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3-(3-chlorobenzoyl)-1-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]piperidine
(1S,4S)-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-3,3-dimethyl-2-methylidenebicyclo[2.2.1]heptane-1-carboxamide
5-(naphthalen-2-ylmethyl)-5-{3-oxo-3-[2-(1,3-thiazol-2-yl)piperidin-1-yl]propyl}pyrrolidin-2-one
2-{1-[(2-ethoxyphenyl)methyl]-4-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperazin-2-yl}ethan-1-ol
1-cyclohexyl-N-methyl-N-[3-(1H-pyrazol-1-yl)propyl]piperidine-4-carboxamide
4-(hydroxymethyl)-1-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}azepan-4-ol
1-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
(2R)-2-[(3-methoxy-5-methylthiophen-2-yl)formamido]-3-methylbutanamide
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylic acid
1-[4-({4-[(2-fluoro-4-methoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazin-1-yl]ethan-1-one
N-[4-(furan-2-yl)phenyl]-1-(5-methyl-1,2-oxazole-4-carbonyl)piperidine-3-carboxamide
(2S)-2-{[2-(2-phenylethyl)-1,3-benzoxazol-5-yl]formamido}propanamide
2-[4-(1-benzofuran-5-carbonyl)piperazin-1-yl]-1,3-benzothiazole
1-[2-({2,7-dimethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)ethyl]imidazolidin-2-one
6,6-dimethyl-1-(4-methylphenyl)-N-(thian-4-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-[(2S,4R)-1-[(3,4-difluorophenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carbonyl]-4-methyl-1,4-diazepane
({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(oxolan-2-ylmethyl){[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}amine
6-(1-methylazepane-2-carbonyl)-1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-6-azaspiro[2.5]octane
[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]({[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl})methylamine
3-[5-(4-propyl-1,2,3-thiadiazol-5-yl)-1,2,4-oxadiazol-3-yl]pyridazine
4-[(5-ethyl-2-methylpyrimidin-4-yl)amino]-N-phenylpiperidine-1-carboxamide
(2S)-2-(3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}propanamido)-4-methylpentanamide
3-(2,3-dihydro-1H-inden-2-yl)-5-[1-(4-methoxybenzoyl)piperidin-4-yl]-5-methylimidazolidine-2,4-dione
N-[(3S,4R)-1-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
N-{[7-chloro-5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-6-methylpyridine-3-carboxamide
ethyl 3-[(3-chlorophenyl)methyl]-1-(5-methylpyrazine-2-carbonyl)piperidine-3-carboxylate
(3R,5S)-1-benzyl-5-[(2,3-dihydro-1H-inden-5-yloxy)methyl]-N-(2-methylpropyl)piperidine-3-carboxamide
5-ethyl-5-{1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]piperidin-4-yl}-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]imidazolidine-2,4-dione
(1S,5R)-3-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{2-[2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydroquinoxalin-2-one
N-methyl-2-(methylamino)-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1,3-thiazole-4-carboxamide
4-(3,4-dimethylbenzoyl)-2-[(3-methoxyphenyl)methyl]morpholine
1-[(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]cyclopropane-1-carboxamide
4-{[2-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]sulfamoyl}-N-(propan-2-yl)benzamide
2-[(5-fluoroquinazolin-4-yl)amino]-1-(furan-2-yl)ethan-1-ol
1-[(2-methyl-1,3-oxazol-4-yl)methyl]-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
ethyl 5-[(5-acetamidothiophen-2-yl)methyl]-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-1-[4-(1H-pyrazol-5-yl)phenyl]piperidin-4-amine
2-[4-(hydroxymethyl)-4-(2-phenoxyethyl)piperidin-1-yl]pyridine-4-carbonitrile
6-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridine-6-carbonyl]-2-(4-fluorophenyl)imidazo[1,2-a]pyridine
3-[(methylsulfanyl)methyl]-5-[(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)methyl]-1,2,4-oxadiazole
8-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{[7-(3,6-dimethylpyrazin-2-yl)-4-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-1,3-dimethyl-1H-pyrazole-5-carboxamide
1-(3-{1-oxa-7-azaspiro[3.5]nonane-7-carbonyl}benzenesulfonyl)pyrrolidin-3-amine
N-{2-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]ethyl}morpholine-2-carboxamide
2-{1-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]piperidin-2-yl}pyridine
N-[(3S,4R)-4-(4-methylphenyl)-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]acetamide
N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
4-{1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)acetyl]piperidin-3-yl}benzoic acid
(3R,4S)-1-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)-4-propylpyrrolidin-3-amine