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4-[4-({7-[ethoxy(phenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}methyl)phenyl]-2-methylbut-3-yn-2-ol
4-{[(1-ethyl-1H-imidazol-2-yl)methyl]amino}-1-[(4-fluorophenyl)methyl]pyrrolidin-2-one
(1S,6R)-N-(2-phenoxyphenyl)-3,9-diazabicyclo[4.2.1]nonane-9-carboxamide
4-(4-chlorophenyl)-1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-ol
1-[(3-fluorophenyl)methyl]-4-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-2-one
N-[(3S,4R)-1-[(1-ethyl-1H-indol-4-yl)methyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
N-[(2S)-1-hydroxy-3-(1H-indol-3-yl)propan-2-yl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
1-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}-2-propoxyethan-1-one
N-(2,1,3-benzothiadiazol-5-ylmethyl)-3-ethyl-5-hydroxyadamantane-1-carboxamide
(2S,4S)-4-amino-N,N-diethyl-1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]pyrrolidine-2-carboxamide
2-[5-(4-chloro-3-methyl-1H-pyrazol-5-yl)-1-(2,3-dihydro-1H-inden-4-yl)-1H-1,2,4-triazol-3-yl]acetamide
N-{[7-(3,6-dimethylpyrazin-2-yl)-4-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}pyridine-2-carboxamide
2-phenoxy-1-{4-[4-(pyridin-2-yl)pyrimidin-2-yl]piperazin-1-yl}ethan-1-one
N-{[3-methyl-7-(2,4,5-trifluorobenzoyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(methylsulfanyl)benzamide
N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-methoxypropanamide
methyl 2-[N-methyl-1-(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidin-3-yl)formamido]acetate
(1R,5R)-6-(1H-imidazol-2-ylmethyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
4-{[4-benzyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}-5-chloro-2-methoxyphenol
N-methyl-N-[2-(pyridin-2-yl)ethyl]-3-(1-{[2-(trifluoromethyl)phenyl]methyl}piperidin-3-yl)propanamide
5-(2-chloro-4-methoxyphenoxymethyl)-N-(1-phenylcyclopropyl)-1,2-oxazole-3-carboxamide
N-cyclopentyl-N-[(2-methoxyphenyl)methyl]-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
4-(3,6-dimethylpyrazin-2-yl)benzoic acid
N-{2-[3-(4-phenoxybenzoyl)piperidin-1-yl]ethyl}acetamide
3-[3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-6-methylpyridazine
(5-methyl-7-{thieno[3,2-d]pyrimidin-4-yl}-2,3-dihydro-1-benzofuran-2-yl)methanamine
ethyl 5-({2-[4-(2-fluorobenzamido)-1H-pyrazol-1-yl]acetamido}methyl)furan-2-carboxylate
9-[(2-fluoro-4-methoxyphenyl)methyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)[2-(pyridin-3-yloxy)ethyl]amine
4-(2,3-dihydro-1H-inden-2-yl)-3-[2-oxo-2-(pyrrolidin-1-yl)ethyl]piperazin-2-one
1-[2-(phenoxymethyl)-1,3-oxazole-4-carbonyl]-4-(propan-2-yl)piperazine
methyl({[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}){[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}amine
N-cyclobutyl-2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N,2-dimethyl-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]furan-3-carboxamide
3-({[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl](methyl)amino}methyl)-N-(1-methyl-1H-imidazol-2-yl)benzamide
5-(2-methoxyacetamido)-N-[(3-methylphenyl)methyl]-1-(2-phenylethyl)-1H-1,3-benzodiazole-7-carboxamide
1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(phenylsulfanyl)ethan-1-one
1-cyclopentyl-N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-5-oxopyrrolidine-3-carboxamide
(2S)-2-{4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]butanamido}-3-phenylpropanoic acid
methyl 5-(4-{2-[(3-methoxyphenyl)carbamoyl]ethyl}piperidin-1-yl)-5-oxopentanoate
ethyl 4-[(4-chlorophenyl)methyl]-1-[2-(morpholin-4-yl)propanoyl]piperidine-4-carboxylate
2-(1-methyl-1H-pyrrol-3-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}acetamide
5-acetamido-1-ethyl-2-(3-methoxyphenyl)-N-(2,2,2-trifluoroethyl)-1H-1,3-benzodiazole-7-carboxamide
1-cyclopentyl-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-6-oxopiperidine-3-carboxamide
1-[2-(1H-imidazol-4-yl)ethyl]-5-(6-methyl-2H-1,3-benzodioxol-5-yl)-4-phenyl-1H-imidazole
2-(4-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}phenyl)-3H,4H,5H,6H,7H-cyclopenta[d]pyrimidin-4-one
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
1-[2-(phenoxymethyl)-1,3-oxazole-4-carbonyl]-4-(piperidin-1-yl)piperidine
1-butyl-3-[2-(methylsulfanyl)ethyl]-5-(propan-2-yl)-1H-1,2,4-triazole
ethyl 3-[(2-fluorophenyl)methyl]-1-(5-methoxyfuran-2-carbonyl)piperidine-3-carboxylate
2-[4-(6-ethylpyrimidin-4-yl)piperazin-1-yl]-4-(pyridin-3-yl)pyrimidine