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8-{[1-(3-methylbutyl)-1H-1,3-benzodiazol-2-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
[3-(methylsulfanyl)butyl]({[1-(morpholin-4-yl)cycloheptyl]methyl})amine
2-{[1-(3-methoxyphenyl)propan-2-yl]amino}-N-(2-methylphenyl)acetamide
5-(2-fluorophenoxymethyl)-N-(oxolan-2-ylmethyl)-1H-pyrazole-3-carboxamide
1-(2,5-dimethylbenzoyl)-4-[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]piperidine
4-(3-hydroxy-3-methylbutyl)-N-methyl-N-[(7-methyl-1H-1,3-benzodiazol-2-yl)methyl]benzamide
2-(3,5-dimethoxyphenyl)-N-(propan-2-yl)benzamide
1-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-3-(4-fluorophenoxymethyl)piperidine
1-cyclobutanecarbonyl-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}piperidine-4-carboxamide
3-(1-methylpiperidin-2-yl)-N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]propanamide
3-[4-(4-methoxyphenoxy)piperidine-1-carbonyl]benzonitrile
1-[2-(2H-1,3-benzodioxol-5-ylmethyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-benzyl-N-methylpiperidine-4-carboxamide
3-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-9-methoxy-N-[(2-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-(4-fluorophenyl)-2-hydroxy-N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}acetamide
methyl({[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl})(quinolin-5-ylmethyl)amine
1-(4,6-dimethylquinazolin-2-yl)-N-(6-hydroxy-6-methylheptan-2-yl)piperidine-4-carboxamide
N-{[2-(2-ethanesulfonamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
8-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]-2-(propan-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
N-methyl-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-[2-(4-methylphenoxy)ethyl]acetamide
2-acetamido-3-methyl-N-{[5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}butanamide
2-[(3,5-dimethoxyphenyl)methyl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(4-methyl-1H-pyrazol-1-yl)propanamide
2-{3-cyclopentyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}-1H-pyrrole
2-[2-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)phenoxy]propanoic acid
1-(2-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}-2-oxoethyl)-1,2-dihydropyridin-2-one
2-[1-cyclohexyl-4-(quinolin-2-yl)piperazin-2-yl]ethan-1-ol
N-[(3R,4R)-3-hydroxy-1-[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)ethyl]piperidin-4-yl]pyridine-4-carboxamide
2-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}acetamide
N-[1-(4-fluorophenyl)-4-(propan-2-yloxy)-1H-indazol-3-yl]-2-[methyl(propan-2-yl)amino]acetamide
2-(4-chloro-2-{[2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methyl}phenoxy)acetic acid
5-ethyl-N-{[1-(4-methylpiperazin-1-yl)cyclopentyl]methyl}pyrimidin-2-amine
2-(1,3-dioxo-2,3-dihydro-1H-isoindol-2-yl)-N-{[8-(pyridine-4-carbonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}acetamide
3-{imidazo[1,2-a]pyridin-2-yl}-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]propanamide
4-(1-benzofuran-2-yl)-2-[5-cyclopropyl-4-(4-ethylpiperazine-1-carbonyl)-1H-pyrazol-1-yl]pyrimidine
4-(5-acetyl-4-methylpyrimidin-2-yl)-1-cyclopentylpiperazin-2-one
(3aS,6aS)-2-cyclohexyl-5-[(3-methylpyridin-4-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(2-methoxy-2-phenylacetyl)-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
1-{[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl}-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
5-fluoro-N-[1-(pyridin-4-yl)propan-2-yl]-4-(pyrrolidin-1-yl)pyrimidin-2-amine
1-(2-methoxypyridine-4-carbonyl)-N-(pyridin-2-ylmethyl)piperazine-2-carboxamide
N-methyl-N-{2-[4-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)phenoxy]ethyl}-2-(trifluoromethyl)benzamide
(4S,4aS,8aS)-1-(1H-1,3-benzodiazole-5-carbonyl)-4-phenyl-decahydroquinolin-4-ol
8-(5-acetyl-2,4-dimethyl-1H-pyrrole-3-carbonyl)-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methoxyethyl)-8-[(3-methylquinoxalin-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2S)-3-(1H-indol-3-yl)-2-[3-(1,2-oxazinan-2-yl)propanamido]propanoic acid
2-({4-[1-(2-methoxyethyl)pyrrolidine-3-carbonyl]piperazin-1-yl}methyl)benzonitrile
1-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(3-fluorobenzoyl)pyrrolidin-3-yl]methanol
4-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)-1-[(5-methylfuran-2-yl)methyl]piperidine
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-3-(piperazine-1-carbonyl)benzene-1-sulfonamide