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3-[(3R,4S)-3-(2-carboxyethyl)-4-(4-methylpiperazin-1-yl)piperidine-1-carbonyl]benzoic acid
N-[2-(cyclohex-1-en-1-yl)ethyl]-6-{[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
4-(4-methoxyphenoxymethyl)-1-(1,3-thiazol-4-ylmethyl)piperidine
4-(cyclopropylmethyl)-2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-methyl-2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}-N-[(3-methylpyridin-4-yl)methyl]acetamide
5-(2-{[(3-fluorophenyl)methyl]amino}ethyl)-1-[2-(2-methoxyphenyl)ethyl]pyrrolidin-2-one
1-[3-(3-methylphenoxy)azetidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
3-[4-hydroxy-4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-N-(2-methylphenyl)-3-oxopropanamide
3-fluoro-N-(1-{1-[2-(3-methylphenyl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
9-methoxy-3-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-7-oxo-N-[3-(1H-pyrazol-1-yl)propyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-methyl-4-(4-{[2-(pyridin-3-yl)morpholin-4-yl]methyl}phenyl)butan-2-ol
4-{3-oxo-3-[4-(propan-2-yl)piperazin-1-yl]propyl}-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
4-cyclobutaneamido-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]benzamide
4-benzyl-3-ethyl-1-[(5-ethylpyridin-2-yl)methyl]-1,4-diazepan-5-one
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-(morpholin-4-yl)butanamide
2-methyl-5-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrazine
N-{[1-(hydroxymethyl)cyclopentyl]methyl}-N-methyl-2-(pyridin-4-yl)acetamide
N-({7-[3-(furan-2-yl)benzoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)cyclopropanecarboxamide
(4aS,7aR)-1-(3-chloro-4-hydroxybenzoyl)-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N,N-dimethyl-1-(prop-2-en-1-yl)-5-({[4-(trifluoromethyl)phenyl]methyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
8-methoxy-N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(3-{5-[2-(methylsulfanyl)ethyl]-1,2,4-oxadiazol-3-yl}phenyl)methanol
4-{6-[(3-fluorophenyl)methoxy]-3-oxo-4-(2-phenylethyl)-1,4-diazepane-1-carbonyl}pyridin-1-ium-1-olate
N-(1-{7-[(2-fluoro-5-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)pyridine-3-carboxamide
1-(5-fluoro-2-methoxybenzoyl)-3-(2-methoxyethyl)piperidine-3-carboxylic acid
1-[5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-yl]azocane
(2E)-1-[7-(5-chloropyridin-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(thiophen-2-yl)prop-2-en-1-one
2-[(5-methylpyrazin-2-yl)methyl]-8-(pyridin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
1-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
3-{2,8-diazaspiro[4.5]decan-2-ylmethyl}-3-hydroxy-1-(2-phenylethyl)piperidin-2-one
1-(2-aminoethyl)-N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
4-{[4-(3-hydroxy-3-methylbutyl)phenyl]formamido}-N,4-dimethylpentanamide
N-{[3-methyl-7-(4-phenylbutanoyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}propane-1-sulfonamide
2-chloro-N-{[1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]methyl}benzamide
1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-3-propoxypiperidine
5-{4-[(4-cyanopiperidin-1-yl)methyl]phenoxymethyl}furan-2-carboxylic acid
3-[3-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
1-{3-chloro-6-methylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-4-(hydroxymethyl)piperidin-4-ol
N-({3-methyl-7-[3-(1H-pyrazol-1-yl)benzoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-3-carboxamide
3-(2,3-dihydro-1H-isoindole-2-sulfonyl)-N,N-dipropylbenzamide
4-methyl-5-({2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)pentane-1,4-diol
2-(3-{[ethyl({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)amino]methyl}phenoxy)ethan-1-ol
8-chloro-N-[(1S,2R)-1-hydroxy-1-(4-hydroxyphenyl)propan-2-yl]-2-methylquinoline-4-carboxamide
5-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]-2-(methylsulfanyl)pyrimidine
2-(ethanesulfonyl)-1-(2-methoxyethyl)-5-({1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}methyl)-1H-imidazole
3-(2-chloro-4-fluorophenyl)-5-methoxypyridine
3-{[5-(2,6-dimethoxyphenyl)-1,2,4-triazin-3-yl](methyl)amino}-1-phenylpropan-1-ol
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-3-(piperidin-4-ylmethyl)benzamide
2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N,N-bis(prop-2-en-1-yl)acetamide
1-{8-methyl-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one