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N-(2-methylphenyl)-3-oxo-3-[(1S,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]propanamide
3,5-dichloro-N,4-dimethyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]benzamide
3-cyclopropyl-1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]propan-1-one
2,2-dimethylpropyl 7-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-2,7-diazaspiro[4.5]decane-2-carboxylate
1-(1-benzylpiperidin-4-yl)-N-butylpiperidine-3-carboxamide
5-{[3-(4-phenylbenzoyl)piperidin-1-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[(1,4-dimethylpiperazin-2-yl)methyl]-4-hydroxybenzamide
3-[(4-fluoro-3-methoxyphenyl)methyl]-N-[1-(furan-2-yl)ethyl]-9-methoxy-N-methyl-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
(cyclobutylmethyl)({[3-(3-methylbutyl)-1,2,4-oxadiazol-5-yl]methyl})(oxolan-2-ylmethyl)amine
methyl 9-(cyclopentyloxy)-3-[(3-fluoro-4-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[4-(2-carbamoylethyl)-2-(propan-2-yl)phenyl]-2-methylbenzamide
N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
3-{[4-methyl-6-({[3-(pyrazin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}amino)pyrimidin-2-yl]amino}phenol
6-(2-aminoethyl)-N-[2-(dimethylamino)-1-phenylethyl]-2-methylpyrimidin-4-amine
N-(adamantan-2-yl)-3-{5-[methoxy(phenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
1-cyclohexyl-3-(cyclopropylmethyl)-5-(4-fluoropiperidine-1-carbonyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-[(2S,4R)-1-[(2-fluorophenyl)methyl]-4-[(1-methyl-1H-imidazol-2-yl)sulfanyl]pyrrolidine-2-carbonyl]-4-methyl-1,4-diazepane
2-[(4-methoxyphenyl)methyl]-N-(oxolan-3-yl)-1,3-benzoxazole-6-carboxamide
6-[(3R,4S)-3-(2-cyclopentylacetamido)-4-cyclopropylpyrrolidin-1-yl]pyrazine-2-carboxamide
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-2-propylpyridine-4-carboxamide
1-(2-propoxybenzoyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-(5-acetylthiophen-3-yl)-N-[(4-fluorophenyl)methyl]acetamide
(3R,9aR)-8-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}-3-(hydroxymethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
methyl 5-(cyclopentylamino)-3-(furan-2-amido)-1-(3-methylbutyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-(4-{[4-methoxy-3-({1-[2-(trifluoromethyl)benzoyl]piperidin-4-yl}oxy)phenyl]methyl}piperazin-1-yl)ethan-1-one
3-[(3-fluorophenyl)methyl]-N-(naphthalen-1-ylmethyl)-1,2-oxazole-5-carboxamide
3-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]pyridin-2-ol
N-{3-[(4-chlorophenyl)sulfanyl]propyl}-1-ethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
2-({4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}methyl)benzonitrile
N-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-2-(ethylamino)pyrimidine-5-carboxamide
N-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-4,6-dimethyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
1-{5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl}azocane
N-{[1-(2-methoxyethyl)piperidin-3-yl]methyl}-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
N-[(3R,5S)-5-(2,5-dihydro-1H-pyrrole-1-carbonyl)pyrrolidin-3-yl]-2-(4-methoxyphenyl)acetamide
3-(1-butyl-1H-imidazol-2-yl)-1-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]piperidine
3,4,7-trimethyl-N-(2-methylpropyl)-N-(pyridin-2-ylmethyl)-1H-indole-2-carboxamide
4-cyclopentyl-2-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
2-methoxy-4-{[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]methyl}phenol
1-(4-{[3-(2-fluorophenoxy)azetidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
3-{4-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-4-oxobutyl}-3,4-dihydroquinazolin-4-one
2-[1-(3-methoxypropyl)-2,5-dioxo-3-phenylpyrrolidin-3-yl]-N-(2-methylpropyl)acetamide
ethyl 1-(3-{5-[(2,5-dimethoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanoyl)piperidine-3-carboxylate
N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-{[2-(3-phenylpropyl)-1,3-benzoxazol-5-yl]formamido}acetamide
(4aS,7aR)-1-[(3-hydroxyphenyl)methyl]-4-(3-methylbutanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(2,4-dichloro-3-methylphenyl)-2-(2-acetamidoethyl)piperidine-1-carboxamide
(4aS,7aR)-1-(1-aminocyclopropanecarbonyl)-4-benzyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(3-hydroxyphenyl)-1-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
4-(1-{1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]piperidin-4-yl}piperidine-3-carbonyl)morpholine
3-{[(1-acetylpiperidin-3-yl)methyl]sulfamoyl}-N-(2-fluoroethyl)benzamide