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N-(4-fluoro-2-methylphenyl)-3-(1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperidin-3-yl)propanamide
N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(thiophen-2-yl)propanamide
(4aS,7aR)-1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-(1-benzothiophen-3-yl)-4-(furan-3-ylmethyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-methyl-5-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyridine
benzyl (1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carboxylate
(2S,4R)-1-[(2-methoxynaphthalen-1-yl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)-N-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxamide
1-(2-{[(2,2-dimethylpropyl)(methyl)amino]methyl}-5-methoxyphenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
{3-benzyl-1-[(6-fluoroquinolin-2-yl)methyl]piperidin-3-yl}methanol
1'-[6-(4H-1,2,4-triazol-4-yl)pyridine-3-carbonyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
5-cyclopropanecarbonyl-1'-(3-methylthiophene-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)but-3-enamide
2-chloro-5-acetamido-N-[4-(pyridin-2-yl)butyl]benzamide
7-methyl-3-(morpholin-4-ylmethyl)-1,2-dihydroquinolin-2-one
8-(3-chloropyridin-2-yl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(pyridin-2-yl)piperazine
1-{4-[(dimethylsulfamoyl)amino]phenyl}-N-[1-(thiophen-3-yl)propan-2-yl]piperidin-4-amine
(3S,4R)-1-(1,3-dihydroxypropan-2-yl)-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
methyl 3-[(3S,4R)-4-(dimethylamino)-1-[(4-methylphenyl)methyl]piperidin-3-yl]propanoate
2-(2-methoxyphenyl)-1-{7-methyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}ethan-1-one
1-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidine-3-carboxamide
4-{[6-chloro-4-(4-methoxypiperidin-1-yl)quinazolin-2-yl]methyl}piperazine-1-carbaldehyde
2-ethyl-5-{[2-(2-phenylethyl)piperidin-1-yl]methyl}pyrimidine
8-methoxy-2-methyl-5-[5-(morpholine-4-carbonyl)-1H-pyrrol-3-yl]quinoline
6-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carbonyl]quinoline
N-[(1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-3-yl)methyl]acetamide
2-methyl-5-[1-(6-methylpyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]pyrazine
1-(2-{methyl[2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}ethyl)piperidin-2-one
3-[2-(azocan-1-yl)-2-oxoethyl]-4-(3-methylbut-2-en-1-yl)piperazin-2-one
N-ethyl-2-{4-[2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carbonyl]piperazin-1-yl}acetamide
N-[1-(4-fluorophenyl)ethyl]-N-methyl-3-(1,2-oxazolidin-2-yl)propanamide
6-(2-methoxybenzoyl)-1-[2-(piperidin-1-yl)ethyl]-3-(pyridin-4-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
methyl 2-(benzylsulfamoyl)-6-(pyrazine-2-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-[3-benzyl-1-(2-methoxyphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]acetamide
5-methoxy-2-{5-propyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-1,3-benzodiazole
1-methyl-1'-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
3-[1-(2-methoxyethyl)-2-methyl-1H-indol-5-yl]-1-[2-(thiophen-2-yl)ethyl]urea
(1-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}-4-(2-phenoxyethyl)piperidin-4-yl)methanol
N-[(2S,4R,6S)-2-benzyl-6-[4-(1H-1,2,4-triazol-1-yl)phenyl]oxan-4-yl]acetamide
2-(2H-1,3-benzodioxol-5-yl)-5-fluoro-1-[1-(thiophen-2-ylmethyl)piperidin-4-yl]-1H-1,3-benzodiazole
N-cyclohexyl-2-(4-ethyl-2,3-dioxopiperazin-1-yl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
ethyl 5-[(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)methyl]-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-[(2S,3S)-1-hydroxy-3-methylpentan-2-yl]-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
N-[(8-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1-oxa-8-azaspiro[4.5]decan-2-yl)methyl]-2-methyl-1,3-thiazole-4-carboxamide
methyl(quinolin-6-ylmethyl)[(3-{[1-(4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]amine
1-[benzyl(methyl)amino]-3-[2-methoxy-5-({[2-(2-methylphenyl)ethyl]amino}methyl)phenoxy]propan-2-ol
1-ethyl-N-[(2-methylphenyl)methyl]-2-oxo-N-(oxolan-2-ylmethyl)-1,2-dihydropyridine-4-carboxamide
4-[4-(azepane-1-carbonyl)piperidin-1-yl]-2-(thiophen-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-({methyl[(4-methylphenyl)methyl]amino}methyl)piperidin-2-one
2-[1-cyclohexyl-5-(6-methoxy-3-methyl-1-benzofuran-2-yl)-1H-1,2,4-triazol-3-yl]acetamide