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N-methyl-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-4-(1H-1,2,4-triazol-1-yl)butanamide
2-(3,5-dimethoxyphenyl)-4-(piperidine-1-carbonyl)pyridine
[1-(5-chlorothiophene-2-carbonyl)-3-ethylpiperidin-3-yl]methanol
5-methyl-N-{[1-methyl-5-(trifluoromethyl)-1H-1,3-benzodiazol-2-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
1-(1-{1-[(2,3-difluoro-4-methoxyphenyl)methyl]piperidin-4-yl}ethyl)-4-methylpiperazine
(4aS,8aR)-1-(3-methoxypropyl)-6-(6-oxo-1,6-dihydropyridazine-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
N-[1-(cyclohexylmethyl)piperidin-3-yl]-3-(2-oxopiperidin-1-yl)propanamide
2-amino-4-ethyl-N-[3-(pyridin-2-yl)propyl]-1,3-thiazole-5-carboxamide
1,3-dimethyl-5-{2-oxo-2-[4-(2-phenylethyl)piperazin-1-yl]ethyl}imidazolidine-2,4-dione
N-{1-[(4-phenoxyphenyl)methyl]piperidin-4-yl}methanesulfonamide
6-(4-hydroxypiperidin-1-yl)-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}pyridine-3-carboxamide
1-(3-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}phenyl)ethan-1-one
5-methoxy-N-methyl-4-oxo-N-[1-(pyridin-2-yl)propyl]-1,4-dihydropyridine-2-carboxamide
5-[2-methoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]-1-azabicyclo[3.2.1]octane
2-(3,5-dimethoxyphenyl)-2-[methyl(pyridin-2-ylmethyl)amino]acetic acid
7-chloro-N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N,3,5-trimethyl-1-benzofuran-2-carboxamide
2-methyl-6-({3-[3-(1-methyl-1H-pyrazol-4-yl)phenyl]-1H-pyrazol-1-yl}methyl)pyridine
N-methyl-3-(1H-pyrazol-1-ylmethyl)-N-[1-(1,3-thiazol-5-yl)ethyl]benzamide
2-({2-oxo-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-yl}sulfonyl)benzonitrile
N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-4-methyl-3,4-dihydro-2H-1,4-benzoxazine-7-carboxamide
2-[4-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)phenoxy]ethan-1-amine
(2R,3R)-1'-(3-methoxypyrazin-2-yl)-3-(pyrrolidin-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-[2-(1H-imidazol-2-yl)ethyl]-5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyridin-2-amine
ethyl 3-benzyl-1-[(4-hydroxy-2-methoxyphenyl)methyl]piperidine-3-carboxylate
1-(1-{[5-(4-ethoxyphenyl)furan-2-yl]methyl}piperidin-4-yl)piperidin-4-ol
2-[4-(3,4-dimethoxyphenyl)-1H-1,2,3-triazol-1-yl]-N-methylethane-1-sulfonamide
methyl 2-(cyclopentylsulfamoyl)-6-[(3-fluorophenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(4aR,7aS)-1-cyclobutanecarbonyl-4-[2-(thiophen-3-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-(2-hydroxyethyl)-2-{2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetyl}-2,7-diazaspiro[4.5]decan-6-one
7-[(2-methoxyquinolin-3-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
4-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-N-(pyridin-2-ylmethyl)piperazine-2-carboxamide
1-(4-{[2-chloro-5-methoxy-4-(propan-2-yloxy)phenyl]methyl}piperazin-1-yl)ethan-1-one
N-methyl-N-[2-(pyridin-2-yl)ethyl]-1-[3-(trifluoromethyl)benzoyl]piperidin-3-amine
6-methyl-1-(3-{[4-(pyridin-2-yl)pyrimidin-2-yl]amino}propyl)-1,2-dihydropyridin-2-one
2-[(4-chlorophenyl)methyl]-8-(pyridin-4-yl)-2,8-diazaspiro[4.5]decan-3-one
(3R,4R)-3-cyclobutyl-4-methyl-1-[1-(pyridine-4-carbonyl)piperidin-4-yl]pyrrolidin-3-ol
[(2-cyclohexylpyrimidin-5-yl)methyl](1,4-dioxan-2-ylmethyl)methylamine
2-(5-acetylthiophen-3-yl)-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}acetamide
N-[(2R,3R)-2-(2-methoxyethoxy)-1'-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
1-[1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]-3,5-dimethyl-1H-pyrazole
3-[(dimethylamino)methyl]-1-(3-fluoro-2-methoxybenzoyl)pyrrolidin-3-ol
3-methyl-5-[1-methyl-3-(trifluoromethyl)-1H-pyrazol-5-yl]-1H-1,2,4-triazole
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(oxane-4-carbonyl)piperidine-2-carboxamide
N-{3-[4-(piperazin-1-yl)phenyl]phenyl}acetamide
2-[(3-chlorophenyl)methyl]-N-[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]-1,3-benzoxazole-6-carboxamide
6-[4-(3-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-2,3,4,5-tetrahydropyridazin-3-one
5-chloro-2-methyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}benzamide
N-[3-(4-methoxyphenyl)propyl]-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-[2-methyl-2-(morpholin-4-yl)propyl]pyrrolidin-3-yl]pyrimidin-2-amine
3-(5-benzyl-1,3,4-thiadiazol-2-yl)-1-{[2-(1H-imidazol-1-yl)phenyl]methyl}urea