methoxybenzoyl)-4-[1-(pyrrolidin-1-yl)ethyl]piperidine
[(3R,4R)-4-[(dimethylamino)methyl]-1-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-yl]methanol
N-cyclopropyl-4-methoxy-2-[(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-4-yl)oxy]benzamide
3-methyl-5-{2-oxo-2-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-oxo-4-[3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]butanamide
1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-2-methyl-N-(oxolan-2-ylmethyl)-1,3-thiazole-4-carboxamide
2-tert-butyl-6-({[(1,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)phenol
3-methoxy-1-[2-(4-methoxy-4-phenylpiperidin-1-yl)-2-oxoethyl]-1,2-dihydropyridin-2-one
methyl 3-[2-(2,3-difluorophenyl)acetyl]-7-oxo-9-[2-(pyridin-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-(furan-3-yl)-1-[(2,3,4-trimethoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one