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2-(1-{3-chloro-6-methylpyrazolo[1,5-a]pyrimidine-2-carbonyl}pyrrolidin-2-yl)pyridine
ethyl 2-[1-(5-chloro-2-oxo-1,2-dihydropyridine-3-carbonyl)piperidin-2-yl]acetate
3-(1H-imidazol-1-yl)-1-[4-(3-methylphenoxy)piperidin-1-yl]butan-1-one
2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)-N-[2-(pyridin-2-yl)ethyl]acetamide
4-(hydroxymethyl)-1-{5-[(4-methylpiperidin-1-yl)methyl]furan-2-carbonyl}azepan-4-ol
(2S)-2-({4-[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}amino)-3-methylbutan-1-ol
N-(3-{[ethyl(pyridin-4-ylmethyl)carbamoyl]amino}-2-methylphenyl)-2-methoxyacetamide
3-[5-(2-fluorophenyl)-4H-1,2,4-triazol-3-yl]-1-methyl-1-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}urea
3-[1-(cyclohex-1-ene-1-carbonyl)piperidin-4-yl]-N-phenylpropanamide
(2S)-1-{[7-methyl-2-(3-methylphenyl)quinolin-3-yl]methyl}pyrrolidine-2-carboxamide
3-[(1S,4S)-2-azabicyclo[2.2.1]heptan-2-yl]-N-(2-ethoxyphenyl)-3-oxopropanamide
N-butyl-1-(6-ethoxy-4-methylquinazolin-2-yl)-N-methylpyrrolidine-2-carboxamide
N-(2-{[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}ethyl)pyridine-3-carboxamide
6-[4-(benzyloxy)piperidin-1-yl]pyrimidin-4-amine
N-[2-ethyl-4-(2,3,4-trimethoxyphenyl)phenyl]acetamide
8-[2-chloro-5-(1H-pyrazol-1-yl)benzoyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(5S,9aS,9bS)-2-methyl-5-[1-(pyridin-3-yl)-1H-pyrrol-2-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-methoxy-6-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-2-amine
ethyl 4-[(2-benzylmorpholin-4-yl)methyl]-1H-pyrazole-3-carboxylate
5-(2-fluorophenyl)-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}pyrazolo[1,5-a]pyrimidin-7-amine
N-{1-[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-4-yl]-2-phenylethyl}-N-methylthiophene-3-carboxamide
1-cyclopentyl-4-{[(1H-imidazol-2-ylmethyl)(methyl)amino]methyl}pyrrolidin-2-one
(2S)-N-[2-ethyl-5-(4H-1,2,4-triazol-4-yl)phenyl]-2-(methoxymethyl)pyrrolidine-1-carboxamide
3-(1,3-benzothiazol-2-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]propanamide
3-[(isoquinolin-5-ylmethyl)[(5-methylthiophen-2-yl)methyl]amino]propan-1-ol
2-(dimethylamino)-2-(2-fluorophenyl)-1-[4-(4-hydroxybutyl)piperazin-1-yl]ethan-1-one
8-(butan-2-yl)-3-(2-methoxyethyl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(8-{[3-(2-hydroxyethoxy)phenyl]methyl}-1-oxa-8-azaspiro[4.5]decan-2-yl)methyl]-2-methyl-1,3-thiazole-4-carboxamide
1-[(5-methylthiophen-2-yl)methyl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
1-(2-{[ethyl(pyridin-4-ylmethyl)amino]methyl}phenoxy)-3-(thiomorpholin-4-yl)propan-2-ol
N-{1-[1-(adamantan-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-2H-1,3-benzodioxole-5-carboxamide
ethyl 4-{[4-(azepan-1-yl)quinazolin-2-yl]methyl}piperazine-1-carboxylate
8-(8-fluoroquinoline-2-carbonyl)-1,3-dioxa-8-azaspiro[4.5]decan-2-one
N,N-dimethyl-4-oxo-4-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}butanamide
N-{3-methyl-1-[7-(naphthalen-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]butyl}furan-2-carboxamide
(1S,5R)-6-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-[4-methoxy-2-(1H-pyrazol-1-yl)phenyl]pyrazine
N-{4-[(1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-6-azaspiro[2.5]octan-6-yl)methyl]phenyl}acetamide
3-{[4-(2,5-dimethylphenyl)piperazin-1-yl]methyl}pyrrolidin-3-ol
N-[2-({2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]acetamide
2-[4-({3-[(3,4-dimethoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperazin-1-yl]-1,3-benzothiazole
methyl 3-(2-ethylbutanoyl)-7-oxo-9-[2-(piperidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)methyl]propanamide
1-(4-methoxyphenyl)-6,6-dimethyl-4-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]piperazin-2-one
2-[3-(3-methoxyphenoxymethyl)piperidine-1-carbonyl]thiophen-3-amine
2-acetyl-8-[(3-chloro-4-hydroxyphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
ethyl({[4-(1H-imidazol-1-yl)phenyl]methyl}){[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N,2,5-trimethyl-1,3-thiazole-4-carboxamide
methyl 4-oxo-4-[2-(2-phenylethyl)morpholin-4-yl]butanoate
N-cyclopentyl-4-[(oxan-4-yl)sulfamoyl]benzamide