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6-(2-methylpropyl)-4-[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1,2-dihydropyrimidin-2-one
(3-{[ethyl({[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl})amino]methyl}-2,4,6-trimethylphenyl)methanol
methyl 1-[(3R,5S)-1-(pyridin-3-ylmethyl)-5-({[3-(trifluoromethyl)phenyl]methyl}carbamoyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
2-{3-[6-amino-5-cyano-4-(furan-3-yl)pyridin-2-yl]-1H-indol-1-yl}acetic acid
(1R,5R)-10-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-3,7,10-triazatricyclo[3.3.3.01,5]undecane-2,6-dione
1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-3-{2-methyl-[1,2,4]triazolo[1,5-a]pyridin-8-yl}urea
N-[2-(4-chlorophenoxy)ethyl]-N-(furan-2-ylmethyl)-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
2-amino-4-(1,5-dimethyl-1H-pyrazol-4-yl)-6-[4-fluoro-2-(trifluoromethyl)phenyl]pyridine-3-carbonitrile
N-methyl-5-(3-methyl-1,2,4-oxadiazol-5-yl)-N-(1,3-thiazol-2-ylmethyl)pyridin-2-amine
methyl 3-acetamido-5-[(4-hydroxy-4-methylpentan-2-yl)amino]-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(1R,9aR)-1-[2-(4-methoxy-6-methylpyrimidin-2-yl)phenoxymethyl]-octahydro-1H-quinolizine
3-(2-{2-azabicyclo[2.2.1]heptan-2-yl}-2-oxoethyl)-3-(2-chlorophenyl)-1-(2-methoxyethyl)pyrrolidine-2,5-dione
2-[5-cyclopropyl-4-(4-methylpiperazine-1-carbonyl)-1H-pyrazol-1-yl]-5-methyl-4-(thiophen-2-yl)pyrimidine
4-({2-oxo-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-3-yl}methyl)-1λ6-thiomorpholine-1,1-dione
N-[1-(cyclohexylmethyl)piperidin-3-yl]-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
(2S,4S)-1-(cyclohexylmethyl)-4-[(4,6-dimethylpyrimidin-2-yl)sulfanyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-(2-fluorophenyl)-1-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[(2,2-dimethyl-1-phenylcyclopropyl)methyl]methylamine
3-(3-chloro-4-fluorophenyl)-N,N,1-trimethyl-1H-1,2,4-triazol-5-amine
N-{1-[(4-methoxy-2,3,6-trimethylphenyl)methyl]piperidin-3-yl}acetamide
1-[3-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)phenyl]-1H-1,2,4-triazole
1-(4-{1-[methyl(pyridin-3-ylmethyl)amino]-2-phenylethyl}piperidin-1-yl)-3-(2-methyl-1H-1,3-benzodiazol-1-yl)propan-1-one
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(pyridine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-7-fluoroquinazolin-4-amine
4-(4-{[(3S,4S)-3,4-bis(hydroxymethyl)pyrrolidin-1-yl]methyl}phenyl)-2-methylbutan-2-ol
2-amino-N-cyclopropyl-3-ethyl-N-{[4-(methylsulfanyl)phenyl]methyl}-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperazin-2-yl}ethan-1-ol
2-(1-ethyl-2,4-dioxo-8-{[4-(pyrrolidin-1-yl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decan-3-yl)acetamide
N-cyclopropyl-3-[5-(2,3-dihydro-1-benzofuran-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanamide
5-methyl-5-{1-[(2E)-2-methylbut-2-en-1-yl]piperidin-4-yl}-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
2-ethyl-7-(2-methoxybenzamido)-1-methyl-N-(3-methylbutyl)-1H-1,3-benzodiazole-5-carboxamide
6-methyl-2-[(2-methylphenyl)methyl]-4-oxo-N-[(3S)-2-oxoazepan-3-yl]-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
2-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-2,3-dihydro-1H-isoindole
(3S,5R)-5-[(4-fluorophenyl)carbamoyl]-1-[(3-hydroxyphenyl)methyl]piperidine-3-carboxylic acid
4-fluoro-N-{3-[4-(1H-imidazol-2-yl)piperidin-1-yl]-3-oxopropyl}benzamide
3-(2-aminopyridin-4-yl)-5-[2-(piperidin-2-yl)ethyl]phenol
N-(3-butanamidophenyl)-2-(1H-imidazol-4-ylmethyl)-3-oxopiperazine-1-carboxamide
2-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]-6-chloroimidazo[1,2-a]pyrimidine
N-({5-[(5-fluoro-2-methoxyphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)methanesulfonamide
[(4-fluorophenyl)methyl]({[2-methanesulfonyl-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl})methylamine
1-ethyl-8-(1-hydroxypropan-2-yl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-methyl-N-{1-[1-(pyrimidin-2-ylmethyl)-1,2,5,6-tetrahydropyridin-3-yl]propyl}propanamide
3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-4-({8-methyl-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)-1H-pyrazole
5-({2-[2-(dimethylamino)ethyl]morpholin-4-yl}methyl)-N,N-dimethyl-1,3-thiazol-2-amine
1-(2,3-dihydro-1H-inden-5-yl)-4-{4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}piperidine
[5-({1-[5-fluoro-4-(pyrrolidin-1-yl)pyrimidin-2-yl]piperidin-4-yl}methyl)-4-methyl-4H-1,2,4-triazol-3-yl]methanol
(5-{1-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-1H-imidazol-2-yl}furan-2-yl)methanol
1-{[4-(1H-imidazol-1-yl)phenyl]methyl}-4-(1,2,4-oxadiazol-3-yl)piperidine
1-methyl-N-[2-(N-methylmethanesulfonamido)ethyl]-1H-indole-3-carboxamide
4-benzamido-N-[1-methyl-3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine-1-carboxamide