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{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}({[4-(methylsulfanyl)phenyl]methyl})amine
6-(methoxymethyl)-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)pyridine-2-carboxamide
N-(1-{7-[(5-ethylfuran-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-methoxypropanamide
1-[1-(furan-2-ylmethyl)piperidine-3-carbonyl]-4-(pyrimidin-2-yl)-1,4-diazepane
methyl 4-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}piperazine-1-carboxylate
2-(1-{1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-2-yl)-5-fluoro-1H-1,3-benzodiazole
5-{[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-N-(propan-2-yl)pyrimidin-2-amine
4-{[2-(2-hydroxyethyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]methyl}benzamide
N-ethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)furan-3-carboxamide
2-chloro-4-fluoro-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]benzamide
N-benzyl-2-[4-(4-{[3-(1H-pyrazol-1-yl)propyl]amino}piperidin-1-yl)phenyl]acetamide
4-[1-(2-phenylethyl)pyrrolidin-3-yl]-1-(1,3-thiazole-4-carbonyl)piperidine
2-(2-{[5-(naphthalen-2-yl)-1,2,4-triazin-3-yl]amino}ethyl)-6-phenyl-2,3-dihydropyridazin-3-one
N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-1-benzofuran-5-carboxamide
4-{1-[2-amino-6-(propan-2-yl)pyrimidine-4-carbonyl]piperidin-3-yl}benzoic acid
1-{4-[1-(cyclopropylmethyl)-1,2,3,6-tetrahydropyridin-4-yl]-1H-pyrazol-1-yl}butan-2-ol
2-{methyl[2-(1H-pyrazol-4-yl)ethyl]amino}-N-[1-(4-methylphenyl)ethyl]acetamide
2-{3-[(3,3-difluoropiperidin-1-yl)methyl]phenyl}-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
8-{6-methylthieno[2,3-d]pyrimidin-4-yl}-2,8-diazaspiro[4.5]decan-3-one
2-[2-(trifluoromethyl)morpholin-4-yl]quinoxaline
2-amino-6-(furan-2-yl)-4-(1-methyl-3-phenyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
N-cyclopropyl-2-(thiophen-3-yl)-N-{[5,6,7-trimethoxy-2-(2-methylphenyl)quinolin-3-yl]methyl}acetamide
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-(pyridin-4-ylmethyl)piperazin-2-yl}ethan-1-ol
1-[1-(cyclohexylmethyl)-1H-1,2,3-triazole-4-carbonyl]azepane
(2S)-2-(2-{1-[(4-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}acetamido)propanamide
2-(5-fluoro-2-methyl-1H-indol-3-yl)-1-[4-(thian-4-yl)piperazin-1-yl]ethan-1-one
(4-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}morpholin-2-yl)methanamine
4-benzyl-3-ethyl-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1,4-diazepan-5-one
1-(2-chlorophenyl)-2-{[4-(methylamino)pyrimidin-2-yl]amino}ethan-1-ol
1-acetyl-N-[4-(2-fluorophenoxy)phenyl]piperidine-4-carboxamide
(3-{2-[1-(5-fluoropyridine-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
(4-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}phenyl)methanamine
2-(3-hydroxypropyl)-9-(2-methoxy-4-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
2-{1-[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}pyridine
1-ethyl-3-methyl-4-{5-methyl-[1,2,4]triazolo[4,3-a]pyridin-3-yl}-1H-pyrazole
1-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)-4-(hydroxymethyl)azepan-4-ol
7-(cyclopropylmethyl)-2-[(2,5-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
1-ethyl-N-(3-phenyl-1,2,4-thiadiazol-5-yl)-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carboxamide
1-(cyclobutylmethyl)-3-({[(dimethyl-1,3-thiazol-2-yl)methyl]amino}methyl)-3-hydroxypiperidin-2-one
N2,N4,N4,5-tetramethyl-N2-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}pyrimidine-2,4-diamine
1-ethyl-2-{[1-(4-fluoro-3-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-imidazole
1-benzyl-4-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)piperazine
3-(2-methoxybenzoyl)-1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidine
5-(propane-1-sulfonyl)-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-[2-(pyridin-3-ylformamido)ethyl]propanamide
5-methyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-1-propyl-1H-pyrazole-4-carboxamide
N-methyl-N-[4-(morpholin-4-yl)butyl]-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamide
2-methoxy-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)acetamide
N-cyclopropyl-N-[(3-hydroxyphenyl)methyl]-3-methyl-3-phenylbutanamide
N-[2-(4-methoxyphenyl)ethyl]-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide