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N-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
4-(furan-2-ylmethyl)-N-[4-(oxolan-2-ylmethoxy)phenyl]piperazine-1-carboxamide
1-(2-methoxy-5-{[(2-phenoxyethyl)amino]methyl}phenoxy)-3-(pyrrolidin-1-yl)propan-2-ol
3-(2,2-dimethylpropyl)-5-{spiro[2.3]hexane-1-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
5-{[(1S,4R)-7,7-dimethyl-2-oxobicyclo[2.2.1]heptan-1-yl]methanesulfonyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
N-[3-(1H-pyrazol-1-yl)propyl]-2-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
5-({[6-(methoxymethyl)pyrimidin-4-yl]amino}methyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
(2R,6R)-10-methoxy-4-[(1s,4s)-4-hydroxycyclohexanecarbonyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
(3aR,5S,6S,7aS)-2-[4-methyl-2-(4-methylpiperazin-1-yl)pyrimidine-5-carbonyl]-octahydro-1H-isoindole-5,6-diol
2-[3-cyclopropyl-5-(2,3-dihydro-1,4-benzodioxin-2-yl)-1H-1,2,4-triazol-1-yl]pyridine
3-(2-aminoethyl)-6-ethyl-5-phenyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
4-(1H-indol-5-ylmethyl)-1-(2-methylphenyl)piperazin-2-one
4-{[3-hydroxy-5-(hydroxymethyl)-2-methylpyridin-4-yl]methyl}-1-[(4-methylphenyl)methyl]piperazin-2-one
3-(2-{2-azabicyclo[2.2.1]heptan-2-yl}-2-oxoethyl)-1-(3-methoxypropyl)-3-phenylpyrrolidine-2,5-dione
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1H-pyrazole-3-carbonyl)piperidine
(4aS,7aR)-1-(2-phenoxyethyl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
[(1-cyclopentylpiperidin-4-yl)methyl][(1-ethyl-1H-imidazol-2-yl)methyl](pyridin-3-ylmethyl)amine
1-(7-chloro-3,5-dimethyl-1-benzofuran-2-carbonyl)-4-(pyridin-3-ylmethyl)piperazine
7-[2,2-dimethyl-1-(thiophen-2-yl)cyclopropanecarbonyl]-5H,6H,7H,8H-imidazo[1,5-a]pyrazine
9-methoxy-7-oxo-N-(thiophen-2-ylmethyl)-3-{[2-(trifluoromethyl)phenyl]methyl}-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-{1-[4-(thiomorpholine-4-carbonyl)phenyl]-1H-pyrazol-4-yl}oxolane-3-carboxamide
1-(2-methoxy-5-{[methyl(pyridin-2-ylmethyl)amino]methyl}phenoxy)-3-(4-methyl-1,4-diazepan-1-yl)propan-2-ol
5-[(3S,4S)-3-hydroxy-4-(pyrrolidin-1-yl)pyrrolidine-1-carbonyl]-2-(4-methylphenyl)pyrimidin-4-ol
N,N,2-trimethyl-7-(2-methyl-1H-1,3-benzodiazole-4-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-(1-benzoxepine-4-carbonyl)-4-(3-methylpyridin-4-yl)-1,4-diazepane
3-methyl-N-{1-[1-(quinolin-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}butanamide
1-methanesulfonyl-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-{2-[ethyl(3-methylphenyl)amino]ethyl}acetamide
(cyclobutylmethyl)({[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})(oxolan-2-ylmethyl)amine
5-{6-[(pyridin-4-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-1,3-benzothiazol-2-amine
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-1-benzoxepine-4-carboxamide
2-chloro-4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenol
5-({3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}methyl)-N-methyl-1,2,4-oxadiazole-3-carboxamide
1-{[3-(3-methylpiperidine-1-carbonyl)-1,2-oxazol-5-yl]methyl}piperidin-4-ol
(3-{[1-(5-phenyl-1,3,4-thiadiazol-2-yl)pyrrolidin-3-yl]methyl}phenyl)methanol
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-methyl-1H-pyrazole-4-carboxamide
2-(2-hydroxyethyl)-8-{[4-(pyridin-2-yl)phenyl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
3-(2-methoxyethyl)-1-(4-methoxyphenyl)-5-(1H-pyrazol-3-yl)-1H-1,2,4-triazole
2-{2-[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]-1H-imidazol-1-yl}ethan-1-ol
(2S,4R)-4-(dimethylamino)-1-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}pyrrolidine-2-carboxylic acid
N-benzyl-1-{2-[(2-chlorophenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-(2-hydroxyethyl)piperidine-4-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-{1-[2-(4H-1,2,4-triazol-4-yl)ethyl]piperidin-4-yl}propanamide
3-acetyl-N-[cyclohexyl(thiophen-2-yl)methyl]-1H-pyrazole-5-carboxamide
1-[(1S,4R)-7,7-dimethyl-2-oxobicyclo[2.2.1]heptan-1-yl]-N-({3-methoxy-4-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)methanesulfonamide
N-(2,4-difluorophenyl)-3-{[1-(methoxymethyl)cyclopropyl](methyl)amino}propanamide
2-(1-benzofuran-2-yl)-2-[methyl({[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl})amino]acetic acid
2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(4-ethylphenyl)methyl]-N-methylacetamide
3-(5-methyl-1H-1,2,4-triazol-3-yl)-1-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
N-[2-(4-ethoxyphenyl)ethyl]-2-(morpholin-3-yl)acetamide
3-[(3-chlorophenyl)methyl]-1-(1,3-thiazol-2-yl)piperidine-3-carboxylic acid